KR830009112A - 페니실란산 1,1-디옥사이드의 할로메틸 에스테르(및 관련 에스테르)의 제조방법 - Google Patents

페니실란산 1,1-디옥사이드의 할로메틸 에스테르(및 관련 에스테르)의 제조방법 Download PDF

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Publication number
KR830009112A
KR830009112A KR1019820001222A KR820001222A KR830009112A KR 830009112 A KR830009112 A KR 830009112A KR 1019820001222 A KR1019820001222 A KR 1019820001222A KR 820001222 A KR820001222 A KR 820001222A KR 830009112 A KR830009112 A KR 830009112A
Authority
KR
South Korea
Prior art keywords
group
general formula
alkyl
acid
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
KR1019820001222A
Other languages
English (en)
Korean (ko)
Inventor
찰스 크라우포드 토마스
존 재시스 비타우타스
Original Assignee
윌리암 데이비스 헌
화이자 인코포레이티드
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 윌리암 데이비스 헌, 화이자 인코포레이티드 filed Critical 윌리암 데이비스 헌
Publication of KR830009112A publication Critical patent/KR830009112A/ko
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
KR1019820001222A 1981-03-23 1982-03-22 페니실란산 1,1-디옥사이드의 할로메틸 에스테르(및 관련 에스테르)의 제조방법 Abandoned KR830009112A (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US246453 1981-03-23
US06/246,453 US4419284A (en) 1981-03-23 1981-03-23 Preparation of halomethyl esters (and related esters) of penicillanic acid 1,1-dioxide

Publications (1)

Publication Number Publication Date
KR830009112A true KR830009112A (ko) 1983-12-17

Family

ID=22930753

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019820001222A Abandoned KR830009112A (ko) 1981-03-23 1982-03-22 페니실란산 1,1-디옥사이드의 할로메틸 에스테르(및 관련 에스테르)의 제조방법

Country Status (19)

Country Link
US (1) US4419284A (ref)
EP (1) EP0061315A1 (ref)
JP (1) JPS57169486A (ref)
KR (1) KR830009112A (ref)
AR (1) AR231292A1 (ref)
AU (1) AU527896B2 (ref)
CS (1) CS228919B2 (ref)
DK (1) DK127082A (ref)
ES (2) ES8305767A1 (ref)
FI (1) FI820994L (ref)
GB (1) GB2095667A (ref)
GR (1) GR76480B (ref)
IL (1) IL65307A0 (ref)
NO (1) NO820899L (ref)
PH (1) PH17749A (ref)
PL (2) PL239642A1 (ref)
PT (1) PT74620B (ref)
YU (1) YU62082A (ref)
ZA (1) ZA821902B (ref)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT76527B (en) * 1982-04-19 1985-12-09 Gist Brocades Nv A process for the preparation of penicillanic acid 1,1-dioxide and derivatives thereof
US5266693A (en) * 1982-04-19 1993-11-30 Gist-Brocades N.V. 6-diazo-penicillanic acid 1,1-dioxide derivatives
PH20068A (en) * 1982-12-06 1986-09-18 Pfizer Process and intermediates for sultamicillin and analogs
EP0139048A1 (en) * 1983-10-18 1985-05-02 Gist-Brocades N.V. Process for the dehalogenation of 6,6-dibromopenicillanic acid 1,1-dioxide
US4826833A (en) * 1984-01-30 1989-05-02 Pfizer Inc. 6-(Substituted)methylene-penicillanic and 6-(substituted)hydroxymethylpenicillanic acids and derivatives thereof
US5015473A (en) * 1984-01-30 1991-05-14 Pfizer Inc. 6-(substituted)methylenepenicillanic and 6-(substituted)hydroxymethylpenicillanic acids and derivatives thereof
EP0262202B1 (en) * 1986-04-10 1992-07-01 Leo Pharmaceutical Products Ltd. A/S (Lovens Kemiske Fabrik Produktionsaktieselskab) Method for preparing penicillanic acid derivatives
KR910009271B1 (ko) * 1989-06-20 1991-11-08 김영설 1,1-디옥소페닐실라노일 옥시메틸 D-6-[α-(메틸렌아미노)페닐-아세트아미도]-페니실라네이트와 그의 파라-톨루엔술폰산염
ES2039299B1 (es) * 1991-10-04 1994-05-16 Asturpharma S A Procedimiento de obtencion de esteres de acido 1,1-dioxopenicilanico y sus sales.
ES2100125B1 (es) * 1995-06-02 1998-04-01 Asturpharma S A Procedimiento de preparacion de esteres de metanodiol de acido dioxopenicilanico.
IT202000031070A1 (it) 2020-12-16 2022-06-16 Paolo Bonomi Procedimento di sintesi di derivati ammidici dell’acido 8-idrossi penicillanico

