NO20014792L - Med sukkerrester substituerte 1,4-benzotiazepin-1,1-dioksid- derivater, fremgangsmåte for deres fremstilling, legemidler sominneholder disse og forbindelser og deres anvendelse - Google Patents

Med sukkerrester substituerte 1,4-benzotiazepin-1,1-dioksid- derivater, fremgangsmåte for deres fremstilling, legemidler sominneholder disse og forbindelser og deres anvendelse

Info

Publication number
NO20014792L
NO20014792L NO20014792A NO20014792A NO20014792L NO 20014792 L NO20014792 L NO 20014792L NO 20014792 A NO20014792 A NO 20014792A NO 20014792 A NO20014792 A NO 20014792A NO 20014792 L NO20014792 L NO 20014792L
Authority
NO
Norway
Prior art keywords
benzothiazepine
compounds
preparation
sugar residues
drugs containing
Prior art date
Application number
NO20014792A
Other languages
English (en)
Other versions
NO319836B1 (no
NO20014792D0 (no
Inventor
Wendelin Frick
Heiner Glombik
Hubert Heuer
Hans-Ludwig Schaefer
Original Assignee
Aventis Pharma Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Gmbh filed Critical Aventis Pharma Gmbh
Publication of NO20014792L publication Critical patent/NO20014792L/no
Publication of NO20014792D0 publication Critical patent/NO20014792D0/no
Publication of NO319836B1 publication Critical patent/NO319836B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D281/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D281/02—Seven-membered rings
    • C07D281/04—Seven-membered rings having the hetero atoms in positions 1 and 4
    • C07D281/08—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D281/10—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/554—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one sulfur as ring hetero atoms, e.g. clothiapine, diltiazem
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Obesity (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
NO20014792A 1999-04-09 2001-10-02 Med sukkerrester substituerte 1,4-benzotiazepin-1,1-dioksid-derivater, fremgangsmate for deres fremstilling, legemidler som inneholder disse og forbindelser og deres anvendelse NO319836B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19916108A DE19916108C1 (de) 1999-04-09 1999-04-09 Mit Zuckerresten substituierte 1,4-Benzothiazepin-1,1-dioxidderivate, Verfahren zu deren Herstellung und deren Verwendung
PCT/EP2000/002570 WO2000061568A2 (de) 1999-04-09 2000-03-23 Mit zuckerresten substituierte 1,4-benzothiazepin-1,1-dioxidderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung

Publications (3)

Publication Number Publication Date
NO20014792L true NO20014792L (no) 2001-10-02
NO20014792D0 NO20014792D0 (no) 2001-10-02
NO319836B1 NO319836B1 (no) 2005-09-19

Family

ID=7904060

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20014792A NO319836B1 (no) 1999-04-09 2001-10-02 Med sukkerrester substituerte 1,4-benzotiazepin-1,1-dioksid-derivater, fremgangsmate for deres fremstilling, legemidler som inneholder disse og forbindelser og deres anvendelse

Country Status (32)

Country Link
US (1) US6277831B1 (no)
EP (1) EP1169313B1 (no)
JP (1) JP2002541248A (no)
KR (1) KR100686905B1 (no)
CN (1) CN1145619C (no)
AR (1) AR023401A1 (no)
AT (1) ATE243686T1 (no)
AU (1) AU765199B2 (no)
BR (1) BR0009641A (no)
CA (1) CA2369070C (no)
CZ (1) CZ300410B6 (no)
DE (2) DE19916108C1 (no)
DK (1) DK1169313T3 (no)
EE (1) EE04613B1 (no)
ES (1) ES2200860T3 (no)
HK (1) HK1044537B (no)
HR (1) HRP20010725A2 (no)
HU (1) HUP0200644A3 (no)
IL (2) IL145647A0 (no)
MY (1) MY120842A (no)
NO (1) NO319836B1 (no)
NZ (1) NZ514656A (no)
PL (1) PL203806B1 (no)
PT (1) PT1169313E (no)
RS (1) RS49850B (no)
RU (1) RU2232155C2 (no)
SI (1) SI1169313T1 (no)
SK (1) SK286744B6 (no)
TR (1) TR200102910T2 (no)
TW (1) TWI254045B (no)
WO (1) WO2000061568A2 (no)
ZA (1) ZA200107989B (no)

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JP2023504643A (ja) 2019-12-04 2023-02-06 アルビレオ・アクチボラグ ベンゾチア（ジ）アゼピン化合物及び胆汁酸モジュレータとしてのそれらの使用
PE20230234A1 (es) 2019-12-04 2023-02-07 Albireo Ab Compuestos de benzoti(di)azepina y su uso como moduladores del acido biliar
JP2023504644A (ja) 2019-12-04 2023-02-06 アルビレオ・アクチボラグ ベンゾチアジアゼピン化合物及び胆汁酸モジュレータとしてのそれらの使用
AR120683A1 (es) 2019-12-04 2022-03-09 Albireo Ab Compuestos de benzoti(di)azepina y su uso como ácido biliar
HUE065571T2 (hu) 2019-12-04 2024-06-28 Albireo Ab Benzotia(di)azepin vegyületek és alkalmazásuk epesav modulátorként
JP2023537285A (ja) 2020-08-03 2023-08-31 アルビレオ・アクチボラグ ベンゾチア（ジ）アゼピン化合物及び胆汁酸モジュレータとしてのそれらの使用
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KR20230117393A (ko) 2020-12-04 2023-08-08 알비레오 에이비 벤조티아(디)아제핀 화합물 및 담즙산 조절제로서의용도
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