KR20160033697A - 치환된 퀴나졸린-4-온 유도체 - Google Patents

치환된 퀴나졸린-4-온 유도체 Download PDF

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KR20160033697A
KR20160033697A KR1020167001639A KR20167001639A KR20160033697A KR 20160033697 A KR20160033697 A KR 20160033697A KR 1020167001639 A KR1020167001639 A KR 1020167001639A KR 20167001639 A KR20167001639 A KR 20167001639A KR 20160033697 A KR20160033697 A KR 20160033697A
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formula
compound
fluoro
substituted
methyl
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전싱 두
사무엘 힌터만
콘스탄츠 허트
세바스티앵 자키에
한스요르크 레만
헨리크 뫼비츠
니콜라스 솔더만
알렉산다르 스토야노비치
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노파르티스 아게
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    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52—Purines, e.g. adenine
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    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
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    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
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  • Neurology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Vascular Medicine (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Cardiology (AREA)
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  • Rheumatology (AREA)
  • Biomedical Technology (AREA)
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  • Otolaryngology (AREA)
  • Transplantation (AREA)
  • Urology & Nephrology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
KR1020167001639A 2013-07-24 2014-07-24 치환된 퀴나졸린-4-온 유도체 Ceased KR20160033697A (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP13177827.6 2013-07-24
EP13177827 2013-07-24
PCT/CN2014/082946 WO2015010641A1 (en) 2013-07-24 2014-07-24 Substituted quinazolin-4-one derivatives

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KR20160033697A true KR20160033697A (ko) 2016-03-28

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Country Link
US (1) US9840498B2 (https=)
EP (1) EP3024827B1 (https=)
JP (1) JP6437544B2 (https=)
KR (1) KR20160033697A (https=)
CN (1) CN105452235B (https=)
AR (1) AR097024A1 (https=)
AU (1) AU2014295538B2 (https=)
CA (1) CA2917433A1 (https=)
EA (1) EA031430B1 (https=)
ES (1) ES2803513T3 (https=)
MX (1) MX368066B (https=)
PL (1) PL3024827T3 (https=)
PT (1) PT3024827T (https=)
TW (1) TW201534598A (https=)
UY (1) UY35675A (https=)
WO (1) WO2015010641A1 (https=)

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