DE602007009205D1 - Pyrrolochinoxalinonderivate als antibakterielle mittel - Google Patents

Pyrrolochinoxalinonderivate als antibakterielle mittel

Info

Publication number
DE602007009205D1
DE602007009205D1 DE602007009205T DE602007009205T DE602007009205D1 DE 602007009205 D1 DE602007009205 D1 DE 602007009205D1 DE 602007009205 T DE602007009205 T DE 602007009205T DE 602007009205 T DE602007009205 T DE 602007009205T DE 602007009205 D1 DE602007009205 D1 DE 602007009205D1
Authority
DE
Germany
Prior art keywords
pyrrolochinoxalinone
derivatives
antibacterial agents
antibacterial
agents
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
DE602007009205T
Other languages
English (en)
Inventor
Graham Elgin Jones
Timothy James Miles
Neil David Pearson
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Glaxo Group Ltd
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0606970A external-priority patent/GB0606970D0/en
Priority claimed from GB0706023A external-priority patent/GB0706023D0/en
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of DE602007009205D1 publication Critical patent/DE602007009205D1/de
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/06—Peri-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DE602007009205T 2006-04-06 2007-03-29 Pyrrolochinoxalinonderivate als antibakterielle mittel Active DE602007009205D1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0606970A GB0606970D0 (en) 2006-04-06 2006-04-06 Compounds
GB0706023A GB0706023D0 (en) 2007-03-26 2007-03-26 Compounds
PCT/EP2007/053056 WO2007115947A1 (en) 2006-04-06 2007-03-29 Pyrrolo-quinoxalinone derivatives as antibacterials

Publications (1)

Publication Number Publication Date
DE602007009205D1 true DE602007009205D1 (de) 2010-10-28

Family

ID=38580721

Family Applications (1)

Application Number Title Priority Date Filing Date
DE602007009205T Active DE602007009205D1 (de) 2006-04-06 2007-03-29 Pyrrolochinoxalinonderivate als antibakterielle mittel

Country Status (9)

Country Link
US (1) US7709483B2 (de)
EP (1) EP2001887B1 (de)
JP (1) JP2009532423A (de)
AR (1) AR060287A1 (de)
AT (1) ATE481406T1 (de)
DE (1) DE602007009205D1 (de)
PE (1) PE20080182A1 (de)
TW (1) TW200815450A (de)
WO (1) WO2007115947A1 (de)

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CA2626641A1 (en) * 2005-10-21 2007-07-19 Glaxo Group Limited Compounds
US20070185153A1 (en) 2005-12-22 2007-08-09 Nathalie Cailleau Compounds
GB0608263D0 (en) 2006-04-26 2006-06-07 Glaxo Group Ltd Compounds
GB0613208D0 (en) * 2006-07-03 2006-08-09 Glaxo Group Ltd Compounds
DE602008002912D1 (de) * 2007-04-20 2010-11-18 Glaxo Group Ltd Tricyclische stickstoffhaltige verbindungen als antibakterielle wirkstoffe
CN101874032B (zh) * 2007-11-26 2013-02-06 富山化学工业株式会社 二氮杂萘衍生物一水合物及其制备方法
EP2080761A1 (de) 2008-01-18 2009-07-22 Glaxo Group Limited Verbindungen
US8349828B2 (en) 2008-02-20 2013-01-08 Actelion Pharmaceuticals Ltd. Azatricyclic antibiotic compounds
KR20110016947A (ko) 2008-05-23 2011-02-18 글락소 그룹 리미티드 트리시클릭 질소 함유 화합물 및 항박테리아제로서의 그의 용도
EP2300477A1 (de) * 2008-05-23 2011-03-30 Glaxo Group Limited Tricyclische, stickstoffhaltige verbindungen und ihre verwendung als antibakterielle mittel
RU2530884C2 (ru) 2008-10-07 2014-10-20 Актелион Фармасьютиклз Лтд Трициклические оксазолидиноновые антибиотические соединения
JP2012505866A (ja) 2008-10-17 2012-03-08 グラクソ グループ リミテッド 抗菌剤として使用される三環式窒素化合物
NZ593891A (en) 2008-12-12 2013-05-31 Actelion Pharmaceuticals Ltd 5-amino-2-(1-hydroxy-ethyl)-tetrahydropyran derivatives
WO2010081874A1 (en) 2009-01-15 2010-07-22 Glaxo Group Limited Naphthyridin-2 (1 h)-one compounds useful as antibacterials
CN101870653B (zh) * 2009-04-23 2013-07-10 上海合全药业有限公司 一种2-甲基-3-氟-6-硝基苯甲酸的合成方法
SG11201700566SA (en) 2014-08-22 2017-03-30 Glaxosmithkline Ip Dev Ltd Tricyclic nitrogen containing compounds for treating neisseria gonorrhoea infection
CN111655690B (zh) 2017-11-24 2023-01-10 詹森药业有限公司 吡唑并吡啶酮化合物

