KR830009112A - 페니실란산 1,1-디옥사이드의 할로메틸 에스테르(및 관련 에스테르)의 제조방법 - Google Patents

페니실란산 1,1-디옥사이드의 할로메틸 에스테르(및 관련 에스테르)의 제조방법 Download PDF

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Publication number
KR830009112A
KR830009112A KR1019820001222A KR820001222A KR830009112A KR 830009112 A KR830009112 A KR 830009112A KR 1019820001222 A KR1019820001222 A KR 1019820001222A KR 820001222 A KR820001222 A KR 820001222A KR 830009112 A KR830009112 A KR 830009112A
Authority
KR
South Korea
Prior art keywords
group
general formula
alkyl
acid
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
KR1019820001222A
Other languages
English (en)
Korean (ko)
Inventor
찰스 크라우포드 토마스
존 재시스 비타우타스
Original Assignee
윌리암 데이비스 헌
화이자 인코포레이티드
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 윌리암 데이비스 헌, 화이자 인코포레이티드 filed Critical 윌리암 데이비스 헌
Publication of KR830009112A publication Critical patent/KR830009112A/ko
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
KR1019820001222A 1981-03-23 1982-03-22 페니실란산 1,1-디옥사이드의 할로메틸 에스테르(및 관련 에스테르)의 제조방법 Abandoned KR830009112A (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US246453 1981-03-23
US06/246,453 US4419284A (en) 1981-03-23 1981-03-23 Preparation of halomethyl esters (and related esters) of penicillanic acid 1,1-dioxide

Publications (1)

Publication Number Publication Date
KR830009112A true KR830009112A (ko) 1983-12-17

Family

ID=22930753

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019820001222A Abandoned KR830009112A (ko) 1981-03-23 1982-03-22 페니실란산 1,1-디옥사이드의 할로메틸 에스테르(및 관련 에스테르)의 제조방법

Country Status (19)

Country Link
US (1) US4419284A (en:Method)
EP (1) EP0061315A1 (en:Method)
JP (1) JPS57169486A (en:Method)
KR (1) KR830009112A (en:Method)
AR (1) AR231292A1 (en:Method)
AU (1) AU527896B2 (en:Method)
CS (1) CS228919B2 (en:Method)
DK (1) DK127082A (en:Method)
ES (2) ES8305767A1 (en:Method)
FI (1) FI820994L (en:Method)
GB (1) GB2095667A (en:Method)
GR (1) GR76480B (en:Method)
IL (1) IL65307A0 (en:Method)
NO (1) NO820899L (en:Method)
PH (1) PH17749A (en:Method)
PL (2) PL239642A1 (en:Method)
PT (1) PT74620B (en:Method)
YU (1) YU62082A (en:Method)
ZA (1) ZA821902B (en:Method)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT76527B (en) * 1982-04-19 1985-12-09 Gist Brocades Nv A process for the preparation of penicillanic acid 1,1-dioxide and derivatives thereof
US5266693A (en) * 1982-04-19 1993-11-30 Gist-Brocades N.V. 6-diazo-penicillanic acid 1,1-dioxide derivatives
PH20068A (en) * 1982-12-06 1986-09-18 Pfizer Process and intermediates for sultamicillin and analogs
EP0139048A1 (en) * 1983-10-18 1985-05-02 Gist-Brocades N.V. Process for the dehalogenation of 6,6-dibromopenicillanic acid 1,1-dioxide
US4826833A (en) * 1984-01-30 1989-05-02 Pfizer Inc. 6-(Substituted)methylene-penicillanic and 6-(substituted)hydroxymethylpenicillanic acids and derivatives thereof
US5015473A (en) * 1984-01-30 1991-05-14 Pfizer Inc. 6-(substituted)methylenepenicillanic and 6-(substituted)hydroxymethylpenicillanic acids and derivatives thereof
EP0262202B1 (en) * 1986-04-10 1992-07-01 Leo Pharmaceutical Products Ltd. A/S (Lovens Kemiske Fabrik Produktionsaktieselskab) Method for preparing penicillanic acid derivatives
KR910009271B1 (ko) * 1989-06-20 1991-11-08 김영설 1,1-디옥소페닐실라노일 옥시메틸 D-6-[α-(메틸렌아미노)페닐-아세트아미도]-페니실라네이트와 그의 파라-톨루엔술폰산염
ES2039299B1 (es) * 1991-10-04 1994-05-16 Asturpharma S A Procedimiento de obtencion de esteres de acido 1,1-dioxopenicilanico y sus sales.
ES2100125B1 (es) * 1995-06-02 1998-04-01 Asturpharma S A Procedimiento de preparacion de esteres de metanodiol de acido dioxopenicilanico.
IT202000031070A1 (it) 2020-12-16 2022-06-16 Paolo Bonomi Procedimento di sintesi di derivati ammidici dell’acido 8-idrossi penicillanico

