KR100955589B1 - 신규한 디하이드로프테리디논, 이의 제조방법 및 이를 함유하는 약제학적 조성물 - Google Patents

신규한 디하이드로프테리디논, 이의 제조방법 및 이를 함유하는 약제학적 조성물 Download PDF

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KR100955589B1
KR100955589B1 KR1020047003248A KR20047003248A KR100955589B1 KR 100955589 B1 KR100955589 B1 KR 100955589B1 KR 1020047003248 A KR1020047003248 A KR 1020047003248A KR 20047003248 A KR20047003248 A KR 20047003248A KR 100955589 B1 KR100955589 B1 KR 100955589B1
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formula
hydrogen
compound
substituted
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KR20040029465A (ko
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호프만맛티아스
그라우에르트맛티아스
브라이트펠더슈테펜
아이크마이어크리스티안
폴게랄트
레만-린츠토르스텐
레데만노르베르트
슈나프기젤라
슈테그마이어마르틴
바우어에크하르트
크반트옌스위르겐
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베링거 잉겔하임 파르마 게엠베하 운트 코 카게
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Virology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • AIDS & HIV (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Transplantation (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
KR1020047003248A 2001-09-04 2002-08-30 신규한 디하이드로프테리디논, 이의 제조방법 및 이를 함유하는 약제학적 조성물 Expired - Fee Related KR100955589B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE10143272.0 2001-09-04
DE10143272 2001-09-04
PCT/EP2002/009728 WO2003020722A1 (de) 2001-09-04 2002-08-30 Neue dihydropteridinone, verfahren zu deren herstellung und deren verwendung als arzneimittel

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KR20040029465A KR20040029465A (ko) 2004-04-06
KR100955589B1 true KR100955589B1 (ko) 2010-04-30

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EP (1) EP1427730B1 (https=)
JP (1) JP3876254B2 (https=)
KR (1) KR100955589B1 (https=)
CN (1) CN1551881A (https=)
AR (1) AR036586A1 (https=)
AT (1) ATE332898T1 (https=)
AU (1) AU2002337047B2 (https=)
BR (1) BRPI0212137A2 (https=)
CA (1) CA2458699C (https=)
CO (1) CO5560575A2 (https=)
CY (1) CY1105337T1 (https=)
DE (1) DE50207522D1 (https=)
DK (1) DK1427730T3 (https=)
EA (1) EA007062B1 (https=)
EC (1) ECSP045003A (https=)
ES (1) ES2268093T3 (https=)
HR (1) HRP20040213A2 (https=)
HU (1) HUP0401293A3 (https=)
IL (2) IL160440A0 (https=)
MX (1) MXPA04002067A (https=)
MY (1) MY129751A (https=)
NO (1) NO328804B1 (https=)
NZ (1) NZ531928A (https=)
PL (1) PL369740A1 (https=)
PT (1) PT1427730E (https=)
RS (1) RS51012B (https=)
UA (1) UA76512C2 (https=)
UY (1) UY27427A1 (https=)
WO (1) WO2003020722A1 (https=)
ZA (1) ZA200401365B (https=)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR101221864B1 (ko) 2004-08-14 2013-01-14 베링거 인겔하임 인터내셔날 게엠베하 4-［［(7ｒ)-8-사이클로펜틸-7-에틸-5,6,7,8-테트라하이드로-5-메틸-6-옥소-2-프테리디닐］아미노］-3-메톡시-ｎ-(1-메틸-4-피페리디닐)벤즈아미드의 수화물 및 다형체, 이들의 제조방법, 및 약제로서의 이들의 용도

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