KR930016091A - 거의 수불용성인 약제의 고체 분산액을 제조하는 방법 - Google Patents

거의 수불용성인 약제의 고체 분산액을 제조하는 방법 Download PDF

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Publication number
KR930016091A
KR930016091A KR1019930000603A KR930000603A KR930016091A KR 930016091 A KR930016091 A KR 930016091A KR 1019930000603 A KR1019930000603 A KR 1019930000603A KR 930000603 A KR930000603 A KR 930000603A KR 930016091 A KR930016091 A KR 930016091A
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South Korea
Prior art keywords
water
insoluble drug
solid dispersion
preparing
melted
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Withdrawn
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KR1019930000603A
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English (en)
Korean (ko)
Inventor
미노루 나카노
도시노부 우에무라
신이치 모리자네
기요시 오쿠다
게이코 나카타
Original Assignee
후지야마 아키라
후지사와야쿠힝코교가부시키가이샤
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Publication of KR930016091A publication Critical patent/KR930016091A/ko
Withdrawn legal-status Critical Current

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/146Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic macromolecular compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Dispersion Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
KR1019930000603A 1992-01-24 1993-01-19 거의 수불용성인 약제의 고체 분산액을 제조하는 방법 Withdrawn KR930016091A (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP1079692 1992-01-24
JP92-10796.0 1992-01-24

Publications (1)

Publication Number Publication Date
KR930016091A true KR930016091A (ko) 1993-08-26

Family

ID=11760311

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019930000603A Withdrawn KR930016091A (ko) 1992-01-24 1993-01-19 거의 수불용성인 약제의 고체 분산액을 제조하는 방법

Country Status (6)

Country Link
US (1) US5340591A (enExample)
EP (1) EP0552708A1 (enExample)
JP (1) JPH05262642A (enExample)
KR (1) KR930016091A (enExample)
CA (1) CA2087932A1 (enExample)
TW (1) TW259712B (enExample)

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EP0552708A1 (en) 1993-07-28
CA2087932A1 (en) 1993-07-25

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