KR20190109590A - 선택적인 bcl­2 억제제를 사용하는 치료 방법 - Google Patents

선택적인 bcl­2 억제제를 사용하는 치료 방법 Download PDF

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KR20190109590A
KR20190109590A KR1020197027331A KR20197027331A KR20190109590A KR 20190109590 A KR20190109590 A KR 20190109590A KR 1020197027331 A KR1020197027331 A KR 1020197027331A KR 20197027331 A KR20197027331 A KR 20197027331A KR 20190109590 A KR20190109590 A KR 20190109590A
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methyl
chlorophenyl
sulfonyl
dimethylcyclohex
piperazin
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Korean (ko)
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스티븐 엘모어
앤드류 사우어스
리 춘 왕
타리크 가유르
스튜어트 제이. 퍼퍼
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애브비 아일랜드 언리미티드 컴퍼니
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/53751,4-Oxazines, e.g. morpholine
    • A61K31/53771,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/12Drugs for disorders of the urinary system of the kidneys
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Immunology (AREA)
  • Urology & Nephrology (AREA)
  • Transplantation (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
KR1020197027331A 2010-11-23 2011-11-22 선택적인 bcl­2 억제제를 사용하는 치료 방법 Withdrawn KR20190109590A (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US41668910P 2010-11-23 2010-11-23
US61/416,689 2010-11-23
PCT/US2011/061769 WO2012071374A1 (en) 2010-11-23 2011-11-22 Methods of treatment using selective bcl-2 inhibitors

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KR1020187007228A Division KR20180030257A (ko) 2010-11-23 2011-11-22 선택적인 bcl­2 억제제를 사용하는 치료 방법

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KR20190109590A true KR20190109590A (ko) 2019-09-25

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KR1020197027331A Withdrawn KR20190109590A (ko) 2010-11-23 2011-11-22 선택적인 bcl­2 억제제를 사용하는 치료 방법
KR1020187007228A Ceased KR20180030257A (ko) 2010-11-23 2011-11-22 선택적인 bcl­2 억제제를 사용하는 치료 방법
KR1020137016217A Expired - Fee Related KR101841084B1 (ko) 2010-11-23 2011-11-22 선택적인 bcl­2 억제제를 사용하는 치료 방법

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KR1020187007228A Ceased KR20180030257A (ko) 2010-11-23 2011-11-22 선택적인 bcl­2 억제제를 사용하는 치료 방법
KR1020137016217A Expired - Fee Related KR101841084B1 (ko) 2010-11-23 2011-11-22 선택적인 bcl­2 억제제를 사용하는 치료 방법

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AU (2) AU2011332000B2 (enExample)
BR (1) BR112013012854B1 (enExample)
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DK (1) DK2642999T3 (enExample)
DO (1) DOP2017000056A (enExample)
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NZ (2) NZ708508A (enExample)
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PT (1) PT2642999T (enExample)
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RU (1) RU2593231C2 (enExample)
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SI (1) SI2642999T1 (enExample)
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UA (2) UA113157C2 (enExample)
UY (1) UY33746A (enExample)
WO (1) WO2012071374A1 (enExample)
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