LT1562567T - Pasirinktų analgetikų ir cox-ii slopiklių derinys - Google Patents

Pasirinktų analgetikų ir cox-ii slopiklių derinys

Info

Publication number
LT1562567T
LT1562567T LTEP03775368.8T LT03775368T LT1562567T LT 1562567 T LT1562567 T LT 1562567T LT 03775368 T LT03775368 T LT 03775368T LT 1562567 T LT1562567 T LT 1562567T
Authority
LT
Lithuania
Prior art keywords
alkyl
hydrogen
optionally substituted
och
hydroxy
Prior art date
Application number
LTEP03775368.8T
Other languages
English (en)
Inventor
Klaus Schiene
Günter HAASE
Babette-Yvonne Kögel
Elmar Friderichs
Ulrich Jahnel
Original Assignee
Grünenthal GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=32395002&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=LT1562567(T) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from DE10254785A external-priority patent/DE10254785A1/de
Priority claimed from DE2003126103 external-priority patent/DE10326103A1/de
Application filed by Grünenthal GmbH filed Critical Grünenthal GmbH
Publication of LT1562567T publication Critical patent/LT1562567T/lt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/63—Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide
    • A61K31/635—Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide having a heterocyclic ring, e.g. sulfadiazine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
    • A61K31/341—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide not condensed with another ring, e.g. ranitidine, furosemide, bufetolol, muscarine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/365—Lactones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A61P29/02—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect
LTEP03775368.8T 2002-11-22 2003-11-18 Pasirinktų analgetikų ir cox-ii slopiklių derinys LT1562567T (lt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE10254785A DE10254785A1 (de) 2002-11-22 2002-11-22 Kombination ausgewählter Analgetika mit COX II-Inhibitoren
DE2003126103 DE10326103A1 (de) 2003-06-06 2003-06-06 Kombination ausgewählter Analgetika mit COX II-Inhibitoren
PCT/EP2003/012882 WO2004047823A1 (de) 2002-11-22 2003-11-18 Kombination ausgewählter analgetika mit cox ii-inhibitoren

Publications (1)

Publication Number Publication Date
LT1562567T true LT1562567T (lt) 2017-08-25

Family

ID=32395002

Family Applications (1)

Application Number Title Priority Date Filing Date
LTEP03775368.8T LT1562567T (lt) 2002-11-22 2003-11-18 Pasirinktų analgetikų ir cox-ii slopiklių derinys

Country Status (13)

Country Link
US (7) US7786160B2 (lt)
EP (6) EP3662904A1 (lt)
AT (2) ATE465726T1 (lt)
AU (1) AU2003283410A1 (lt)
CY (4) CY1108141T1 (lt)
DE (2) DE50312678D1 (lt)
DK (4) DK3241550T3 (lt)
ES (4) ES2819854T3 (lt)
HU (2) HUE051024T2 (lt)
LT (1) LT1562567T (lt)
PT (4) PT1685829E (lt)
SI (4) SI3241550T1 (lt)
WO (1) WO2004047823A1 (lt)

