NO20032187L - Heterocyklylalkylpiperidinderivater, deres fremstilling samt preparater inneholdende forbindelsene - Google Patents

Heterocyklylalkylpiperidinderivater, deres fremstilling samt preparater inneholdende forbindelsene

Info

Publication number
NO20032187L
NO20032187L NO20032187A NO20032187A NO20032187L NO 20032187 L NO20032187 L NO 20032187L NO 20032187 A NO20032187 A NO 20032187A NO 20032187 A NO20032187 A NO 20032187A NO 20032187 L NO20032187 L NO 20032187L
Authority
NO
Norway
Prior art keywords
compounds
preparation
preparations containing
heterocyclylalkylpiperidine derivatives
heterocyclylalkylpiperidine
Prior art date
Application number
NO20032187A
Other languages
English (en)
Other versions
NO20032187D0 (no
Inventor
Eric Bacque
Jean-Christophe Carry
Youssef El-Ahmad
Michel Evers
Philippe Hubert
Jean-Luc Malleron
Serge Mignani
Guy Pantel
Michel Tabart
Fabrice Viviani
Original Assignee
Aventis Pharma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa
Publication of NO20032187D0 publication Critical patent/NO20032187D0/no
Publication of NO20032187L publication Critical patent/NO20032187L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/20—Oxygen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
NO20032187A 2000-11-15 2003-05-14 Heterocyklylalkylpiperidinderivater, deres fremstilling samt preparater inneholdende forbindelsene NO20032187L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0014738A FR2816618B1 (fr) 2000-11-15 2000-11-15 Derives heterocyclylalcoyl piperidine, leur preparation et les compositions qui les contiennent
PCT/FR2001/003559 WO2002040474A2 (fr) 2000-11-15 2001-11-14 Derives heterocyclylalcoyl piperidine et leur application comme antimicrobiens

Publications (2)

Publication Number Publication Date
NO20032187D0 NO20032187D0 (no) 2003-05-14
NO20032187L true NO20032187L (no) 2003-06-26

Family

ID=8856503

Family Applications (2)

Application Number Title Priority Date Filing Date
NO20032187A NO20032187L (no) 2000-11-15 2003-05-14 Heterocyklylalkylpiperidinderivater, deres fremstilling samt preparater inneholdende forbindelsene
NO20072142A NO20072142L (no) 2000-11-15 2007-04-25 Mellomprodukter for fremstilling av heterocyklylalkylpiperidinderivater og forbindelser for fremstilling av disse

Family Applications After (1)

Application Number Title Priority Date Filing Date
NO20072142A NO20072142L (no) 2000-11-15 2007-04-25 Mellomprodukter for fremstilling av heterocyklylalkylpiperidinderivater og forbindelser for fremstilling av disse

Country Status (28)

Country Link
EP (2) EP1337529B1 (no)
JP (1) JP2004514661A (no)
KR (1) KR100849608B1 (no)
CN (1) CN1483031A (no)
AR (1) AR034006A1 (no)
AT (1) ATE337311T1 (no)
AU (2) AU1836502A (no)
BG (1) BG107793A (no)
BR (1) BR0115312A (no)
CA (1) CA2429311A1 (no)
CZ (1) CZ20031316A3 (no)
DE (1) DE60122567T2 (no)
DK (1) DK1337529T3 (no)
EA (1) EA200300568A1 (no)
EE (1) EE200300207A (no)
ES (1) ES2271119T3 (no)
FR (1) FR2816618B1 (no)
HR (1) HRP20030379A2 (no)
HU (1) HUP0303758A3 (no)
IL (1) IL155841A0 (no)
NO (2) NO20032187L (no)
PL (1) PL363004A1 (no)
PT (1) PT1337529E (no)
SK (1) SK5822003A3 (no)
TN (1) TNSN01160A1 (no)
WO (1) WO2002040474A2 (no)
YU (1) YU46803A (no)
ZA (1) ZA200303794B (no)

