MA24563A1 - Derives de macrolides substitues en position c-4 - Google Patents
Derives de macrolides substitues en position c-4Info
- Publication number
- MA24563A1 MA24563A1 MA25106A MA25106A MA24563A1 MA 24563 A1 MA24563 A1 MA 24563A1 MA 25106 A MA25106 A MA 25106A MA 25106 A MA25106 A MA 25106A MA 24563 A1 MA24563 A1 MA 24563A1
- Authority
- MA
- Morocco
- Prior art keywords
- derivatives
- macrolides
- substituted
- substituted macrolides
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicinal Chemistry (AREA)
- Biochemistry (AREA)
- Engineering & Computer Science (AREA)
- Genetics & Genomics (AREA)
- Tropical Medicine & Parasitology (AREA)
- Biotechnology (AREA)
- Molecular Biology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US4998097P | 1997-06-11 | 1997-06-11 |
Publications (1)
Publication Number | Publication Date |
---|---|
MA24563A1 true MA24563A1 (fr) | 1998-12-31 |
Family
ID=21962765
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MA25106A MA24563A1 (fr) | 1997-06-11 | 1998-06-10 | Derives de macrolides substitues en position c-4 |
Country Status (40)
Country | Link |
---|---|
EP (1) | EP0988309B1 (fr) |
JP (1) | JP3262806B2 (fr) |
KR (1) | KR100369959B1 (fr) |
CN (1) | CN1145636C (fr) |
AP (1) | AP1189A (fr) |
AR (1) | AR013085A1 (fr) |
AT (1) | ATE310742T1 (fr) |
AU (1) | AU745006C (fr) |
BG (1) | BG64357B1 (fr) |
BR (1) | BR9810097A (fr) |
CA (1) | CA2293397C (fr) |
CO (1) | CO4950584A1 (fr) |
DE (1) | DE69832486T2 (fr) |
DZ (1) | DZ2515A1 (fr) |
EA (1) | EA002440B1 (fr) |
ES (1) | ES2251081T3 (fr) |
GT (1) | GT199800075A (fr) |
HK (1) | HK1025974A1 (fr) |
HN (1) | HN1998000074A (fr) |
HR (1) | HRP980315A2 (fr) |
HU (1) | HUP0004076A3 (fr) |
ID (1) | ID24530A (fr) |
IL (1) | IL132808A (fr) |
IS (1) | IS1979B (fr) |
MA (1) | MA24563A1 (fr) |
MY (1) | MY133027A (fr) |
NO (1) | NO315560B1 (fr) |
NZ (1) | NZ500652A (fr) |
OA (1) | OA11226A (fr) |
PA (1) | PA8452001A1 (fr) |
PE (1) | PE79999A1 (fr) |
PL (1) | PL337497A1 (fr) |
SK (1) | SK168299A3 (fr) |
TN (1) | TNSN98084A1 (fr) |
TW (2) | TWI224106B (fr) |
UA (1) | UA70298A (fr) |
UY (1) | UY25041A1 (fr) |
WO (1) | WO1998056801A1 (fr) |
YU (1) | YU62999A (fr) |
ZA (1) | ZA985016B (fr) |
Families Citing this family (37)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6339063B1 (en) | 1997-09-10 | 2002-01-15 | Merck & Co., Inc. | 9a-azalides as veterinary antimicrobial agents |
EP1779853A3 (fr) * | 1997-09-10 | 2010-01-27 | Merial Ltd. | 9a-azalides en tant qu'agents anti-microbiens à usage vétérinaire |
DE69837007T2 (de) * | 1997-09-10 | 2007-11-22 | Merial Ltd. | Verwendung von 9a-azaliden als antimikrobielle mittel für tiere |
AP9801420A0 (en) * | 1998-01-02 | 1998-12-31 | Pfizer Prod Inc | Novel macrolides. |
EP1437360A3 (fr) * | 1998-08-19 | 2005-04-06 | Pfizer Products Inc. | C11-carbamates des macrolides antibactériens |
US6043227A (en) * | 1998-08-19 | 2000-03-28 | Pfizer Inc. | C11 carbamates of macrolide antibacterials |
US6100240A (en) * | 1998-10-09 | 2000-08-08 | Pfizer Inc | Macrolide derivatives |
HUP0104192A3 (en) | 1998-11-03 | 2003-12-29 | Pfizer Prod Inc | Novel macrolide antibiotics |
CA2292359C (fr) * | 1999-01-28 | 2004-09-28 | Pfizer Products Inc. | Nouveaux azalides et procede de fabrication |
DK1206476T3 (da) * | 1999-08-24 | 2006-05-15 | Abbott Lab | 9a-azalider med antibakteriel virkning |
US6764996B1 (en) | 1999-08-24 | 2004-07-20 | Abbott Laboratories | 9a-azalides with antibacterial activity |
PT1250343E (pt) | 2000-01-27 | 2003-11-28 | Pfizer Prod Inc | Composicoes de antibioticos de azalida |
