MX6289E - Procedimiento mejorado para la preparacion de 2-metil-2-hidroxipropil-piperazin-1-carboxilatos 4-substituidos - Google Patents

Procedimiento mejorado para la preparacion de 2-metil-2-hidroxipropil-piperazin-1-carboxilatos 4-substituidos

Info

Publication number
MX6289E
MX6289E MX797985U MX798579U MX6289E MX 6289 E MX6289 E MX 6289E MX 797985 U MX797985 U MX 797985U MX 798579 U MX798579 U MX 798579U MX 6289 E MX6289 E MX 6289E
Authority
MX
Mexico
Prior art keywords
hydroxipropil
piperazin
carboxylates
substituted
methyl
Prior art date
Application number
MX797985U
Other languages
English (en)
Inventor
Irving Maurice Goldman
Donald Ernest Kuhla
Constantine Sklavouwnos
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of MX6289E publication Critical patent/MX6289E/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/16Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/20Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof
    • C07D295/205Radicals derived from carbonic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/95Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Hydrogenated Pyridines (AREA)
MX797985U 1978-05-18 1979-05-17 Procedimiento mejorado para la preparacion de 2-metil-2-hidroxipropil-piperazin-1-carboxilatos 4-substituidos MX6289E (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US90708278A 1978-05-18 1978-05-18

Publications (1)

Publication Number Publication Date
MX6289E true MX6289E (es) 1985-03-18

Family

ID=25423490

Family Applications (1)

Application Number Title Priority Date Filing Date
MX797985U MX6289E (es) 1978-05-18 1979-05-17 Procedimiento mejorado para la preparacion de 2-metil-2-hidroxipropil-piperazin-1-carboxilatos 4-substituidos

Country Status (42)

Country Link
US (1) US4550164A (es)
JP (1) JPS5946512B2 (es)
AR (1) AR220195A1 (es)
AT (1) AT375357B (es)
AU (1) AU510441B2 (es)
BE (1) BE876311A (es)
BG (1) BG31228A3 (es)
CA (1) CA1097643A (es)
CH (1) CH638796A5 (es)
CS (1) CS236762B2 (es)
DD (1) DD143428A5 (es)
DE (1) DE2919799C2 (es)
DK (6) DK153878C (es)
EG (1) EG13904A (es)
ES (1) ES480669A1 (es)
FI (1) FI64588C (es)
FR (2) FR2432022A1 (es)
GB (1) GB2021107B (es)
GR (1) GR72720B (es)
GT (1) GT197957903A (es)
HK (1) HK13484A (es)
HU (1) HU180282B (es)
IE (1) IE48048B1 (es)
IL (1) IL57295A (es)
IN (1) IN151190B (es)
IT (1) IT1114238B (es)
KE (1) KE3353A (es)
LU (1) LU81271A1 (es)
MX (1) MX6289E (es)
MY (1) MY8500095A (es)
NL (1) NL183190C (es)
NO (1) NO151156C (es)
NZ (1) NZ190473A (es)
PH (2) PH15546A (es)
PL (1) PL118664B1 (es)
PT (1) PT69623A (es)
RO (1) RO76812A (es)
SE (1) SE446183B (es)
SG (1) SG65783G (es)
SU (1) SU1007557A3 (es)
YU (1) YU41633B (es)
ZA (1) ZA792391B (es)

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1096204A (fr) * 1949-06-30 1955-06-16 Saint Gobain Procédé de fabrication d'uréthanes dérivées des glycols
FR62617E (fr) * 1951-06-29 1955-06-15 Saint Gobain Procédé de fabrication d'uréthanes dérivées des glycols
DE1249852B (de) * 1964-10-07 1967-09-14 Dr Christian Brunnengraber Che mische Fabrik &. Co mbH Lübeck Verfahren zur Herstellung von Carbamm saureestern von a Glycermathern
US3703538A (en) * 1969-02-03 1972-11-21 Jefferson Chem Co Inc Production of anhydrous beta-hydroxy-alkyl carbamates
US3935213A (en) * 1973-12-05 1976-01-27 Pfizer Inc. Process for hypotensive 4-amino-2-(piperazin-1-yl) quinazoline derivatives

