KR20120105449A - 오렉신 수용체 조절제로서의 이치환된 옥타하이드로피롤로［3,4-ｃ］피롤 - Google Patents

오렉신 수용체 조절제로서의 이치환된 옥타하이드로피롤로［3,4-ｃ］피롤 Download PDF

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KR20120105449A
KR20120105449A KR1020127013101A KR20127013101A KR20120105449A KR 20120105449 A KR20120105449 A KR 20120105449A KR 1020127013101 A KR1020127013101 A KR 1020127013101A KR 20127013101 A KR20127013101 A KR 20127013101A KR 20120105449 A KR20120105449 A KR 20120105449A
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South Korea
Prior art keywords
pyrrole
phenyl
triazol
carbonyl
fluoro
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Korean (ko)
Inventor
웨닝 차이
마이클 에이. 레타빅
키브 에스. 라이
다니엘 제이. 피펠
데일 에이. 루돌프
캐슬린 씨. 스트로더
브래드 엠. 사발
챈드라바댄 알. 샤
브락 티. 셔먼
아키놀라 소요데-존슨
에밀리 엠. 스톡킹
데빈 엠. 스완슨
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얀센 파마슈티카 엔.브이.
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
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KR1020127013101A 2009-10-23 2010-10-21 오렉신 수용체 조절제로서의 이치환된 옥타하이드로피롤로［3,4-ｃ］피롤 Withdrawn KR20120105449A (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US25450909P 2009-10-23 2009-10-23
US61/254,509 2009-10-23

Related Child Applications (2)

Application Number Title Priority Date Filing Date
KR1020177034281A Division KR101859409B1 (ko) 2009-10-23 2010-10-21 오렉신 수용체 조절제로서의 이치환된 옥타하이드로피롤로［3,4-ｃ］피롤
KR1020177034279A Division KR101859400B1 (ko) 2009-10-23 2010-10-21 오렉신 수용체 조절제로서의 이치환된 옥타하이드로피롤로［3,4-ｃ］피롤

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KR20120105449A true KR20120105449A (ko) 2012-09-25

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KR1020177034281A Active KR101859409B1 (ko) 2009-10-23 2010-10-21 오렉신 수용체 조절제로서의 이치환된 옥타하이드로피롤로［3,4-ｃ］피롤
KR1020177034279A Active KR101859400B1 (ko) 2009-10-23 2010-10-21 오렉신 수용체 조절제로서의 이치환된 옥타하이드로피롤로［3,4-ｃ］피롤
KR1020127013101A Withdrawn KR20120105449A (ko) 2009-10-23 2010-10-21 오렉신 수용체 조절제로서의 이치환된 옥타하이드로피롤로［3,4-ｃ］피롤

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KR1020177034281A Active KR101859409B1 (ko) 2009-10-23 2010-10-21 오렉신 수용체 조절제로서의 이치환된 옥타하이드로피롤로［3,4-ｃ］피롤
KR1020177034279A Active KR101859400B1 (ko) 2009-10-23 2010-10-21 오렉신 수용체 조절제로서의 이치환된 옥타하이드로피롤로［3,4-ｃ］피롤

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Cited By (2)

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