Families Citing this family (37)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2001289749B9 (en) 2000-07-26 2004-08-19 Smithkline Beecham P.L.C. Aminopiperidine quinolines and their azaisosteric analogues with antibacterial activity
GB0101577D0 (en) 2001-01-22 2001-03-07 Smithkline Beecham Plc Compounds
GB0112834D0 (en) 2001-05-25 2001-07-18 Smithkline Beecham Plc Medicaments
GB0112836D0 (en) 2001-05-25 2001-07-18 Smithkline Beecham Plc Medicaments
GB0118238D0 (en) * 2001-07-26 2001-09-19 Smithkline Beecham Plc Medicaments
JP4445753B2 (ja) 2002-01-29 2010-04-07 グラクソ グループ リミテッド アミノピペリジン誘導体
AU2003239302A1 (en) 2002-01-29 2003-09-02 Glaxo Group Limited Aminopiperidine compounds, process for their preparation, and pharmaceutical compositions containing them
TW200409637A (en) 2002-06-26 2004-06-16 Glaxo Group Ltd Compounds
AR040335A1 (es) 2002-06-26 2005-03-30 Glaxo Group Ltd Compuesto de ciclohexano o ciclohexeno, uso del mismo para preparar un medicamento, composicion farmaceutica que lo comprende, procedimiento y compuestos intermediarios de utilidad para preparar dicho compuesto
FR2842807A1 (fr) * 2002-07-23 2004-01-30 Aventis Pharma Sa Derives de la quinolyl propyl piperidine, procede et intermediaires de preparation et compositions les renfermant
GB0217294D0 (en) * 2002-07-25 2002-09-04 Glaxo Group Ltd Medicaments
FR2844270B1 (fr) 2002-09-11 2006-05-19 Aventis Pharma Sa Derives de la quinolyl propyl piperidine, leur procede et intermediaires de preparation et les compositions qui les contiennent
FR2844268B1 (fr) * 2002-09-11 2004-10-22 Aventis Pharma Sa Derives de la quinolyl propyl piperidine, leurs procedes et intermediaires de preparation et les compositions qui les contiennent
DE10256405A1 (de) * 2002-12-02 2004-06-17 Morphochem Aktiengesellschaft für kombinatorische Chemie Neue Verbindungen, die Topoisomerase IV inhibieren
ATE461928T1 (de) 2002-11-05 2010-04-15 Glaxosmithkline Llc Antibakterielle wirkstoffe
US7491714B2 (en) 2002-12-04 2009-02-17 Glaxo Group Limited Quinolines and nitrogenated derivatives thereof and their use as antibacterial agents
FR2852954B1 (fr) * 2003-03-28 2006-07-14 Aventis Pharma Sa Derives de quinoleines-4-substituees, leurs procede et intermediaires de preparation et les compositions pharmaceutiques qui les contiennent
US7232833B2 (en) 2003-03-28 2007-06-19 Novexel 4-substituted quinoline derivatives, method and intermediates for their preparation and pharmaceutical compositions containing them
FR2862301B1 (fr) * 2003-11-17 2007-12-21 Aventis Pharma Sa Nouveau procede de preparation de quinoleines 3-fluorees
FR2867472B1 (fr) * 2004-03-12 2008-07-18 Aventis Pharma Sa Derives de quinoleines-4-substituees, leurs procede et intermediaires de preparation et les compositions pharmaceutiques qui les contiennent
EP1846417A4 (en) 2005-01-25 2009-12-23 Glaxo Group Ltd ANTIBACTERIAL ACTIVE SUBSTANCES
US7592334B2 (en) 2005-01-25 2009-09-22 Glaxo Group Limited Antibacterial agents
US7648980B2 (en) 2005-01-25 2010-01-19 Glaxo Group Limited Antibacterial agents
WO2006081179A1 (en) 2005-01-25 2006-08-03 Glaxo Group Limited Antibacterial agents
US7700595B2 (en) 2005-03-01 2010-04-20 Wyeth Llc Cinnoline compounds
MY150958A (en) 2005-06-16 2014-03-31 Astrazeneca Ab Compounds for the treatment of multi-drug resistant bacterial infections
EP1981881B1 (en) 2006-01-26 2011-12-07 Actelion Pharmaceuticals Ltd. Tetrahydropyrane antibiotics
DE602007009205D1 (de) 2006-04-06 2010-10-28 Glaxo Group Ltd Pyrrolochinoxalinonderivate als antibakterielle mittel
EP1992628A1 (en) 2007-05-18 2008-11-19 Glaxo Group Limited Derivatives and analogs of N-ethylquinolones and N-ethylazaquinolones
BRPI0812942B1 (pt) 2007-06-15 2018-11-21 Actelion Pharmaceuticals Ltd composto derivado de 3-amino-6 - (1-amino-etil) - tetra-hidropirano, composição farmacêutica e uso de referido composto.
EP2080761A1 (en) 2008-01-18 2009-07-22 Glaxo Group Limited Compounds
WO2010043714A1 (en) 2008-10-17 2010-04-22 Glaxo Group Limited Tricyclic nitrogen compounds used as antibacterials
US8318940B2 (en) 2009-01-15 2012-11-27 Glaxo Group Limited Naphthyridin-2 (1 H)-one compounds useful as antibacterials
IN2015KN00323A (no) * 2012-08-15 2015-07-10 Glaxo Group Ltd
TW201618779A (zh) 2014-08-22 2016-06-01 葛蘭素史克智慧財產發展有限公司 方法
WO2016138988A1 (en) * 2015-03-02 2016-09-09 University Of Copenhagen Piperazine inhibitors of bacterial gyrase and topoisomerase iv
TW201722965A (zh) 2015-08-16 2017-07-01 葛蘭素史密斯克藍智慧財產發展有限公司 用於抗菌應用之化合物