CA2445306C (fr) * | 2001-04-27 | 2008-02-12 | Pfizer Products Inc. | Procede de preparation de derives de 9-deoxo-9a-aza-9a-homoerythromycine a substitues en 4'' |
JP2003040782A (ja) * | 2001-05-31 | 2003-02-13 | Pfizer Prod Inc | アザリド抗生物質組成物 |
WO2004005313A2 (fr) | 2002-07-08 | 2004-01-15 | Pliva - Istrazivacki Institut D.O.O. | Nouveaux composes, compositions en tant que porteurs pour molecules actives anti-inflammatoires steroidiennes/non-steroidiennes, antineoplasiques et antivirales |
EP1521763A2 (fr) * | 2002-07-08 | 2005-04-13 | Pliva - Istrazivacki Institut d.o.o. | Substances anti-inflammatoires non steroidiennes, compositions et procedes d'utilisation de celles-ci |
WO2004005310A2 (fr) | 2002-07-08 | 2004-01-15 | Pliva-Istrazivacki Institut D.O.O. | Nouveaux composes, compositions et procedes pour traiter les maladies et etats inflammatoires |
AR043050A1 (es) | 2002-09-26 | 2005-07-13 | Rib X Pharmaceuticals Inc | Compuestos heterociclicos bifuncionales y metodos para preparar y usar los mismos |
US7601695B2 (en) * | 2003-03-10 | 2009-10-13 | Optimer Pharmaceuticals, Inc. | Antibacterial agents |
US7276487B2 (en) | 2003-09-23 | 2007-10-02 | Enanta Pharmaceuticals, Inc. | 9a, 11-3C-bicyclic 9a-azalide derivatives |
CN102816194A (zh) | 2004-02-27 | 2012-12-12 | 瑞伯-X医药品有限公司 | 大环化合物以及其制作和使用方法 |
JPWO2009019868A1 (ja) | 2007-08-06 | 2010-10-28 | 大正製薬株式会社 | 10a、12位架橋型10a−アザライド化合物 |
CA2703475A1 (fr) | 2007-10-25 | 2009-04-30 | Cempra Pharmaceuticals, Inc. | Procede pour la preparation d'agents antibacteriens macrolides |
US8299035B2 (en) | 2008-05-15 | 2012-10-30 | Taisho Pharmaceutucal Co., Ltd. | 10a-azalide compound having 4-membered ring structure |
CN102245195B (zh) | 2008-10-24 | 2016-01-13 | 森普拉制药公司 | 使用含三唑的大环内酯的生物防御 |
US9937194B1 (en) | 2009-06-12 | 2018-04-10 | Cempra Pharmaceuticals, Inc. | Compounds and methods for treating inflammatory diseases |
JP5908479B2 (ja) * | 2010-09-20 | 2016-04-26 | ノバルティス ティーアゲズントハイト アーゲー | クラジノース環のC−4”をエポキシド基で修飾した9−デオキソ−9a−アザ−9a−ホモエリスロマイシンAの新規製造方法 |
AR085286A1 (es) | 2011-02-21 | 2013-09-18 | Taisho Pharmaceutical Co Ltd | Derivado de macrolido sustituido en la posicion c-4 |
EP2830632A4 (fr) | 2012-03-27 | 2015-10-21 | Cempra Pharmaceuticals Inc | Formulations parentérales pour l'administration d'antibiotiques macrolides |
JP5857008B2 (ja) * | 2012-08-20 | 2016-02-10 | 大正製薬株式会社 | C−4”位置換マクロライド誘導体を含有する医薬 |
CN105246334A (zh) | 2013-04-04 | 2016-01-13 | 哈佛大学的校长及成员们 | 大环内酯及其制备和使用方法 |
CN105669798B (zh) * | 2013-08-23 | 2019-07-26 | 普莱柯生物工程股份有限公司 | 一种大环内酯类化合物 |
CN103965273B (zh) | 2013-08-23 | 2016-05-25 | 普莱柯生物工程股份有限公司 | 一种大环内酯类化合物 |
AR102810A1 (es) | 2014-08-18 | 2017-03-29 | Taisho Pharmaceutical Co Ltd | Derivado de macrólido sustituido en la posición c-4 |
US10633407B2 (en) | 2014-10-08 | 2020-04-28 | President And Fellows Of Harvard College | 14-membered ketolides and methods of their preparation and use |
JP2018509452A (ja) | 2015-03-25 | 2018-04-05 | プレジデント アンド フェローズ オブ ハーバード カレッジ | 修飾デソサミン糖をもつマクロライドおよびその使用 |
CN108003207B (zh) | 2017-12-19 | 2019-05-10 | 海门慧聚药业有限公司 | 制备泰拉霉素的方法 |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SE445223B (sv) * | 1977-02-04 | 1986-06-09 | Pfizer | Sett att framstella 4"-amino-erytomylin-a-derivat |
US4150220A (en) * | 1977-02-04 | 1979-04-17 | Pfizer Inc. | Semi-synthetic 4"-erythromycin A derivatives |
YU43006B (en) * | 1981-03-06 | 1989-02-28 | Pliva Pharm & Chem Works | Process for preparing n-methyl-11-aza-10-deoxo-10-dihydro erythromycin and derivatives thereof |
