KR20020063292A - N-(5,7-디메톡시[1,2,4]트리아졸로[1,5-a]피리미딘-2-일)아릴설폰아미드 화합물 및 제초제로서의 이의 용도 - Google Patents
N-(5,7-디메톡시[1,2,4]트리아졸로[1,5-a]피리미딘-2-일)아릴설폰아미드 화합물 및 제초제로서의 이의 용도 Download PDFInfo
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- KR20020063292A KR20020063292A KR1020027008656A KR20027008656A KR20020063292A KR 20020063292 A KR20020063292 A KR 20020063292A KR 1020027008656 A KR1020027008656 A KR 1020027008656A KR 20027008656 A KR20027008656 A KR 20027008656A KR 20020063292 A KR20020063292 A KR 20020063292A
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
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- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
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- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Health & Medical Sciences (AREA)
- Plant Pathology (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- General Health & Medical Sciences (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Pest Control & Pesticides (AREA)
- Agronomy & Crop Science (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Abstract
Description
Claims (10)
- 화학식 I의 N-(5,7-디메톡시[1,2,4]트리아졸로[1,5-a]피리미딘-2-일)아릴설폰아미드 화합물, 및 T가 H인 경우 이의 농업적으로 허용되는 염.화학식 I상기 화학식 I에 있어서,Q는 N 또는 C-H를 나타내고;A 및 B는 독립적으로 H, 할로, R, OR' 또는 CO2R"를 나타내고, 단 A 및 B가 둘다 H는 아니어야 하며;D는 H, 할로 또는 R을 나타내고;T는 H, SO2R", C(O)R", C(O)OR", C(O)NR"2또는 CH2CH2C(O)OR"을 나타내며;R은 각각 플루오로 치환체를 최대의 가능한 수까지 임의로 갖는 C1-C3알킬을 나타내고;R'는 각각 플루오로 치환체를 최대의 가능한 수까지 임의로 갖는 C1-C4알킬, C3-C4알케닐 또는 C3-C4알키닐을 나타내고;R"은 H 또는 C1-C4알킬을 나타낸다.
- 제1항에 있어서, T가 H인 화합물 또는 이의 농업적으로 허용되는 염.
- 제2항에 있어서, Q가 N인 화합물.
- 제2항에 있어서, Q가 CH인 화합물.
- 제1항 내지 제4항 중 어느 한 항에 있어서, A 또는 B 중 어느 하나가 OCH3이고, A 또는 B 중 다른 하나가 할로, R, OR' 또는 CO2R"이며, D가 H인 화합물.
- 제1항 내지 제4항 중 어느 한 항에 있어서, A가 OCH3이고, B가 H이며, D가 H, CH3또는 Cl인 화합물.
- 제1항 내지 제4항 중 어느 한 항에 있어서, A가 할로, R, OR' 또는 CO2R"이고, B가 CF3이며, D가 H인 화합물.
- 농업적으로 허용되는 보조제 또는 담체와 배합된 제1항 내지 제7항 중 어느한 항의 화합물의 제초량을 포함하는 조성물.
- 제1항 내지 제7항 중 어느 한 항의 화합물의 제초 유효량을 식물 또는 이들의 서식지에 적용하는 것을 포함하여, 원치 않는 식물을 조절하는 방법.
- 무수 조건 하의 극성, 비양성자성 용매 중에서 하기 화학식 II의 화합물을 하기 화학식 III의 아릴설포닐 클로라이드 화합물과 혼합하고, 염기로서 피리딘, 및 디메틸 설폭사이드의 촉매량을 첨가함을 포함하는, 화학식 I의 N-(5,7-디메톡시[1,2,4]트리아졸로[1,5-a]피리미딘-2-일)아릴설폰아미드 화합물의 제조 방법.화학식 I화학식 II화학식 III상기 화학식 I 및 III에 있어서,Q는 N 또는 C-H를 나타내고;A 및 B는 독립적으로 H, 할로, R, OR' 또는 CO2R"를 나타내고, 단 A 및 B가 둘다 H는 아니어야 하며;D는 H, 할로 또는 R을 나타내고;T는 H, SO2R", C(O)R", C(O)OR", C(O)NR"2또는 CH2CH2C(O)OR"을 나타내고;R은 각각 플루오로 치환체를 최대의 가능한 수까지 임의로 갖는 C1-C3알킬을 나타내고;R'는 각각 플루오로 치환체를 최대의 가능한 수까지 임의로 갖는 C1-C4알킬, C3-C4알케닐 또는 C3-C4알키닐을 나타내고;R"은 H 또는 C1-C4알킬을 나타낸다.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US24583600P | 2000-11-03 | 2000-11-03 | |
US60/245,836 | 2000-11-03 | ||
PCT/US2001/046150 WO2002036595A2 (en) | 2000-11-03 | 2001-11-02 | N-(5,7-DIMETHOXY[1,2,4]TRIAZOLO[1,5-a]PYRIMIDIN-2-YL) ARYLSULFONAMIDE COMPOUNDS AND THEIR USE AS HERBICIDES |
Publications (2)
Publication Number | Publication Date |
---|---|
KR20020063292A true KR20020063292A (ko) | 2002-08-01 |
KR100467128B1 KR100467128B1 (ko) | 2005-01-24 |
Family
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Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
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KR10-2002-7008656A KR100467128B1 (ko) | 2000-11-03 | 2001-11-02 | N-(5,7-디메톡시[1,2,4]트리아졸로[1,5-a]피리미딘-2-일)아릴설폰아미드 화합물 및 제초제로서의 이의 용도 |
Country Status (29)
Country | Link |
---|---|
US (1) | US6559101B2 (ko) |
EP (1) | EP1242425B1 (ko) |
JP (1) | JP3911236B2 (ko) |
KR (1) | KR100467128B1 (ko) |
CN (1) | CN1262552C (ko) |
AR (1) | AR035209A1 (ko) |
AT (1) | ATE260917T1 (ko) |
AU (1) | AU780115B2 (ko) |
BG (1) | BG65806B1 (ko) |
BR (1) | BRPI0107403B8 (ko) |
CA (1) | CA2395050C (ko) |
CZ (1) | CZ300942B6 (ko) |
DE (2) | DE60102215T2 (ko) |
DK (1) | DK1242425T3 (ko) |
EA (1) | EA004941B1 (ko) |
ES (1) | ES2213124T3 (ko) |
FR (1) | FR09C0056I2 (ko) |
HU (1) | HU227229B1 (ko) |
IL (2) | IL150493A0 (ko) |
MX (1) | MX226072B (ko) |
NL (1) | NL350045I1 (ko) |
PL (1) | PL208906B1 (ko) |
PT (1) | PT1242425E (ko) |
RO (1) | RO121339B1 (ko) |
SK (1) | SK286484B6 (ko) |
TR (1) | TR200400746T4 (ko) |
UA (1) | UA66952C2 (ko) |
WO (1) | WO2002036595A2 (ko) |
ZA (1) | ZA200205097B (ko) |
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- 2001-11-02 MX MXPA02006640 patent/MX226072B/es active IP Right Grant
- 2001-11-02 HU HU0204346A patent/HU227229B1/hu active Protection Beyond IP Right Term
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