BR0316775A - Novos análogos de benzopirano e seu uso para o tratamento de glaucoma - Google Patents

Novos análogos de benzopirano e seu uso para o tratamento de glaucoma

Info

Publication number
BR0316775A
BR0316775A BR0316775-5A BR0316775A BR0316775A BR 0316775 A BR0316775 A BR 0316775A BR 0316775 A BR0316775 A BR 0316775A BR 0316775 A BR0316775 A BR 0316775A
Authority
BR
Brazil
Prior art keywords
analogues
treating glaucoma
new benzopyran
new
benzopyran
Prior art date
Application number
BR0316775-5A
Other languages
English (en)
Inventor
Mark R Hellberg
Abdelmoula Namil
Original Assignee
Alcon Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Alcon Inc filed Critical Alcon Inc
Publication of BR0316775A publication Critical patent/BR0316775A/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
    • A61K31/353—3,4-Dihydrobenzopyrans, e.g. chroman, catechin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/76—Benzo[c]pyrans

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrane Compounds (AREA)

Abstract

"NOVOS ANáLOGOS DE BENZOPIRANO E SEU USO PARA O TRATAMENTO DE GLAUCOMA". Divulgam-se novos análogos de benzopirano. Divulgam-se também métodos para diminuir e controlar pressão intra-ocular elevada ou normal assim como um método para o tratamento de glaucoma usando composições contendo um ou mais compostos da invenção presente.
BR0316775-5A 2002-12-13 2003-12-12 Novos análogos de benzopirano e seu uso para o tratamento de glaucoma BR0316775A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US43346802P 2002-12-13 2002-12-13
PCT/US2003/039751 WO2004054572A2 (en) 2002-12-13 2003-12-12 Novel benzopyran analogs and their use for the treatment of glaucoma

Publications (1)

Publication Number Publication Date
BR0316775A true BR0316775A (pt) 2005-11-01

Family

ID=32595196

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0316775-5A BR0316775A (pt) 2002-12-13 2003-12-12 Novos análogos de benzopirano e seu uso para o tratamento de glaucoma

Country Status (9)

Country Link
US (1) US7396856B2 (pt)
EP (1) EP1581209A4 (pt)
JP (1) JP2006511556A (pt)
AU (1) AU2003300915B2 (pt)
BR (1) BR0316775A (pt)
CA (1) CA2506204A1 (pt)
MX (1) MXPA05006277A (pt)
WO (1) WO2004054572A2 (pt)
ZA (1) ZA200504145B (pt)

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WO2004054572A2 (en) 2002-12-13 2004-07-01 Alcon, Inc. Novel benzopyran analogs and their use for the treatment of glaucoma
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TW200520760A (en) 2003-12-15 2005-07-01 Alcon Inc Substituted [1,4] oxazino [2,3-g] indazoles for the treatment of glaucoma
US7129257B1 (en) 2003-12-15 2006-10-31 Alcon, Inc. Pyrazolo[3,4- e]benzoxazoles for the treatment of glaucoma
WO2006062839A1 (en) 2004-12-08 2006-06-15 Alcon, Inc. Use of dioxindoindazoles and dioxoloindazoles for treating glaucoma
TW200744567A (en) * 2005-09-23 2007-12-16 Alcon Inc Phenylethylamine analogs and their use for treating glaucoma
US20070293475A1 (en) * 2006-06-20 2007-12-20 Alcon Manufacturing Ltd. Aryl and heteroaryl tetrahydrobenzazepine derivatives and their use for treating glaucoma

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Also Published As

Publication number Publication date
JP2006511556A (ja) 2006-04-06
AU2003300915B2 (en) 2008-08-28
MXPA05006277A (es) 2005-09-08
ZA200504145B (en) 2006-07-26
WO2004054572A2 (en) 2004-07-01
US20050209314A1 (en) 2005-09-22
EP1581209A2 (en) 2005-10-05
US7396856B2 (en) 2008-07-08
CA2506204A1 (en) 2004-07-01
AU2003300915A1 (en) 2004-07-09
EP1581209A4 (en) 2009-03-11
WO2004054572A3 (en) 2004-08-26

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE 7A. E 8A. ANUIDADE(S),

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2129 DE 25/10/2011.