LV12354B - USE OF CENTRAL CANABINOIDECEPTIC ANTAGONISTS FOR ADJUSTMENT OF STRAWBERG - Google Patents

USE OF CENTRAL CANABINOIDECEPTIC ANTAGONISTS FOR ADJUSTMENT OF STRAWBERG Download PDF

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Publication number
LV12354B
LV12354B LVP-99-114A LV990114A LV12354B LV 12354 B LV12354 B LV 12354B LV 990114 A LV990114 A LV 990114A LV 12354 B LV12354 B LV 12354B
Authority
LV
Latvia
Prior art keywords
alkyl
group
hydrogen
phenyl
alkoxy
Prior art date
Application number
LVP-99-114A
Other languages
English (en)
Latvian (lv)
Other versions
LV12354A (lv
Inventor
Jeanne Maruani
Phillipe Soubrie
Original Assignee
Sanofi-Synthelabo, Joint Stock Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi-Synthelabo, Joint Stock Company filed Critical Sanofi-Synthelabo, Joint Stock Company
Publication of LV12354A publication Critical patent/LV12354A/xx
Publication of LV12354B publication Critical patent/LV12354B/en

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/32—Alcohol-abuse
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Addiction (AREA)
  • Biomedical Technology (AREA)
  • Obesity (AREA)
  • Diabetes (AREA)
  • Psychiatry (AREA)
  • Hematology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Steroid Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
LVP-99-114A 1997-01-28 1999-07-27 USE OF CENTRAL CANABINOIDECEPTIC ANTAGONISTS FOR ADJUSTMENT OF STRAWBERG LV12354B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9700870A FR2758723B1 (fr) 1997-01-28 1997-01-28 Utilisation des antagonistes des recepteurs aux cannabinoides centraux pour la preparation de medicaments
PCT/FR1998/000154 WO1998032441A1 (fr) 1997-01-28 1998-01-28 Utilisation des antagonistes des recepteurs aux cannabinoides centraux pour reguler l'appetance

Publications (2)

Publication Number Publication Date
LV12354A LV12354A (lv) 1999-10-20
LV12354B true LV12354B (en) 2000-02-20

Family

ID=9503028

Family Applications (1)

Application Number Title Priority Date Filing Date
LVP-99-114A LV12354B (en) 1997-01-28 1999-07-27 USE OF CENTRAL CANABINOIDECEPTIC ANTAGONISTS FOR ADJUSTMENT OF STRAWBERG

Country Status (32)

Country Link
US (3) US6344474B1 (pt)
EP (2) EP1795194A3 (pt)
JP (1) JP3676383B2 (pt)
AR (1) AR011776A1 (pt)
AT (1) ATE358480T1 (pt)
AU (1) AU6219398A (pt)
BR (1) BR9806801A (pt)
CA (1) CA2278661A1 (pt)
DE (1) DE69837473T2 (pt)
DK (1) DK0969835T3 (pt)
DZ (1) DZ2405A1 (pt)
EE (1) EE04630B1 (pt)
ES (1) ES2285760T3 (pt)
FR (1) FR2758723B1 (pt)
GT (1) GT199800021A (pt)
HK (1) HK1022829A1 (pt)
HR (1) HRP980042A2 (pt)
ID (1) ID22216A (pt)
IS (1) IS5113A (pt)
LV (1) LV12354B (pt)
ME (1) MEP26508A (pt)
MY (1) MY117251A (pt)
NO (1) NO323696B1 (pt)
PT (1) PT969835E (pt)
RS (1) RS49830B (pt)
SA (1) SA98181113B1 (pt)
SK (1) SK99799A3 (pt)
TR (1) TR199901721T2 (pt)
TW (1) TW450808B (pt)
UY (1) UY24847A1 (pt)
WO (1) WO1998032441A1 (pt)
ZA (1) ZA98691B (pt)

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SA98181113B1 (ar) 2006-06-25
JP2001501971A (ja) 2001-02-13
MEP26508A (en) 2010-06-10
EP1795194A2 (fr) 2007-06-13
US20020128302A1 (en) 2002-09-12
HK1022829A1 (en) 2000-08-25
CA2278661A1 (en) 1998-07-30
MY117251A (en) 2004-06-30
EP1795194A3 (fr) 2008-04-30
HRP980042A2 (en) 1998-10-31
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NO993634D0 (no) 1999-07-27
ID22216A (id) 1999-09-16
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BR9806801A (pt) 2000-05-16
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EE04630B1 (et) 2006-06-15
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FR2758723B1 (fr) 1999-04-23
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