Also Published As

Publication number Publication date
DK153840B (da) 1988-09-12
DE2919799C2 (de) 1985-12-05
IT7922759A0 (it) 1979-05-17
SE7904313L (sv) 1979-11-19
HU180282B (en) 1983-02-28
IL57295A (en) 1982-01-31
GT197957903A (es) 1980-11-07
HK13484A (en) 1984-02-24
LU81271A1 (fr) 1979-12-07
SE446183B (sv) 1986-08-18
GB2021107B (en) 1982-07-28
DK153880C (da) 1989-02-06
FR2429788A1 (fr) 1980-01-25
DK153878B (da) 1988-09-19
DK153878C (da) 1989-02-06
DK19287A (da) 1987-01-15
ATA366579A (de) 1983-12-15
DK95979A (da) 1979-11-19
PL118664B1 (en) 1981-10-31
CH638796A5 (fr) 1983-10-14
FR2429788B1 (es) 1982-04-16
PL215383A1 (es) 1980-08-11
CS236762B2 (en) 1985-05-15
DK19587A (da) 1987-01-15
MY8500095A (en) 1985-12-31
GB2021107A (en) 1979-11-28
YU41633B (en) 1987-12-31
DK153879C (da) 1989-02-06
SU1007557A3 (ru) 1983-03-23
YU113979A (en) 1983-02-28
IN151190B (es) 1983-03-05
SG65783G (en) 1984-07-27
AT375357B (de) 1984-07-25
FI791579A (fi) 1979-11-19
US4550164A (en) 1985-10-29
IE790962L (en) 1979-11-18
DK153879B (da) 1988-09-19
AR220195A1 (es) 1980-10-15
DK153880B (da) 1988-09-19
CA1097643A (en) 1981-03-17
AU510441B2 (en) 1980-06-26
NO151156C (no) 1985-02-20
DK19287D0 (da) 1987-01-15
JPS54151991A (en) 1979-11-29
NO151156B (no) 1984-11-12
ES480669A1 (es) 1980-05-16
DK19687D0 (da) 1987-01-15
NL183190C (nl) 1988-08-16
DK19487A (da) 1987-01-15
DE2919799A1 (de) 1979-11-22
IE48048B1 (en) 1984-09-05
DK19587D0 (da) 1987-01-15
DK19687A (da) 1987-01-15
DK153881C (da) 1989-02-06
GR72720B (es) 1983-12-01
DD143428A5 (de) 1980-08-20
DK153840C (da) 1989-01-30
FR2432022A1 (fr) 1980-02-22
RO76812A (ro) 1981-05-30
PT69623A (en) 1979-06-01
PH15546A (en) 1983-02-09
NZ190473A (en) 1981-01-23
IT1114238B (it) 1986-01-27
AU4710279A (en) 1979-11-22
NL7903892A (nl) 1979-11-20
PH16236A (en) 1983-08-11
KE3353A (en) 1983-12-16
EG13904A (en) 1983-12-31
NO791641L (no) 1979-11-20
BE876311A (fr) 1979-11-19
FR2432022B1 (es) 1983-07-08
FI64588C (fi) 1983-12-12
DK19487D0 (da) 1987-01-15
ZA792391B (en) 1980-05-28
JPS5946512B2 (ja) 1984-11-13
NL183190B (nl) 1988-03-16
BG31228A3 (en) 1981-11-16
DK19387A (da) 1987-01-15
DK19387D0 (da) 1987-01-15
IL57295A0 (en) 1979-09-30
FI64588B (fi) 1983-08-31
DK153881B (da) 1988-09-19

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