KR20010108025A - 5ＨＴ2Ｃ 효능제인2,3,4,4ａ-테트라하이드로-1Ｈ-피라지노(1,2-ａ)퀴녹살린-5(6Ｈ)온 유도체 - Google Patents

5ＨＴ2Ｃ 효능제인2,3,4,4ａ-테트라하이드로-1Ｈ-피라지노(1,2-ａ)퀴녹살린-5(6Ｈ)온 유도체 Download PDF

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KR20010108025A
KR20010108025A KR1020017007583A KR20017007583A KR20010108025A KR 20010108025 A KR20010108025 A KR 20010108025A KR 1020017007583 A KR1020017007583 A KR 1020017007583A KR 20017007583 A KR20017007583 A KR 20017007583A KR 20010108025 A KR20010108025 A KR 20010108025A
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South Korea
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carbon atoms
alkyl
formula
hydrogen
compound
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KR1020017007583A
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English (en)
Korean (ko)
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사브앤마리루이스
웰메이커그레고리스코트
넬슨제임스앨버트
Original Assignee
이곤 이 버그
아메리칸 홈 푸로닥츠 코포레이션
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Publication of KR20010108025A publication Critical patent/KR20010108025A/ko

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Diabetes (AREA)
  • Pain & Pain Management (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Psychiatry (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Anesthesiology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
KR1020017007583A 1998-12-17 1999-12-16 5ＨＴ2Ｃ 효능제인2,3,4,4ａ-테트라하이드로-1Ｈ-피라지노(1,2-ａ)퀴녹살린-5(6Ｈ)온 유도체 KR20010108025A (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US21347198A 1998-12-17 1998-12-17
US09/213,471 1998-12-17
PCT/US1999/029894 WO2000035922A1 (en) 1998-12-17 1999-12-16 2,3,4,4a-tetrahydro-1h-pyrazino(1,2-a)quinoxalin-5(6h)one derivates being 5ht2c agonists

Publications (1)

Publication Number Publication Date
KR20010108025A true KR20010108025A (ko) 2001-12-07

Family

ID=22795247

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020017007583A KR20010108025A (ko) 1998-12-17 1999-12-16 5ＨＴ2Ｃ 효능제인2,3,4,4ａ-테트라하이드로-1Ｈ-피라지노(1,2-ａ)퀴녹살린-5(6Ｈ)온 유도체

Country Status (18)

Country Link
EP (1) EP1140940A1 (ru)
JP (1) JP2002532504A (ru)
KR (1) KR20010108025A (ru)
CN (1) CN1240701C (ru)
AR (1) AR022687A1 (ru)
AU (1) AU3123400A (ru)
BR (1) BR9916326A (ru)
CA (1) CA2351385A1 (ru)
CZ (1) CZ20012193A3 (ru)
EA (1) EA200100671A1 (ru)
HU (1) HUP0104773A3 (ru)
IL (1) IL143323A0 (ru)
NO (1) NO20013001D0 (ru)
NZ (1) NZ512765A (ru)
PL (1) PL348815A1 (ru)
SK (1) SK8192001A3 (ru)
WO (1) WO2000035922A1 (ru)
ZA (1) ZA200104598B (ru)

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AR031199A1 (es) 2000-11-03 2003-09-10 Wyeth Corp Ciclohepta/b//1,4/diacepino/6,7,1-hi/indoles y derivados
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MXPA03010806A (es) 2001-06-01 2004-11-22 Alcon Inc Nuevos analogos de arilaminopropano y su uso para el tratamiento de glaucoma.
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TWI312781B (en) 2002-04-25 2009-08-01 [1,4]diazepino[6,7,1-ij]quinoline derivatives as antipsychotic and antiobesity agents
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BR0316775A (pt) 2002-12-13 2005-11-01 Alcon Inc Novos análogos de benzopirano e seu uso para o tratamento de glaucoma
ATE509929T1 (de) 2002-12-19 2011-06-15 Bristol Myers Squibb Co Substituierte tricyclische gamma-carbolineals serotonin-rezeptor-agonisten und antagonisten
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Also Published As

Publication number Publication date
HUP0104773A2 (hu) 2002-04-29
BR9916326A (pt) 2001-10-02
IL143323A0 (en) 2002-04-21
EP1140940A1 (en) 2001-10-10
ZA200104598B (en) 2002-09-05
NO20013001L (no) 2001-06-15
CZ20012193A3 (cs) 2001-12-12
PL348815A1 (en) 2002-06-17
CN1240701C (zh) 2006-02-08
WO2000035922A1 (en) 2000-06-22
AU3123400A (en) 2000-07-03
HUP0104773A3 (en) 2004-10-28
CA2351385A1 (en) 2000-06-22
EA200100671A1 (ru) 2001-12-24
NO20013001D0 (no) 2001-06-15
NZ512765A (en) 2003-10-31
AR022687A1 (es) 2002-09-04
JP2002532504A (ja) 2002-10-02
CN1330652A (zh) 2002-01-09
SK8192001A3 (en) 2001-12-03

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