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL7908031A (nl) 1979-11-01 1981-06-01 Acf Chemiefarma Nv Nieuwe chinolinederivaten en farmaceutische preparaten die een dergelijke verbinding bevatten, alsmede werk- wijze voor het bereiden van deze verbindingen.
JPH0239546A (ja) 1988-07-29 1990-02-08 Origin Electric Co Ltd 混成集積回路の製造方法
NZ232091A (en) 1989-01-16 1990-12-21 Bellon Labor Sa Roger 7-fluoro-8-(piperazin-1-yl)-4-oxo-1,4-dihydro-benzo(b)(1,8)naphthyridine-3-carboxylic acid derivatives, preparation and pharmaceutical compositions thereof
JP2002501061A (ja) * 1998-01-26 2002-01-15 スミスクライン・ビーチャム・パブリック・リミテッド・カンパニー 抗菌剤用キノリン誘導体
AU2437900A (en) * 1999-01-20 2000-08-07 Smithkline Beecham Plc Piperidinylquinolines as protein tyrosine kinase inhibitors
FR2852954B1 (fr) * 2003-03-28 2006-07-14 Aventis Pharma Sa Derives de quinoleines-4-substituees, leurs procede et intermediaires de preparation et les compositions pharmaceutiques qui les contiennent

Also Published As

Publication number Publication date
NO20032187D0 (no) 2003-05-14
AU2002218365B2 (en) 2007-07-05
HUP0303758A2 (hu) 2004-03-01
KR100849608B1 (ko) 2008-07-31
EP1337529B1 (fr) 2006-08-23
AU1836502A (en) 2002-05-27
EP1695964A1 (fr) 2006-08-30
FR2816618B1 (fr) 2002-12-27
EA200300568A1 (ru) 2003-12-25
DK1337529T3 (da) 2006-12-18
NO20072142L (no) 2007-04-25
WO2002040474A2 (fr) 2002-05-23
ZA200303794B (en) 2004-06-29
CN1483031A (zh) 2004-03-17
ATE337311T1 (de) 2006-09-15
ES2271119T3 (es) 2007-04-16
YU46803A (sh) 2006-05-25
KR20030060934A (ko) 2003-07-16
DE60122567T2 (de) 2007-08-23
DE60122567D1 (de) 2006-10-05
PL363004A1 (en) 2004-11-15
IL155841A0 (en) 2003-12-23
BG107793A (bg) 2004-08-31
BR0115312A (pt) 2003-09-23
EE200300207A (et) 2003-08-15
WO2002040474A3 (fr) 2002-10-31
AR034006A1 (es) 2004-01-21
PT1337529E (pt) 2006-12-29
EP1337529A2 (fr) 2003-08-27
TNSN01160A1 (fr) 2005-11-10
CA2429311A1 (en) 2002-05-23
JP2004514661A (ja) 2004-05-20
FR2816618A1 (fr) 2002-05-17
SK5822003A3 (en) 2004-06-08
HUP0303758A3 (en) 2009-08-28
HRP20030379A2 (en) 2005-04-30
CZ20031316A3 (cs) 2003-10-15

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