MA41253A - Composés, compositions et procédés pour augmenter l'activité du cftr - Google Patents
Composés, compositions et procédés pour augmenter l'activité du cftrInfo
- Publication number
- MA41253A MA41253A MA041253A MA41253A MA41253A MA 41253 A MA41253 A MA 41253A MA 041253 A MA041253 A MA 041253A MA 41253 A MA41253 A MA 41253A MA 41253 A MA41253 A MA 41253A
- Authority
- MA
- Morocco
- Prior art keywords
- cftr
- compositions
- activity
- compounds
- processes
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title 1
- 239000000203 mixture Substances 0.000 title 1
Classifications
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
- A61K31/341—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide not condensed with another ring, e.g. ranitidine, furosemide, bufetolol, muscarine
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
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- A61K31/42—Oxazoles
- A61K31/422—Oxazoles not condensed and containing further heterocyclic rings
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- A61K31/5375—1,4-Oxazines, e.g. morpholine
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| RU2745977C2 (ru) | 2010-04-22 | 2021-04-05 | Вертекс Фармасьютикалз Инкорпорейтед | Способ получения циклоалкилкарбоксамидо-индольных соединений |
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2015
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- 2015-12-23 EP EP15825647.9A patent/EP3237411B1/fr active Active
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- 2015-12-23 ES ES15825647T patent/ES2962673T3/es active Active
- 2015-12-23 BR BR112017013710-0A patent/BR112017013710B1/pt active IP Right Grant
- 2015-12-23 SG SG11201704859UA patent/SG11201704859UA/en unknown
- 2015-12-23 CN CN201580074407.1A patent/CN107207487B/zh active Active
- 2015-12-23 KR KR1020177020139A patent/KR102677444B1/ko active Active
- 2015-12-23 US US15/539,392 patent/US10392372B2/en active Active
- 2015-12-23 AU AU2015371294A patent/AU2015371294B2/en active Active
- 2015-12-23 NZ NZ732701A patent/NZ732701A/en unknown
- 2015-12-23 MX MX2017008380A patent/MX388421B/es unknown
- 2015-12-23 RU RU2017126232A patent/RU2767460C2/ru active
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2017
- 2017-06-18 IL IL252987A patent/IL252987B/en active IP Right Grant
- 2017-06-26 SA SA517381828A patent/SA517381828B1/ar unknown
-
2019
- 2019-07-12 US US16/510,406 patent/US11098035B2/en active Active
-
2020
- 2020-08-02 IL IL276426A patent/IL276426A/en unknown
- 2020-10-12 AU AU2020256305A patent/AU2020256305A1/en not_active Abandoned
-
2022
- 2022-09-06 AU AU2022228100A patent/AU2022228100A1/en not_active Abandoned
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