US4474768A (en) * | 1982-07-19 | 1984-10-02 | Pfizer Inc. | N-Methyl 11-aza-10-deoxo-10-dihydro-erytromycin A, intermediates therefor |
GR80277B (en) * | 1983-09-06 | 1985-01-04 | Pfizer | Azahomoerythromycin b derivatives and intermediates therefor |
US4512982A (en) * | 1984-04-13 | 1985-04-23 | Pfizer Inc. | 9α-Aza-9α-homoerythromycin compounds, pharmaceutical composition and therapeutic method |
CA2064634C (fr) * | 1991-04-04 | 1998-08-04 | James V. Heck | Derives de 9-desoxo-8a-aza-8a-homoerythromycine a modifies en positions 4"- et 8a |
US5441939A (en) * | 1994-03-04 | 1995-08-15 | Pfizer Inc. | 3"-desmethoxy derivatives of erythromycin and azithromycin |
US5412982A (en) * | 1994-03-10 | 1995-05-09 | Potts; James K. | Windsock support |
-
1998
- 1998-05-20 HN HN1998000074A patent/HN1998000074A/es unknown
- 1998-05-22 PA PA19988452001A patent/PA8452001A1/es unknown
- 1998-05-25 HU HU0004076A patent/HUP0004076A3/hu unknown
- 1998-05-25 PL PL98337497A patent/PL337497A1/xx unknown
- 1998-05-25 EP EP98919414A patent/EP0988309B1/fr not_active Expired - Lifetime
- 1998-05-25 ES ES98919414T patent/ES2251081T3/es not_active Expired - Lifetime
- 1998-05-25 JP JP50192999A patent/JP3262806B2/ja not_active Expired - Fee Related
- 1998-05-25 NZ NZ500652A patent/NZ500652A/en unknown
- 1998-05-25 BR BR9810097-1A patent/BR9810097A/pt not_active IP Right Cessation
- 1998-05-25 CA CA002293397A patent/CA2293397C/fr not_active Expired - Fee Related
- 1998-05-25 ID IDW991565A patent/ID24530A/id unknown
- 1998-05-25 SK SK1682-99A patent/SK168299A3/sk unknown
- 1998-05-25 DE DE69832486T patent/DE69832486T2/de not_active Expired - Fee Related
- 1998-05-25 AT AT98919414T patent/ATE310742T1/de not_active IP Right Cessation
- 1998-05-25 AU AU72281/98A patent/AU745006C/en not_active Ceased
- 1998-05-25 CN CNB988060493A patent/CN1145636C/zh not_active Expired - Fee Related
- 1998-05-25 UA UA99126737A patent/UA70298A/uk unknown
- 1998-05-25 YU YU62999A patent/YU62999A/sh unknown
- 1998-05-25 EA EA199901014A patent/EA002440B1/ru not_active IP Right Cessation
- 1998-05-25 IL IL13280898A patent/IL132808A/en not_active IP Right Cessation
- 1998-05-25 KR KR10-1999-7011643A patent/KR100369959B1/ko not_active IP Right Cessation
- 1998-05-25 WO PCT/IB1998/000799 patent/WO1998056801A1/fr not_active Application Discontinuation
- 1998-06-04 AP APAP/P/1998/001254A patent/AP1189A/en active
- 1998-06-08 GT GT199800075A patent/GT199800075A/es unknown
- 1998-06-08 TW TW087109085A patent/TWI224106B/zh active
- 1998-06-08 TW TW093111859A patent/TW200418871A/zh unknown
- 1998-06-08 PE PE1998000469A patent/PE79999A1/es not_active Application Discontinuation
- 1998-06-09 AR ARP980102704A patent/AR013085A1/es active IP Right Grant
- 1998-06-09 MY MYPI98002563A patent/MY133027A/en unknown
- 1998-06-10 CO CO98033231A patent/CO4950584A1/es unknown
- 1998-06-10 MA MA25106A patent/MA24563A1/fr unknown
- 1998-06-10 DZ DZ980125A patent/DZ2515A1/fr active
- 1998-06-10 ZA ZA9805016A patent/ZA985016B/xx unknown
- 1998-06-10 TN TNTNSN98084A patent/TNSN98084A1/fr unknown
- 1998-06-11 HR HR60/049,980A patent/HRP980315A2/hr not_active Application Discontinuation
- 1998-06-11 UY UY25041A patent/UY25041A1/es not_active IP Right Cessation
-
1999
- 1999-11-16 IS IS5250A patent/IS1979B/is unknown
- 1999-12-03 OA OA9900270A patent/OA11226A/en unknown
- 1999-12-08 BG BG103969A patent/BG64357B1/bg unknown
- 1999-12-10 NO NO19996107A patent/NO315560B1/no unknown
-
2000
- 2000-08-28 HK HK00105362A patent/HK1025974A1/xx not_active IP Right Cessation
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