NO20051036L - 3,4-disubstituerte syklobuten-1,2-dioner som CXC-kjemokinreseptorligander - Google Patents

3,4-disubstituerte syklobuten-1,2-dioner som CXC-kjemokinreseptorligander

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Publication number
NO20051036L
NO20051036L NO20051036A NO20051036A NO20051036L NO 20051036 L NO20051036 L NO 20051036L NO 20051036 A NO20051036 A NO 20051036A NO 20051036 A NO20051036 A NO 20051036A NO 20051036 L NO20051036 L NO 20051036L
Authority
NO
Norway
Prior art keywords
dione
chemokine receptor
receptor ligands
cxc chemokine
cyclobutene
Prior art date
Application number
NO20051036A
Other languages
English (en)
Inventor
Daniel J Lundell
Arthur G Taveras
Jianping Chao
Cynthia J Aki
Michael Dwyer
J Robert Merritt
Jianhua Chao
Younong Yu
James Jakway
Jay S Fine
Purakkattle Biju
Gaifa Lai
Minglang Wu
Evan A Hecker
Original Assignee
Pharmacopeia Drug Discovery
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=31190690&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20051036(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from US10/208,412 external-priority patent/US20040097547A1/en
Application filed by Pharmacopeia Drug Discovery filed Critical Pharmacopeia Drug Discovery
Publication of NO20051036L publication Critical patent/NO20051036L/no

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    • C07C237/30—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a non-condensed six-membered aromatic ring of the carbon skeleton having the nitrogen atom of the carboxamide group bound to hydrogen atoms or to acyclic carbon atoms
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Abstract

Det er beskrevet nye forbindelser med formel (I) eller et farmasøytisk akseptabelt salt eller solvat derav. Det er også beskrevet behandlingen av kjemokinmedierte sykdommer ved å anvende forbindelser med formel (II)
NO20051036A 2002-07-30 2005-02-25 3,4-disubstituerte syklobuten-1,2-dioner som CXC-kjemokinreseptorligander NO20051036L (no)

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US10/208,412 US20040097547A1 (en) 2001-04-16 2002-07-30 3,4-Di-substituted cyclobutene-1,2-diones as CXC-chemokine receptor ligands
US10/241,326 US20040106794A1 (en) 2001-04-16 2002-09-11 3,4-Di-substituted cyclobutene-1,2-diones as CXC-chemokine receptor ligands
PCT/US2003/023785 WO2004011418A1 (en) 2002-07-30 2003-07-30 3,4-di-substituted cyclobutene-1, 2-diones as cxc-chemokine receptor ligands

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US20070021494A1 (en) 2007-01-25
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US7947720B2 (en) 2011-05-24
US20090306079A1 (en) 2009-12-10
BR0313109A (pt) 2005-06-21
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US20040106794A1 (en) 2004-06-03
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