MX2021015546A - Proceso para preparar 4-amino-piridazinas. - Google Patents
Proceso para preparar 4-amino-piridazinas.Info
- Publication number
- MX2021015546A MX2021015546A MX2021015546A MX2021015546A MX2021015546A MX 2021015546 A MX2021015546 A MX 2021015546A MX 2021015546 A MX2021015546 A MX 2021015546A MX 2021015546 A MX2021015546 A MX 2021015546A MX 2021015546 A MX2021015546 A MX 2021015546A
- Authority
- MX
- Mexico
- Prior art keywords
- preparing
- amino
- pyridazines
- ivb
- relates
- Prior art date
Links
- 238000004519 manufacturing process Methods 0.000 title abstract 2
- LUCGBEPEAUHERV-UHFFFAOYSA-N pyridazin-4-amine Chemical class NC1=CC=NN=C1 LUCGBEPEAUHERV-UHFFFAOYSA-N 0.000 title 1
- -1 pyridazine amine compound Chemical class 0.000 abstract 3
- 125000003277 amino group Chemical group 0.000 abstract 1
- 125000000031 ethylamino group Chemical group [H]C([H])([H])C([H])([H])N([H])[*] 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
- C07D237/02—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
- C07D237/06—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
- C07D237/10—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D237/20—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B31/00—Reduction in general
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B39/00—Halogenation
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B43/00—Formation or introduction of functional groups containing nitrogen
- C07B43/04—Formation or introduction of functional groups containing nitrogen of amino groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
- C07D237/02—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
- C07D237/06—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
- C07D237/10—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D237/12—Halogen atoms or nitro radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Health & Medical Sciences (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Abstract
La presente invención se refiere a un proceso para preparar un compuesto de piridazinamina de fórmula V, y a procesos para preparar compuestos de dicloropiridazinamina de fórmula IVa, IVb, o mezclas de las mismas. Además, la presente invención se refiere a los nuevos compuestos de dicloropiridazinamina de fórmula IVa, IVb, o mezclas de las mismas, en donde el grupo amino es un grupo etilamino.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201562159392P | 2015-05-11 | 2015-05-11 | |
EP15169166 | 2015-05-26 |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2021015546A true MX2021015546A (es) | 2022-02-23 |
Family
ID=53274420
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2017014287A MX2017014287A (es) | 2015-05-11 | 2016-05-10 | Proceso para preparar 4-amino-piridazinas. |
MX2021015546A MX2021015546A (es) | 2015-05-11 | 2017-11-07 | Proceso para preparar 4-amino-piridazinas. |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2017014287A MX2017014287A (es) | 2015-05-11 | 2016-05-10 | Proceso para preparar 4-amino-piridazinas. |
Country Status (17)
Country | Link |
---|---|
US (3) | US10584102B2 (es) |
EP (2) | EP3872073A1 (es) |
JP (1) | JP6833718B2 (es) |
KR (3) | KR102585412B1 (es) |
CN (1) | CN107592859A (es) |
AU (1) | AU2016260784B2 (es) |
BR (1) | BR112017023935B1 (es) |
CA (2) | CA2984703C (es) |
CL (1) | CL2017002813A1 (es) |
CO (1) | CO2017012403A2 (es) |
ES (1) | ES2882543T3 (es) |
IL (1) | IL255302B (es) |
