LU84746A1 - Nouveaux acides diphosphoniques,leurs sels,leur procede de preparation et leur application en therapeutique - Google Patents

Nouveaux acides diphosphoniques,leurs sels,leur procede de preparation et leur application en therapeutique Download PDF

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Publication number
LU84746A1
LU84746A1 LU84746A LU84746A LU84746A1 LU 84746 A1 LU84746 A1 LU 84746A1 LU 84746 A LU84746 A LU 84746A LU 84746 A LU84746 A LU 84746A LU 84746 A1 LU84746 A1 LU 84746A1
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LU
Luxembourg
Prior art keywords
acid
amino
diphosphonic
pharmaceutical compositions
acids
Prior art date
Application number
LU84746A
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English (en)
French (fr)
Inventor
Sergio Rosini
Giorgio Staibano
Original Assignee
Gentili Ist Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=11171970&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=LU84746(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Gentili Ist Spa filed Critical Gentili Ist Spa
Publication of LU84746A1 publication Critical patent/LU84746A1/fr

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/3804—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)] not used, see subgroups
    • C07F9/3839—Polyphosphonic acids
    • C07F9/3873—Polyphosphonic acids containing nitrogen substituent, e.g. N.....H or N-hydrocarbon group which can be substituted by halogen or nitro(so), N.....O, N.....S, N.....C(=X)- (X =O, S), N.....N, N...C(=X)...N (X =O, S)
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/3804—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)] not used, see subgroups
    • C07F9/3839—Polyphosphonic acids
    • C07F9/3856—Polyphosphonic acids containing halogen or nitro(so) substituents

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  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
LU84746A 1982-04-15 1983-04-13 Nouveaux acides diphosphoniques,leurs sels,leur procede de preparation et leur application en therapeutique LU84746A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT2078182 1982-04-15
IT8220781A IT1201087B (it) 1982-04-15 1982-04-15 Bifosfonati farmacologicamente attivi,procedimento per la loro preparazione e relative composizioni farmaceutiche

Publications (1)

Publication Number Publication Date
LU84746A1 true LU84746A1 (fr) 1983-11-17

Family

ID=11171970

Family Applications (2)

Application Number Title Priority Date Filing Date
LU84746A LU84746A1 (fr) 1982-04-15 1983-04-13 Nouveaux acides diphosphoniques,leurs sels,leur procede de preparation et leur application en therapeutique
LU88714C LU88714I2 (fr) 1982-04-15 1983-04-13 Acide 4-amino-1-hydroxybutane-1,1-diphosphonique sels de celui-ci avec un métal alcalin ou une base organique ou un acide aminé basique en particulier le sel trihydraté monosodique de l'acide 4-amino-1-hydroxybutane-1,1-diphosphonique

Family Applications After (1)

Application Number Title Priority Date Filing Date
LU88714C LU88714I2 (fr) 1982-04-15 1983-04-13 Acide 4-amino-1-hydroxybutane-1,1-diphosphonique sels de celui-ci avec un métal alcalin ou une base organique ou un acide aminé basique en particulier le sel trihydraté monosodique de l'acide 4-amino-1-hydroxybutane-1,1-diphosphonique

Country Status (12)

Country Link
US (1) US4621077A (cs)
JP (1) JPS58189193A (cs)
BE (1) BE896453A (cs)
CH (1) CH661437A5 (cs)
FR (1) FR2525223B1 (cs)
GB (1) GB2118042B (cs)
HK (1) HK79390A (cs)
IT (1) IT1201087B (cs)
LU (2) LU84746A1 (cs)
MX (1) MX9203428A (cs)
NL (5) NL192562C (cs)
SE (1) SE463239B (cs)

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JPS5759900A (en) * 1980-09-29 1982-04-10 Vysoka Skola Chem Tech 6-amino-1-hydroxyhexylidene diphosphonic acid
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IT1194748B (it) * 1981-02-12 1988-09-28 Gentili Ist Spa Composizioni farmaceutiche per il trattamento di osteopatie

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IT1201087B (it) 1989-01-27
BE896453A (fr) 1983-08-01
JPS58189193A (ja) 1983-11-04
FR2525223A1 (fr) 1983-10-21
NL980005I1 (nl) 1998-04-01
US4621077A (en) 1986-11-04
NL980010I1 (nl) 1998-05-06
SE463239B (sv) 1990-10-29
IT8220781A0 (it) 1982-04-15
NL192562C (nl) 1997-10-03
LU88714I2 (fr) 1996-08-23
SE8302130L (sv) 1983-10-16
NL980004I1 (nl) 1998-04-01
NL8301324A (nl) 1983-11-01
NL970038I1 (nl) 1998-01-05
FR2525223B1 (fr) 1986-04-25
HK79390A (en) 1990-10-12
SE8302130D0 (sv) 1983-04-15
NL192562B (nl) 1997-06-02
CH661437A5 (it) 1987-07-31
JPH0213645B2 (cs) 1990-04-04
NL970038I2 (nl) 2000-11-01
GB2118042A (en) 1983-10-26
GB8308791D0 (en) 1983-05-11
MX9203428A (es) 1992-07-01
GB2118042B (en) 1986-01-15

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