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3996235A (en) * 1974-02-19 1976-12-07 Beecham Group Limited 6-Isocyanato-6-substituted penicillins
IN149747B (en:Method) * 1977-06-07 1982-04-03 Pfizer
JPS6056160B2 (ja) * 1977-06-07 1985-12-09 フアイザ−・インコ−ポレ−テツド β−ラクタマ−ゼ阻害剤としてのペニシラン酸１，１−ジオキシド
US4234579A (en) * 1977-06-07 1980-11-18 Pfizer Inc. Penicillanic acid 1,1-dioxides as β-lactamase inhibitors
US4224951A (en) * 1978-11-30 1980-09-30 Hasson Harrith M Gynecological instrument
US4203992A (en) * 1978-12-11 1980-05-20 E. R. Squibb & Sons, Inc. β-Bromopenicillanic acid sulfone
EP0013617B1 (en) * 1979-01-10 1984-07-04 Beecham Group Plc Penicillin derivatives, process for their preparation and pharmaceutical compositions containing certain of these compounds
JPS5598186A (en) * 1979-01-10 1980-07-25 Beecham Group Ltd Manufacture of penicillin derivative
IE49880B1 (en) 1979-02-13 1986-01-08 Leo Pharm Prod Ltd Penicillin derivatives
ZA80796B (en) * 1979-02-13 1981-02-25 Leo Pharm Prod Ltd Chemical compounds
SE449103B (sv) * 1979-03-05 1987-04-06 Pfizer Sett att framstella penicillansyra-1,1-dioxid samt estrar derav
ZA80646B (en) * 1979-03-05 1981-02-25 Pfizer Process and intermediates for penicillanic acid,1,1-dioxide and esters thereof

Also Published As

Publication number Publication date
ZA821902B (en) 1983-01-26
DK127082A (da) 1982-09-24
IL65307A0 (en) 1982-05-31
PT74620B (en) 1984-11-26
EP0061315A1 (en) 1982-09-29
FI820994A7 (fi) 1982-09-24
ES8403131A1 (es) 1984-03-01
ES518969A0 (es) 1984-03-01
JPS57169486A (en) 1982-10-19
US4419284A (en) 1983-12-06
ES510654A0 (es) 1983-04-16
PH17749A (en) 1984-11-27
PL235579A1 (en) 1983-06-06
AU527896B2 (en) 1983-03-31
YU62082A (en) 1985-03-20
AR231292A1 (es) 1984-10-31
ES8305767A1 (es) 1983-04-16
FI820994L (fi) 1982-09-24
CS228919B2 (en) 1984-05-14
GB2095667A (en) 1982-10-06
PT74620A (en) 1982-04-01
AU8176382A (en) 1982-11-04
PL239642A1 (en) 1983-08-15
GR76480B (en:Method) 1984-08-10
NO820899L (no) 1982-09-24

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Legal Events

Date Code Title Description
PA0109 Patent application

Patent event code: PA01091R01D

Comment text: Patent Application

Patent event date: 19820322

PG1501 Laying open of application
PE0902 Notice of grounds for rejection

Comment text: Notification of reason for refusal

Patent event date: 19851014

Patent event code: PE09021S01D

PC1902 Submission of document of abandonment before decision of registration