BR112013012854A8 - métodos de tratamento usando os inibidores de bcl-2 seletivos - Google Patents

métodos de tratamento usando os inibidores de bcl-2 seletivos

Info

Publication number
BR112013012854A8
BR112013012854A8 BR112013012854A BR112013012854A BR112013012854A8 BR 112013012854 A8 BR112013012854 A8 BR 112013012854A8 BR 112013012854 A BR112013012854 A BR 112013012854A BR 112013012854 A BR112013012854 A BR 112013012854A BR 112013012854 A8 BR112013012854 A8 BR 112013012854A8
Authority
BR
Brazil
Prior art keywords
inhibitors
treatment methods
selective bcl
bcl
selective
Prior art date
Application number
BR112013012854A
Other languages
English (en)
Other versions
BR112013012854A2 (pt
BR112013012854B1 (pt
Inventor
Souers Andrew
Chun Wang Li
Elmore Steven
J Perper Stuart
Ghayur Tariq
Original Assignee
Abbvie Bahamas Ltd
Abbvie Inc
Abbvie Ireland Unlimited Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=45218888&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR112013012854(A8) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Abbvie Bahamas Ltd, Abbvie Inc, Abbvie Ireland Unlimited Co filed Critical Abbvie Bahamas Ltd
Publication of BR112013012854A2 publication Critical patent/BR112013012854A2/pt
Publication of BR112013012854A8 publication Critical patent/BR112013012854A8/pt
Publication of BR112013012854B1 publication Critical patent/BR112013012854B1/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Immunology (AREA)
  • Urology & Nephrology (AREA)
  • Transplantation (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
BR112013012854-2A 2010-11-23 2011-11-22 Composições farmacêuticas compreendendo inibidores de bcl-2 seletivos BR112013012854B1 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US41668910P 2010-11-23 2010-11-23
US61/416,689 2010-11-23
PCT/US2011/061769 WO2012071374A1 (en) 2010-11-23 2011-11-22 Methods of treatment using selective bcl-2 inhibitors

Publications (3)

Publication Number Publication Date
BR112013012854A2 BR112013012854A2 (pt) 2016-08-23
BR112013012854A8 true BR112013012854A8 (pt) 2018-01-16
BR112013012854B1 BR112013012854B1 (pt) 2019-08-06

Family

ID=45218888

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112013012854-2A BR112013012854B1 (pt) 2010-11-23 2011-11-22 Composições farmacêuticas compreendendo inibidores de bcl-2 seletivos

Country Status (36)

Country Link
US (5) US20120129853A1 (pt)
EP (2) EP3028702B1 (pt)
JP (2) JP5876067B2 (pt)
KR (3) KR101841084B1 (pt)
CN (2) CN103402521B (pt)
AR (1) AR083946A1 (pt)
AU (2) AU2011332000B2 (pt)
BR (1) BR112013012854B1 (pt)
CA (1) CA2820618C (pt)
CL (1) CL2013001458A1 (pt)
CR (1) CR20130268A (pt)
CY (1) CY1118442T1 (pt)
DK (1) DK2642999T3 (pt)
DO (1) DOP2017000056A (pt)
EC (1) ECSP13012710A (pt)
ES (2) ES2603129T3 (pt)
GT (1) GT201300136A (pt)
HR (1) HRP20161762T1 (pt)
HU (1) HUE031267T2 (pt)
IL (2) IL226490A (pt)
LT (1) LT2642999T (pt)
MX (1) MX346201B (pt)
MY (2) MY191300A (pt)
NZ (2) NZ610746A (pt)
PH (1) PH12016500939B1 (pt)
PL (1) PL2642999T3 (pt)
PT (1) PT2642999T (pt)
RS (1) RS55545B1 (pt)
RU (1) RU2593231C2 (pt)
SG (2) SG190399A1 (pt)
SI (1) SI2642999T1 (pt)
TW (2) TWI535701B (pt)
UA (2) UA119150C2 (pt)
UY (1) UY33746A (pt)
WO (1) WO2012071374A1 (pt)
ZA (1) ZA201303589B (pt)

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