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DK3241550T3 (da) 2002-11-22 2020-08-24 Gruenenthal Gmbh Anvendelse af (1r,2r)-3-(3-dimethylamino-1-ethyl-2-methyl-propyl)-phenol til behandling af inflammatoriske smerter
DE10356362A1 (de) * 2003-11-28 2005-06-23 Grünenthal GmbH Verwendung von 1-Phenyl-3-dimethylamino-propanverbindungen zur Therapie von Angststörungen
US20070254960A1 (en) * 2006-04-28 2007-11-01 Gruenenthal Gmbh Pharmaceutical combination
RU2465263C2 (ru) * 2006-04-28 2012-10-27 Грюненталь Гмбх Фармацевтическая комбинация, включающая 3-(3-диметиламино-1-этил-2-метилпропил)фенол и нестероидный противовоспалительный препарат
PL2012764T3 (pl) * 2006-04-28 2011-04-29 Gruenenthal Gmbh Kombinacja farmaceutyczna zawierająca 3-(3-dimetyloamino-1-etylo-2-metylopropylo)fenol i Paracetamol
DE102007012165A1 (de) * 2007-03-12 2008-09-18 Grünenthal GmbH Verwendung von 1-Phenyl-3-dimethylamino-propanverbindungen zur Therapie des Neuropathieschmerzes
DE102007022790A1 (de) * 2007-05-11 2008-11-20 Grünenthal GmbH Axomadol zur Schmerzbehandlung bei Arthrose
WO2009067703A2 (en) * 2007-11-23 2009-05-28 Nectid, Inc. Tapentadol compositions
EP2085081A1 (de) 2008-02-04 2009-08-05 Grünenthal GmbH 3-(2-Dimethylaminomethyl-cyclohexyl)-phenol gegen polyneuropathischen Schmerz
RU2011112445A (ru) * 2008-09-05 2012-10-10 Грюненталь ГмбХ (DE) Фармацевтическая комбинация, которая содержит 6-диметиламинометил-1-(3-метоксифенил)-циклогексан-1,3-диол и нпвс
US20100190752A1 (en) 2008-09-05 2010-07-29 Gruenenthal Gmbh Pharmaceutical Combination
BRPI0918566A2 (pt) * 2008-09-05 2016-02-10 Gruenenthal Gmbh combinacao farmacêutica compreendendo 6-dimetilanometil-1-(3-metóxifenil)-ciclo-hexano-1,3-diol e paracetamol
WO2010096045A1 (en) * 2008-10-30 2010-08-26 Nectid, Inc. Novel and potent tapentadol dosage forms
CA2757757C (en) * 2009-04-30 2017-10-24 Ulrich Jahnel Use of 1-phenyl-3-dimethylaminopropane compounds for treating rheumatoid pain
AR077987A1 (es) * 2009-08-28 2011-10-05 Gruenenthal Gmbh Combinacion farmaceutica que comprende 6-dimetilaminometil-1-(3-metoxifenil)-ciclohexano-1,3-diol o 6-dimetilaminometil-1-(3-hidroxifenil)-ciclohexano-1,3-diol y un antiepileptico
CN104276960B (zh) * 2014-09-26 2016-09-28 安徽省逸欣铭医药科技有限公司 盐酸他喷他多和塞来昔布共晶及其组合物和制备方法

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DK3241550T3 (da) 2002-11-22 2020-08-24 Gruenenthal Gmbh Anvendelse af (1r,2r)-3-(3-dimethylamino-1-ethyl-2-methyl-propyl)-phenol til behandling af inflammatoriske smerter

Also Published As

Publication number Publication date
US8404749B2 (en) 2013-03-26
US8420691B2 (en) 2013-04-16
SI1685829T1 (sl) 2008-08-31
DK1685829T3 (da) 2008-07-21
EP3241550A1 (de) 2017-11-08
ATE465726T1 (de) 2010-05-15
ES2640404T3 (es) 2017-11-02
ES2304659T3 (es) 2008-10-16
EP1908460A1 (de) 2008-04-09
ES2819854T3 (es) 2021-04-19
US10471079B2 (en) 2019-11-12
US8003701B2 (en) 2011-08-23
PT1839654E (pt) 2010-07-06
PT1562567T (pt) 2017-08-24
DE50309605D1 (de) 2008-05-21
DK1562567T3 (en) 2017-07-17
CY1119082T1 (el) 2018-01-10
US20100280129A1 (en) 2010-11-04
DE50312678D1 (de) 2010-06-10
SI1562567T1 (sl) 2017-09-29
US20100280017A1 (en) 2010-11-04
EP1562567B1 (de) 2017-06-14
EP1685829A1 (de) 2006-08-02
DK3241550T3 (da) 2020-08-24
EP1839654A2 (de) 2007-10-03
CY1123286T1 (el) 2021-12-31
US7786160B2 (en) 2010-08-31
AU2003283410A1 (en) 2004-06-18
CY1110246T1 (el) 2015-01-14
US20050277687A1 (en) 2005-12-15
US20130109733A1 (en) 2013-05-02
EP3241550B1 (de) 2020-07-22
US8618177B2 (en) 2013-12-31
PT1685829E (pt) 2008-05-15
EP1562567A1 (de) 2005-08-17
EP1685829B1 (de) 2008-04-09
US20070249724A1 (en) 2007-10-25
EP1839654B9 (de) 2012-01-11
ES2345062T3 (es) 2010-09-14
EP1839654A3 (de) 2007-11-07
HUE033042T2 (en) 2017-11-28
SI3241550T1 (sl) 2020-11-30
PT3241550T (pt) 2020-08-11
US20100280126A1 (en) 2010-11-04
DK1839654T3 (da) 2010-08-16
CY1108141T1 (el) 2014-04-09
SI1839654T1 (sl) 2010-08-31
US20160279150A1 (en) 2016-09-29
WO2004047823A1 (de) 2004-06-10
ATE391498T1 (de) 2008-04-15
HUE051024T2 (hu) 2021-03-01
EP1839654B1 (de) 2010-04-28
EP3662904A1 (de) 2020-06-10

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