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WO2004104000A1 (ja) 2003-05-23 2004-12-02 Japan Tobacco Inc. トリサイクリック縮合環化合物およびその医薬用途
FR2858619B1 (fr) 2003-08-08 2006-12-22 Aventis Pharma Sa Derives de quinoleines-4-substituees, leurs procede et intermediaires de preparation et les compositions pharmaceutiques qui les contiennent
FR2867472B1 (fr) 2004-03-12 2008-07-18 Aventis Pharma Sa Derives de quinoleines-4-substituees, leurs procede et intermediaires de preparation et les compositions pharmaceutiques qui les contiennent
WO2006002047A2 (en) 2004-06-15 2006-01-05 Glaxo Group Limited Antibacterial agents
FR2872164B1 (fr) 2004-06-29 2006-11-17 Aventis Pharma Sa Derives de quinoleines-4-substituees, leur procede et intermediaires de preparation et les compositions pharmaceutiques qui les contiennent
EP1773831A1 (de) 2004-07-08 2007-04-18 Glaxo Group Limited Antibakterielle mittel
US20080194547A1 (en) 2004-07-09 2008-08-14 Glaxo Group Limited Antibacterial Agents
JP2008506695A (ja) 2004-07-13 2008-03-06 グラクソ　グループ　リミテッド 抗細菌剤
JP2008507543A (ja) 2004-07-22 2008-03-13 グラクソ　グループ　リミテッド 抗細菌剤
WO2006017468A2 (en) 2004-08-02 2006-02-16 Glaxo Group Limited Antibacterial agents
JP2008509222A (ja) 2004-08-09 2008-03-27 グラクソ グループ リミテッド 抗菌剤
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EP1845995A4 (de) 2005-01-25 2010-03-03 Glaxo Group Ltd Antibakterielle wirkstoffe
JP2008528604A (ja) 2005-01-25 2008-07-31 グラクソ グループ リミテッド 抗菌剤
WO2006081182A2 (en) 2005-01-25 2006-08-03 Glaxo Group Limited Antibacterial agents
JP2008528586A (ja) 2005-01-25 2008-07-31 グラクソ グループ リミテッド 抗菌剤
US7605169B2 (en) 2005-01-25 2009-10-20 Glaxo Group Limited Antibacterial agents
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CA2626641A1 (en) 2005-10-21 2007-07-19 Glaxo Group Limited Compounds
US20070185153A1 (en) 2005-12-22 2007-08-09 Nathalie Cailleau Compounds
GB0608263D0 (en) 2006-04-26 2006-06-07 Glaxo Group Ltd Compounds
GB0613208D0 (en) 2006-07-03 2006-08-09 Glaxo Group Ltd Compounds
GB0705672D0 (en) 2007-03-23 2007-05-02 Glaxo Group Ltd Compounds

Also Published As

Publication number Publication date
US20090062265A1 (en) 2009-03-05
AR060287A1 (es) 2008-06-04
WO2007115947A1 (en) 2007-10-18
EP2001887A1 (de) 2008-12-17
EP2001887B1 (de) 2010-09-15
ATE481406T1 (de) 2010-10-15
PE20080182A1 (es) 2008-05-01
JP2009532423A (ja) 2009-09-10
US7709483B2 (en) 2010-05-04
TW200815450A (en) 2008-04-01

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