MX (2) | MX2017014287A (es) |
PE (1) | PE20180327A1 (es) |
RU (1) | RU2742663C2 (es) |
WO (1) | WO2016180833A1 (es) |
ZA (1) | ZA201708142B (es) |
Families Citing this family (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2016016369A1 (en) | 2014-07-31 | 2016-02-04 | Basf Se | Process for preparing pyrazoles |
EP3294720B1 (en) | 2015-05-08 | 2020-12-02 | BASF Agro B.V. | A process for the preparation of terpinolene epoxide |
DK3294700T3 (da) | 2015-05-08 | 2020-04-14 | Basf Agro Bv | Fremgangsmåde til fremstilling af limonen-4-ol |
EP3872073A1 (en) | 2015-05-11 | 2021-09-01 | Basf Se | Process for preparing 4-amino-pyridazines |
WO2017133942A1 (en) | 2016-02-02 | 2017-08-10 | Basf Se | Catalytic hydrogenation process for preparing pyrazoles |
KR20190017926A (ko) | 2016-06-15 | 2019-02-20 | 바스프 아그로 비.브이. | 사치환된 알켄의 에폭시화 방법 |
ES2833202T3 (es) | 2016-06-15 | 2021-06-14 | Basf Agro Bv | Procedimiento para la epoxidación de un alqueno tetrasustituido |
US10526264B2 (en) | 2016-07-07 | 2020-01-07 | Basf Se | Oxy-cope rearrangement for the manufacture of insecticidal cyclopentene compounds |
WO2018082964A1 (en) | 2016-11-04 | 2018-05-11 | Basf Se | Process for the production of pyridazinyl-amides in a one-pot synthesis |
WO2018083040A1 (en) | 2016-11-04 | 2018-05-11 | Basf Se | Process for purification of pyrazolpyridazines |
US10538493B2 (en) | 2016-11-17 | 2020-01-21 | Basf Se | Process for the purification of 1-(4-chlorophenyl)pyrazol-3-ol |
MX2019009729A (es) | 2017-02-14 | 2019-10-22 | Basf Se | Formulacion estable de plaguicidas de piridazinpirazolamidas. |
JP7005651B2 (ja) | 2017-03-20 | 2022-01-21 | ビーエーエスエフ ソシエタス・ヨーロピア | ブロモトリクロロメタンを調製する方法 |
FI3908584T3 (fi) * | 2019-01-11 | 2023-06-19 | Basf Se | 1-(1,2-dimetyylipropyyli)-N-etyyli-5-metyyli-N-pyridatsin-4-yylipyratsoli-4-karboksamidin kiteisiä muotoja |
EP3962269A1 (en) | 2019-05-03 | 2022-03-09 | Basf Se | Stabilization of suspension concentrates by ethoxylated ricinolein |
CA3135706A1 (en) | 2019-05-03 | 2020-11-12 | Wen Xu | Stabilization of suspension concentrates by highly sulfonated lignosulfonate |
WO2020224943A1 (en) | 2019-05-03 | 2020-11-12 | Basf Se | Stabilization of suspension concentrates by hydrophobic fumed silica |
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US4A (en) * | 1836-08-10 | Stock | ||
US4728355A (en) | 1985-10-10 | 1988-03-01 | Fmc Corporation | Pyridazinylurea plant regulators |
RU2069660C1 (ru) * | 1994-08-23 | 1996-11-27 | Акционерное общество открытого типа "Научно-исследовательский и проектный институт азотной промышленности и продуктов органического синтеза" | Способ получения производных 4-аминопиридина |
DE4430757A1 (de) * | 1994-08-30 | 1996-03-07 | Boehringer Mannheim Gmbh | Neue 4-Aminopyridazine, Verfahren zu ihrer Herstellung sowie diese Verbindungen enthaltende Arzneimittel |
TW406075B (en) * | 1994-12-13 | 2000-09-21 | Upjohn Co | Alkyl substituted piperidinyl and piperazinyl anti-AIDS compounds |
JP4146514B2 (ja) * | 1995-07-06 | 2008-09-10 | ノバルティス アクチエンゲゼルシャフト | ピロロピリミジン類およびその製造方法 |
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HUP0203375A3 (en) | 1999-07-28 | 2005-03-29 | Aventis Pharm Prod Inc | Substituted oxoazaheterocyclyl compounds |
SI1379520T1 (sl) * | 2001-02-23 | 2006-08-31 | Merck & Co Inc | N-substituirani nonaril-heterociklicni NMDA/NR2B antagonisti |
