MX2022006861A - Agonistas del receptor glp2 y metodos de uso. - Google Patents
Agonistas del receptor glp2 y metodos de uso.Info
- Publication number
- MX2022006861A MX2022006861A MX2022006861A MX2022006861A MX2022006861A MX 2022006861 A MX2022006861 A MX 2022006861A MX 2022006861 A MX2022006861 A MX 2022006861A MX 2022006861 A MX2022006861 A MX 2022006861A MX 2022006861 A MX2022006861 A MX 2022006861A
- Authority
- MX
- Mexico
- Prior art keywords
- methods
- receptor agonists
- glp
- glp2
- glp2 receptor
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/575—Hormones
- C07K14/605—Glucagons
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
- A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
- A61K47/54—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic compound
- A61K47/542—Carboxylic acids, e.g. a fatty acid or an amino acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/22—Hormones
- A61K38/26—Glucagons
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
- A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
- A61K47/56—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule
- A61K47/59—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyureas or polyurethanes
- A61K47/60—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyureas or polyurethanes the organic macromolecular compound being a polyoxyalkylene oligomer, polymer or dendrimer, e.g. PEG, PPG, PEO or polyglycerol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Epidemiology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Endocrinology (AREA)
- Diabetes (AREA)
- Gastroenterology & Hepatology (AREA)
- Zoology (AREA)
- Molecular Biology (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- Genetics & Genomics (AREA)
- Toxicology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Hospice & Palliative Care (AREA)
- Child & Adolescent Psychology (AREA)
- Psychiatry (AREA)
- Psychology (AREA)
- Immunology (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Emergency Medicine (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201962943667P | 2019-12-04 | 2019-12-04 | |
| US202062994791P | 2020-03-25 | 2020-03-25 | |
| PCT/US2020/063130 WO2021113524A2 (en) | 2019-12-04 | 2020-12-03 | Glp2 receptor agonists and methods of use |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2022006861A true MX2022006861A (es) | 2022-07-11 |
Family
ID=76222285
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2022006861A MX2022006861A (es) | 2019-12-04 | 2020-12-03 | Agonistas del receptor glp2 y metodos de uso. |
| MX2022006732A MX2022006732A (es) | 2019-12-04 | 2020-12-03 | Conjugados peptidicos y metodos de uso. |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2022006732A MX2022006732A (es) | 2019-12-04 | 2020-12-03 | Conjugados peptidicos y metodos de uso. |
Country Status (10)
| Country | Link |
|---|---|
| US (2) | US12583900B2 (https=) |
| EP (2) | EP4069274A4 (https=) |
| JP (2) | JP7691421B2 (https=) |
| KR (2) | KR20220110244A (https=) |
| CN (2) | CN115052886B (https=) |
| AU (2) | AU2020397917A1 (https=) |
| CA (2) | CA3163522A1 (https=) |
| IL (2) | IL293460A (https=) |
| MX (2) | MX2022006861A (https=) |
| WO (2) | WO2021113535A1 (https=) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2014364589B2 (en) | 2013-12-18 | 2020-02-27 | The California Institute For Biomedical Research | Modified therapeutic agents, stapled peptide lipid conjugates, and compositions thereof |
| AU2020397917A1 (en) | 2019-12-04 | 2022-06-23 | The Scripps Research Institute | GLP2 receptor agonists and methods of use |
| MX2023014771A (es) | 2021-06-09 | 2024-03-19 | Scripps Research Inst | Conjugados peptidicos duales gip/glp-1 de accion prolongada y metodos de uso. |
| WO2023207106A1 (zh) * | 2022-04-29 | 2023-11-02 | 苏州星洲生物科技有限公司 | Glp-1/gip受体共激动剂、包含其的药物组合物及其用途 |
| CN114949183B (zh) * | 2022-05-07 | 2023-02-28 | 山东京卫制药有限公司 | 一种替尔泊肽粉雾剂及其制备方法 |
| TW202410918A (zh) * | 2022-05-27 | 2024-03-16 | 韓商Ｄ＆Ｄ製藥科技股份有限公司 | 用於治療神經病症之組合物及方法 |
| CR20250247A (es) * | 2022-12-21 | 2025-08-18 | Boehringer Ingelheim Int | Agonistas triples de los receptores de glp1/gip/npy2 |
| CN117586374B (zh) * | 2023-10-07 | 2024-11-29 | 深圳湾实验室 | Glp-1r/gipr/gcgr三重激动剂类似物及其用途 |
| WO2025184552A2 (en) * | 2024-03-01 | 2025-09-04 | The Scripps Research Institute | Dual gip/glp-1 peptide conjugates and methods of use |
| WO2025217640A1 (en) * | 2024-04-12 | 2025-10-16 | Eli Lilly And Company | Compositions and methods for treating metabolic diseases |
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-
2020
- 2020-12-03 AU AU2020397917A patent/AU2020397917A1/en active Pending
- 2020-12-03 MX MX2022006861A patent/MX2022006861A/es unknown
- 2020-12-03 WO PCT/US2020/063149 patent/WO2021113535A1/en not_active Ceased
- 2020-12-03 JP JP2022531616A patent/JP7691421B2/ja active Active
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| CA3163522A1 (en) | 2021-06-10 |
| CN115052886B (zh) | 2025-09-09 |
| CA3163507A1 (en) | 2021-06-10 |
| WO2021113524A3 (en) | 2021-07-15 |
| JP7834640B2 (ja) | 2026-03-24 |
| EP4069274A4 (en) | 2024-04-10 |
| JP2023513658A (ja) | 2023-04-03 |
| US12583900B2 (en) | 2026-03-24 |
| AU2020397918A1 (en) | 2022-06-23 |
| EP4069726A2 (en) | 2022-10-12 |
| AU2020397917A1 (en) | 2022-06-23 |
| CN115052615A (zh) | 2022-09-13 |
| KR20220123648A (ko) | 2022-09-08 |
| CN115052886A (zh) | 2022-09-13 |
| EP4069274A1 (en) | 2022-10-12 |
| IL293460A (en) | 2022-07-01 |
| KR20220110244A (ko) | 2022-08-05 |
| EP4069726A4 (en) | 2024-03-20 |
| WO2021113535A1 (en) | 2021-06-10 |
| IL293522A (en) | 2022-08-01 |
| US20230057847A1 (en) | 2023-02-23 |
| MX2022006732A (es) | 2022-08-19 |
| JP7691421B2 (ja) | 2025-06-11 |
| WO2021113524A2 (en) | 2021-06-10 |
| US20230071371A1 (en) | 2023-03-09 |
| JP2023504184A (ja) | 2023-02-01 |
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