MY171483A - Process for making isoquinoline compounds - Google Patents
Process for making isoquinoline compoundsInfo
- Publication number
- MY171483A MY171483A MYPI2015000128A MYPI2015000128A MY171483A MY 171483 A MY171483 A MY 171483A MY PI2015000128 A MYPI2015000128 A MY PI2015000128A MY PI2015000128 A MYPI2015000128 A MY PI2015000128A MY 171483 A MY171483 A MY 171483A
- Authority
- MY
- Malaysia
- Prior art keywords
- compounds
- isoquinoline compounds
- making
- making isoquinoline
- hif
- Prior art date
Links
- 125000002183 isoquinolinyl group Chemical class C1(=NC=CC2=CC=CC=C12)* 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 3
- 230000000694 effects Effects 0.000 abstract 2
- 206010021143 Hypoxia Diseases 0.000 abstract 1
- 102000008109 Mixed Function Oxygenases Human genes 0.000 abstract 1
- 108010074633 Mixed Function Oxygenases Proteins 0.000 abstract 1
- 230000003247 decreasing effect Effects 0.000 abstract 1
- 230000007954 hypoxia Effects 0.000 abstract 1
- 230000001939 inductive effect Effects 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
- C07D217/22—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
- C07D217/26—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P39/00—General protective or antinoxious agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/06—Antianaemics
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Toxicology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Epidemiology (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201261672191P | 2012-07-16 | 2012-07-16 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MY171483A true MY171483A (en) | 2019-10-15 |
Family
ID=48857024
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MYPI2015000128A MY171483A (en) | 2012-07-16 | 2013-07-15 | Process for making isoquinoline compounds |
Country Status (22)
| Country | Link |
|---|---|
| US (2) | US9340511B2 (enExample) |
| EP (2) | EP2872487B1 (enExample) |
| JP (1) | JP6196671B2 (enExample) |
| KR (1) | KR102145272B1 (enExample) |
| CN (2) | CN103435546B (enExample) |
| AU (1) | AU2013290437B2 (enExample) |
| BR (1) | BR112015001106B1 (enExample) |
| CA (1) | CA2879238C (enExample) |
| CY (1) | CY2022018I1 (enExample) |
| DK (1) | DK2872487T3 (enExample) |
| ES (1) | ES2631655T3 (enExample) |
| HU (2) | HUE034409T2 (enExample) |
| IL (1) | IL236625B (enExample) |
| IN (1) | IN2015KN00265A (enExample) |
| MX (1) | MX350922B (enExample) |
| MY (1) | MY171483A (enExample) |
| NZ (1) | NZ704660A (enExample) |
| PL (1) | PL2872487T3 (enExample) |
| PT (1) | PT2872487T (enExample) |
| SG (1) | SG11201500234YA (enExample) |
| WO (1) | WO2014014834A1 (enExample) |
| ZA (1) | ZA201500664B (enExample) |
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| US8883823B2 (en) | 2012-07-16 | 2014-11-11 | Fibrogen, Inc. | Crystalline forms of a prolyl hydroxylase inhibitor |
| BR112015001106B1 (pt) | 2012-07-16 | 2021-11-09 | Fibrogen, Inc | Métodos para a produção de compostos de isoquinolina |
| CN107540607A (zh) * | 2012-07-16 | 2018-01-05 | 菲布罗根有限公司 | 脯氨酰羟化酶抑制剂的晶体形态 |
| PT3003284T (pt) | 2013-06-06 | 2020-08-10 | Fibrogen Inc | Formulações farmacêuticas de um inibidor da hidroxilase do fih |
| CN103694172A (zh) * | 2013-12-26 | 2014-04-02 | 辽宁亿灵科创生物医药科技有限公司 | 含氮杂芳基化合物的衍生物 |
| CN105384687B (zh) | 2014-09-02 | 2018-05-01 | 广东东阳光药业有限公司 | 喹啉酮类化合物及其在药物中应用 |
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| EP2951159B1 (en) | 2013-01-24 | 2018-08-22 | Fibrogen, Inc. | Crystalline forms of {[1-cyano-5-(4-chlorophenoxy)-4-hydroxy-isoquinoline-3-carbonyl]-amino}-acetic acid |
| PT3003284T (pt) | 2013-06-06 | 2020-08-10 | Fibrogen Inc | Formulações farmacêuticas de um inibidor da hidroxilase do fih |
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2013
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