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3996235A (en) * 1974-02-19 1976-12-07 Beecham Group Limited 6-Isocyanato-6-substituted penicillins
IN149747B (ref) * 1977-06-07 1982-04-03 Pfizer
JPS6056160B2 (ja) * 1977-06-07 1985-12-09 フアイザ−・インコ−ポレ−テツド β−ラクタマ−ゼ阻害剤としてのペニシラン酸１，１−ジオキシド
US4234579A (en) * 1977-06-07 1980-11-18 Pfizer Inc. Penicillanic acid 1,1-dioxides as β-lactamase inhibitors
US4224951A (en) * 1978-11-30 1980-09-30 Hasson Harrith M Gynecological instrument
US4203992A (en) * 1978-12-11 1980-05-20 E. R. Squibb & Sons, Inc. β-Bromopenicillanic acid sulfone
EP0013617B1 (en) * 1979-01-10 1984-07-04 Beecham Group Plc Penicillin derivatives, process for their preparation and pharmaceutical compositions containing certain of these compounds
JPS5598186A (en) * 1979-01-10 1980-07-25 Beecham Group Ltd Manufacture of penicillin derivative
IE49880B1 (en) 1979-02-13 1986-01-08 Leo Pharm Prod Ltd Penicillin derivatives
ZA80796B (en) * 1979-02-13 1981-02-25 Leo Pharm Prod Ltd Chemical compounds
SE449103B (sv) * 1979-03-05 1987-04-06 Pfizer Sett att framstella penicillansyra-1,1-dioxid samt estrar derav
ZA80646B (en) * 1979-03-05 1981-02-25 Pfizer Process and intermediates for penicillanic acid,1,1-dioxide and esters thereof

Also Published As

Publication number Publication date
ZA821902B (en) 1983-01-26
DK127082A (da) 1982-09-24
IL65307A0 (en) 1982-05-31
PT74620B (en) 1984-11-26
EP0061315A1 (en) 1982-09-29
FI820994A7 (fi) 1982-09-24
ES8403131A1 (es) 1984-03-01
ES518969A0 (es) 1984-03-01
JPS57169486A (en) 1982-10-19
US4419284A (en) 1983-12-06
ES510654A0 (es) 1983-04-16
PH17749A (en) 1984-11-27
PL235579A1 (en) 1983-06-06
AU527896B2 (en) 1983-03-31
YU62082A (en) 1985-03-20
AR231292A1 (es) 1984-10-31
ES8305767A1 (es) 1983-04-16
FI820994L (fi) 1982-09-24
CS228919B2 (en) 1984-05-14
GB2095667A (en) 1982-10-06
PT74620A (en) 1982-04-01
AU8176382A (en) 1982-11-04
PL239642A1 (en) 1983-08-15
GR76480B (ref) 1984-08-10
NO820899L (no) 1982-09-24

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Legal Events

Date Code Title Description
PA0109 Patent application

Patent event code: PA01091R01D

Comment text: Patent Application

Patent event date: 19820322

PG1501 Laying open of application
PE0902 Notice of grounds for rejection

Comment text: Notification of reason for refusal

Patent event date: 19851014

Patent event code: PE09021S01D

PC1902 Submission of document of abandonment before decision of registration