MX2007001851A - Dihidropteridinonas para el tratamiento de enfermedades oncologicas. - Google Patents
Dihidropteridinonas para el tratamiento de enfermedades oncologicas.Info
- Publication number
- MX2007001851A MX2007001851A MX2007001851A MX2007001851A MX2007001851A MX 2007001851 A MX2007001851 A MX 2007001851A MX 2007001851 A MX2007001851 A MX 2007001851A MX 2007001851 A MX2007001851 A MX 2007001851A MX 2007001851 A MX2007001851 A MX 2007001851A
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- Mexico
- Prior art keywords
- compound
- alkyl
- aryl
- optionally
- group
- Prior art date
Links
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| DE102004033670A1 (de) * | 2004-07-09 | 2006-02-02 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Neue Pyridodihydropyrazinone, Verfahren zu Ihrer Herstellung und Ihre Verwendung als Arzneimittel |
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| US7728134B2 (en) * | 2004-08-14 | 2010-06-01 | Boehringer Ingelheim International Gmbh | Hydrates and polymorphs of 4[[(7R)-8-cyclopentyl-7-ethyl-5,6,7,8-tetrahydro-5-methyl-6-oxo-2-pteridinyl]amino]-3-methoxy-N-(1-methyl-4-piperidinyl)-benzamide, process for their manufacture and their use as medicament |
| US20060058311A1 (en) * | 2004-08-14 | 2006-03-16 | Boehringer Ingelheim International Gmbh | Combinations for the treatment of diseases involving cell proliferation |
| EP1630163A1 (de) * | 2004-08-25 | 2006-03-01 | Boehringer Ingelheim Pharma GmbH & Co.KG | Dihydropteridinonderivative, Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel |
| EP1632493A1 (de) * | 2004-08-25 | 2006-03-08 | Boehringer Ingelheim Pharma GmbH & Co.KG | Dihydropteridinonderivative, Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel |
| JP2008510770A (ja) * | 2004-08-26 | 2008-04-10 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | Ｐｌｋ阻害剤としての新規プテリジノン |
| JP2008510771A (ja) * | 2004-08-27 | 2008-04-10 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | ジヒドロプテリジノン、その製造方法および医薬薬剤としてのその使用 |
| DE102004058337A1 (de) * | 2004-12-02 | 2006-06-14 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Verfahren zur Herstellung von annelierten Piperazin-2-on Derivaten |
| JP2009503014A (ja) * | 2005-08-03 | 2009-01-29 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 呼吸器系疾患の治療におけるジヒドロプテリジノン |
| US7439358B2 (en) * | 2006-02-08 | 2008-10-21 | Boehringer Ingelheim International Gmbh | Specific salt, anhydrous and crystalline form of a dihydropteridione derivative |
| CN101437795A (zh) * | 2006-03-07 | 2009-05-20 | 阿斯利康(瑞典)有限公司 | 哌啶衍生物，制备它们的方法，它们作为治疗剂的用途和含有它们的药物组合物 |
| EP3098223A1 (en) | 2007-08-03 | 2016-11-30 | Boehringer Ingelheim International GmbH | Crystalline form of a dihydropteridione derivative |
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2005
- 2005-07-25 US US11/188,926 patent/US20060074088A1/en not_active Abandoned
- 2005-08-09 MX MX2007001851A patent/MX2007001851A/es active IP Right Grant
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- 2005-08-09 CA CA2575787A patent/CA2575787C/en not_active Expired - Fee Related
- 2005-08-09 EP EP19168693.0A patent/EP3560499B1/en not_active Expired - Lifetime
- 2005-08-09 AU AU2005274387A patent/AU2005274387B2/en not_active Ceased
- 2005-08-09 EP EP11185693A patent/EP2409706A1/en not_active Withdrawn
- 2005-08-09 EP EP05770942.0A patent/EP1778240B1/en not_active Expired - Lifetime
- 2005-08-09 RU RU2007109109/15A patent/RU2406503C2/ru not_active IP Right Cessation
- 2005-08-09 KR KR1020077005855A patent/KR101283378B1/ko not_active Expired - Fee Related
- 2005-08-09 CN CN201410065809.2A patent/CN104055778A/zh active Pending
- 2005-08-09 JP JP2007526350A patent/JP2008509949A/ja not_active Withdrawn
- 2005-08-09 ES ES05770942T patent/ES2800308T3/es not_active Expired - Lifetime
- 2005-08-09 MX MX2012004012A patent/MX343697B/es unknown
- 2005-08-09 KR KR1020137009370A patent/KR101353990B1/ko not_active Expired - Fee Related
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- 2005-08-09 PL PL19168693.0T patent/PL3560499T3/pl unknown
- 2005-08-09 WO PCT/EP2005/008626 patent/WO2006018185A2/en not_active Ceased
- 2005-08-09 BR BRPI0513977-5A patent/BRPI0513977A/pt not_active IP Right Cessation
- 2005-08-09 CN CNA2005800277121A patent/CN101022809A/zh active Pending
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