MXPA05008993A - Derivados de diarilcicloalquilo, metodo para su produccion y su uso como medicamentos. - Google Patents

Derivados de diarilcicloalquilo, metodo para su produccion y su uso como medicamentos.

Info

Publication number
MXPA05008993A
MXPA05008993A MXPA05008993A MXPA05008993A MXPA05008993A MX PA05008993 A MXPA05008993 A MX PA05008993A MX PA05008993 A MXPA05008993 A MX PA05008993A MX PA05008993 A MXPA05008993 A MX PA05008993A MX PA05008993 A MXPA05008993 A MX PA05008993A
Authority
MX
Mexico
Prior art keywords
production
disorders
medicaments
derivatives
diarylcycloalkyl
Prior art date
Application number
MXPA05008993A
Other languages
English (en)
Inventor
Goerlitzer Jochen
Original Assignee
Aventis Pharma Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Gmbh filed Critical Aventis Pharma Gmbh
Publication of MXPA05008993A publication Critical patent/MXPA05008993A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D263/32—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Cardiology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

La invencion se refiere a derivados de diarilcicloalquilo y a sus sales fisiologicamente aceptables, racematos y derivados fisiologicamente funcionales. La invencion se refiere a compuestos de la formula (I), (ver formula (I)), en la que los grupos se definen como se cita en la memoria descriptiva, ademas de sus sales fisiologicamente compatibles y a un metodo para su produccion; Los compuestos son adecuados para el tratamiento y/o prevencion de trastornos del metabolismo de acidos grasos y trastornos de la utilizacion de la glucosa, ademas de trastornos en los que juega parte la resistencia a la insulina.
MXPA05008993A 2003-02-27 2004-02-19 Derivados de diarilcicloalquilo, metodo para su produccion y su uso como medicamentos. MXPA05008993A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10308353A DE10308353A1 (de) 2003-02-27 2003-02-27 Diarylcycloalkylderivate, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
PCT/EP2004/001584 WO2004075815A2 (de) 2003-02-27 2004-02-19 Diarylcycloalkylderivate, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel

Publications (1)

Publication Number Publication Date
MXPA05008993A true MXPA05008993A (es) 2005-10-18

Family

ID=32920627

Family Applications (1)

Application Number Title Priority Date Filing Date
MXPA05008993A MXPA05008993A (es) 2003-02-27 2004-02-19 Derivados de diarilcicloalquilo, metodo para su produccion y su uso como medicamentos.

Country Status (21)

Country Link
US (1) US7160911B2 (es)
EP (1) EP1599454B1 (es)
JP (1) JP2006519197A (es)
KR (1) KR20050106053A (es)
CN (1) CN100439346C (es)
AR (1) AR043430A1 (es)
AU (1) AU2004216520B2 (es)
BR (1) BRPI0407901A (es)
CA (1) CA2516573A1 (es)
CO (1) CO5690579A2 (es)
DE (1) DE10308353A1 (es)
HR (1) HRP20050740A2 (es)
IL (1) IL170313A (es)
MA (1) MA27741A1 (es)
MX (1) MXPA05008993A (es)
NO (1) NO20054382L (es)
PL (1) PL377741A1 (es)
RU (1) RU2005129999A (es)
TW (1) TW200505880A (es)
WO (1) WO2004075815A2 (es)
ZA (1) ZA200505763B (es)

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DE102004040736B4 (de) * 2004-08-23 2007-01-11 Sanofi-Aventis Deutschland Gmbh Verfahren zur Herstellung von Diarylcycloalkylderivaten
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Also Published As

Publication number Publication date
US20040204462A1 (en) 2004-10-14
ZA200505763B (en) 2006-05-31
HRP20050740A2 (en) 2006-08-31
IL170313A (en) 2010-11-30
EP1599454A2 (de) 2005-11-30
PL377741A1 (pl) 2006-02-20
AU2004216520B2 (en) 2010-01-07
AR043430A1 (es) 2005-07-27
CN1753880A (zh) 2006-03-29
CN100439346C (zh) 2008-12-03
MA27741A1 (fr) 2006-02-01
TW200505880A (en) 2005-02-16
CA2516573A1 (en) 2004-09-10
US7160911B2 (en) 2007-01-09
KR20050106053A (ko) 2005-11-08
WO2004075815A2 (de) 2004-09-10
AU2004216520A1 (en) 2004-09-10
NO20054382L (no) 2005-09-21
DE10308353A1 (de) 2004-12-02
JP2006519197A (ja) 2006-08-24
RU2005129999A (ru) 2006-03-27
CO5690579A2 (es) 2006-10-31
WO2004075815A3 (de) 2004-12-29
BRPI0407901A (pt) 2006-02-14
EP1599454B1 (de) 2012-12-26

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