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JP2007326784A (ja) | 2006-06-06 | 2007-12-20 | Sagami Chem Res Center | 1−置換−5−フルオロアルキルピラゾール−4−カルボン酸エステルの製造方法 |
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PL2197280T3 (pl) | 2007-08-27 | 2013-11-29 | Basf Se | Związki pirazolowe do zwalczania szkodników będących bezkręgowcami |
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UA112028C2 (uk) | 2012-12-14 | 2016-07-11 | Пфайзер Лімітед | Похідні імідазопіридазину як модулятори гамка-рецептора |
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CR20160397A (es) | 2014-01-31 | 2016-10-27 | Basf Se | Pirazoles para el control de plagas de invertebrados |
WO2015162133A1 (en) | 2014-04-22 | 2015-10-29 | Basf Se | C3-c4-cycloalkenyl-comprising pyrazoles for controlling invertebrate pests |
WO2015169734A1 (en) | 2014-05-05 | 2015-11-12 | Basf Se | Pyrazoles for controlling invertebrate pests |
WO2015189080A1 (en) | 2014-06-12 | 2015-12-17 | Basf Se | Pesticidally active mixtures |
WO2016016369A1 (en) | 2014-07-31 | 2016-02-04 | Basf Se | Process for preparing pyrazoles |
EP3255990B1 (en) | 2015-02-11 | 2020-06-24 | Basf Se | Pesticidal mixture comprising a pyrazole compound, an insecticide and a fungicide |
WO2016128240A1 (en) | 2015-02-11 | 2016-08-18 | Basf Se | Pesticidal mixture comprising a pyrazole compound and two fungicides |
WO2016128239A1 (en) | 2015-02-11 | 2016-08-18 | Basf Se | Pesticidal mixture comprising a pyrazole compound and a biopesticide |
EP3872073A1 (en) * | 2015-05-11 | 2021-09-01 | Basf Se | Process for preparing 4-amino-pyridazines |
WO2017133942A1 (en) | 2016-02-02 | 2017-08-10 | Basf Se | Catalytic hydrogenation process for preparing pyrazoles |
-
2016
- 2016-05-10 EP EP21163074.4A patent/EP3872073A1/en active Pending
- 2016-05-10 EP EP16724331.0A patent/EP3294725B1/en active Active
- 2016-05-10 MX MX2017014287A patent/MX2017014287A/es unknown
- 2016-05-10 CA CA2984703A patent/CA2984703C/en active Active
- 2016-05-10 ES ES16724331T patent/ES2882543T3/es active Active
- 2016-05-10 KR KR1020177035243A patent/KR102585412B1/ko active IP Right Grant
- 2016-05-10 RU RU2017142621A patent/RU2742663C2/ru active
- 2016-05-10 KR KR1020237033245A patent/KR20230145498A/ko not_active Application Discontinuation
- 2016-05-10 BR BR112017023935-3A patent/BR112017023935B1/pt active IP Right Grant
- 2016-05-10 KR KR1020247006943A patent/KR20240033160A/ko not_active Application Discontinuation
- 2016-05-10 CA CA3187499A patent/CA3187499A1/en active Pending
- 2016-05-10 PE PE2017002379A patent/PE20180327A1/es not_active Application Discontinuation
- 2016-05-10 US US15/572,303 patent/US10584102B2/en active Active
- 2016-05-10 JP JP2017557929A patent/JP6833718B2/ja active Active
- 2016-05-10 CN CN201680026456.2A patent/CN107592859A/zh active Pending
- 2016-05-10 WO PCT/EP2016/060461 patent/WO2016180833A1/en active Application Filing
- 2016-05-10 AU AU2016260784A patent/AU2016260784B2/en active Active
-
2017
- 2017-10-29 IL IL255302A patent/IL255302B/en active IP Right Grant
- 2017-11-07 CL CL2017002813A patent/CL2017002813A1/es unknown
- 2017-11-07 MX MX2021015546A patent/MX2021015546A/es unknown
- 2017-11-30 ZA ZA2017/08142A patent/ZA201708142B/en unknown
- 2017-11-30 CO CONC2017/0012403A patent/CO2017012403A2/es unknown
-
2019
- 2019-12-31 US US16/731,289 patent/US11046656B2/en active Active
-
2021
- 2021-05-18 US US17/323,337 patent/US20210276959A1/en active Pending
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