NL8801733A - Nieuwe toepassing van 5 ht-3 antagonisten. - Google Patents

Nieuwe toepassing van 5 ht-3 antagonisten. Download PDF

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Publication number
NL8801733A
NL8801733A NL8801733A NL8801733A NL8801733A NL 8801733 A NL8801733 A NL 8801733A NL 8801733 A NL8801733 A NL 8801733A NL 8801733 A NL8801733 A NL 8801733A NL 8801733 A NL8801733 A NL 8801733A
Authority
NL
Netherlands
Prior art keywords
group
antagonist
addiction
carbon atoms
inducing agent
Prior art date
Application number
NL8801733A
Other languages
English (en)
Dutch (nl)
Original Assignee
Sandoz Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sandoz Ag filed Critical Sandoz Ag
Publication of NL8801733A publication Critical patent/NL8801733A/nl

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/38—Heterocyclic compounds having sulfur as a ring hetero atom
    • A61K31/381—Heterocyclic compounds having sulfur as a ring hetero atom having five-membered rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/465—Nicotine; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Addiction (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
NL8801733A 1987-07-11 1988-07-08 Nieuwe toepassing van 5 ht-3 antagonisten. NL8801733A (nl)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
DE3722959 1987-07-11
DE3722959 1987-07-11
DE3735719 1987-10-22
DE3735719 1987-10-22
CH451087 1987-11-19
CH451087 1987-11-19

Publications (1)

Publication Number Publication Date
NL8801733A true NL8801733A (nl) 1989-02-01

Family

ID=27174878

Family Applications (1)

Application Number Title Priority Date Filing Date
NL8801733A NL8801733A (nl) 1987-07-11 1988-07-08 Nieuwe toepassing van 5 ht-3 antagonisten.

Country Status (18)

Country Link
US (1) US5039680A (da)
EP (1) EP0302008A3 (da)
JP (1) JPS6431729A (da)
KR (1) KR890001537A (da)
AT (1) AT401615B (da)
AU (3) AU618008B2 (da)
BE (1) BE1004835A5 (da)
DE (1) DE3822792C2 (da)
DK (1) DK385388A (da)
FR (1) FR2617713A1 (da)
GB (2) GB2206788B (da)
HU (1) HU206042B (da)
IT (1) IT1226632B (da)
MY (1) MY103536A (da)
NL (1) NL8801733A (da)
PH (1) PH27002A (da)
PT (1) PT87958B (da)
SE (1) SE8802570L (da)

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DE3822792C2 (de) * 1987-07-11 1997-11-27 Sandoz Ag Neue Verwendung von 5HT¶3¶-Antagonisten
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US5276050A (en) * 1989-08-01 1994-01-04 Glaxo Group Limited Medicaments
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Also Published As

Publication number Publication date
AU1892088A (en) 1989-01-12
FR2617713A1 (fr) 1989-01-13
AU8562891A (en) 1991-12-05
SE8802570D0 (sv) 1988-07-08
EP0302008A2 (en) 1989-02-01
PT87958B (pt) 1995-03-01
IT8848172A0 (it) 1988-07-11
SE8802570L (sv) 1989-03-28
IT1226632B (it) 1991-01-28
GB2240475A (en) 1991-08-07
GB9104598D0 (en) 1991-04-17
EP0302008A3 (en) 1992-12-23
KR890001537A (ko) 1989-03-27
GB2206788B (en) 1992-03-25
PH27002A (en) 1993-02-01
MY103536A (en) 1993-07-31
US5039680A (en) 1991-08-13
AU643075B2 (en) 1993-11-04
AU618008B2 (en) 1991-12-12
PT87958A (pt) 1989-06-30
GB8816298D0 (en) 1988-08-10
GB2206788A (en) 1989-01-18
AU633762B2 (en) 1993-02-04
HUT50038A (en) 1989-12-28
AU8563091A (en) 1991-12-12
HU206042B (en) 1992-08-28
BE1004835A5 (fr) 1993-02-09
DE3822792A1 (de) 1989-01-19
DK385388D0 (da) 1988-07-08
AT401615B (de) 1996-10-25
GB2240475B (en) 1992-03-18
JPS6431729A (en) 1989-02-02
DE3822792C2 (de) 1997-11-27
DK385388A (da) 1989-01-12
FR2617713B1 (da) 1994-08-19

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