MX2008012860A - Desazapurinas de utilidad como inhibidores de janus cinasas. - Google Patents
Desazapurinas de utilidad como inhibidores de janus cinasas.Info
- Publication number
- MX2008012860A MX2008012860A MX2008012860A MX2008012860A MX2008012860A MX 2008012860 A MX2008012860 A MX 2008012860A MX 2008012860 A MX2008012860 A MX 2008012860A MX 2008012860 A MX2008012860 A MX 2008012860A MX 2008012860 A MX2008012860 A MX 2008012860A
- Authority
- MX
- Mexico
- Prior art keywords
- compound according
- ring
- aliphatic
- optionally substituted
- nhc
- Prior art date
Links
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Classifications
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- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
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| US78944106P | 2006-04-05 | 2006-04-05 | |
| PCT/US2007/008367 WO2007117494A1 (en) | 2006-04-05 | 2007-04-05 | Deazapurines useful as inhibitors of janus kinases |
Publications (1)
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| MX2008012860A true MX2008012860A (es) | 2009-01-07 |
Family
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| MX2008012860A MX2008012860A (es) | 2006-04-05 | 2007-04-05 | Desazapurinas de utilidad como inhibidores de janus cinasas. |
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| AR045595A1 (es) | 2003-09-04 | 2005-11-02 | Vertex Pharma | Composiciones utiles como inhibidores de proteinas quinasas |
| US7244735B2 (en) * | 2003-12-02 | 2007-07-17 | Vertex Pharmaceuticals Inc. | Heterocyclic protein kinase inhibitors and uses thereof |
| PT1730146E (pt) | 2004-03-30 | 2011-07-11 | Vertex Pharma | Azaindoles úteis como inibidores de jak e outras proteínas quinases |
| AR049333A1 (es) | 2004-04-02 | 2006-07-19 | Vertex Pharma | Azaindoles inhibidores de proteinquinasas rock y otras proteinas quinasas. composiciones farmaceuticas. |
| JP5213229B2 (ja) * | 2004-04-23 | 2013-06-19 | エグゼリクシス， インコーポレイテッド | キナーゼ調節因子および使用方法 |
| US20060122213A1 (en) | 2004-06-30 | 2006-06-08 | Francoise Pierard | Azaindoles useful as inhibitors of protein kinases |
| WO2006096270A1 (en) | 2005-02-03 | 2006-09-14 | Vertex Pharmaceuticals Incorporated | Pyrrolopyrimidines useful as inhibitors of protein kinase |
| AU2006227790B2 (en) | 2005-03-15 | 2009-09-10 | Irm Llc | Compounds and compositions as protein kinase inhibitors |
| EP1881983B1 (en) | 2005-05-20 | 2012-01-11 | Vertex Pharmaceuticals, Inc. | Pyrrolopyridines useful as inhibitors of protein kinase |
| NZ567133A (en) | 2005-09-30 | 2011-07-29 | Vertex Pharma | Deazapurines useful as inhibitors of janus kinases |
| DK3184526T3 (en) * | 2005-12-13 | 2019-01-14 | Incyte Holdings Corp | PYRROLO [2,3-D] PYRIMIDINE DERIVATIVES AS A JANUS-KINASE INHIBITOR |
| NZ601687A (en) | 2006-01-17 | 2014-03-28 | Vertex Pharma | Azaindoles useful as inhibitors of janus kinases |
| KR20090018895A (ko) | 2006-04-05 | 2009-02-24 | 버텍스 파마슈티칼스 인코포레이티드 | 야누스 키나제의 억제제로서 유용한 데아자푸린 |
-
2007
- 2007-04-05 KR KR1020087027078A patent/KR20090018895A/ko not_active Ceased
- 2007-04-05 WO PCT/US2007/008367 patent/WO2007117494A1/en not_active Ceased
- 2007-04-05 EP EP07754825A patent/EP2001884A1/en not_active Withdrawn
- 2007-04-05 SG SG201102383-5A patent/SG170828A1/en unknown
- 2007-04-05 RU RU2008143361/04A patent/RU2008143361A/ru not_active Application Discontinuation
- 2007-04-05 MX MX2008012860A patent/MX2008012860A/es not_active Application Discontinuation
- 2007-04-05 CN CNA200780020405XA patent/CN101460499A/zh active Pending
- 2007-04-05 CA CA002648250A patent/CA2648250A1/en not_active Abandoned
- 2007-04-05 JP JP2009504273A patent/JP2009532475A/ja active Pending
- 2007-04-05 US US11/732,845 patent/US8741912B2/en not_active Expired - Fee Related
- 2007-04-05 AU AU2007235487A patent/AU2007235487A1/en not_active Abandoned
-
2008
- 2008-10-02 IL IL194460A patent/IL194460A0/en unknown
- 2008-10-03 US US12/245,069 patent/US20090227607A1/en not_active Abandoned
- 2008-10-07 ZA ZA2008/08536A patent/ZA200808536B/en unknown
- 2008-11-05 NO NO20084652A patent/NO20084652L/no not_active Application Discontinuation
-
2012
- 2012-02-23 US US13/403,169 patent/US20120316186A1/en not_active Abandoned
-
2013
- 2013-11-01 JP JP2013228595A patent/JP2014024869A/ja not_active Ceased
-
2014
- 2014-04-11 US US14/250,668 patent/US20140315931A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| WO2007117494A1 (en) | 2007-10-18 |
| KR20090018895A (ko) | 2009-02-24 |
| US20090227607A1 (en) | 2009-09-10 |
| JP2009532475A (ja) | 2009-09-10 |
| US8741912B2 (en) | 2014-06-03 |
| SG170828A1 (en) | 2011-05-30 |
| ZA200808536B (en) | 2012-07-25 |
| AU2007235487A1 (en) | 2007-10-18 |
| NO20084652L (no) | 2008-12-03 |
| IL194460A0 (en) | 2009-08-03 |
| CA2648250A1 (en) | 2007-10-18 |
| US20090088445A1 (en) | 2009-04-02 |
| US20120316186A1 (en) | 2012-12-13 |
| JP2014024869A (ja) | 2014-02-06 |
| US20140315931A1 (en) | 2014-10-23 |
| RU2008143361A (ru) | 2010-05-10 |
| EP2001884A1 (en) | 2008-12-17 |
| CN101460499A (zh) | 2009-06-17 |
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