KR100869616B1 - 프롤린 유도체 및 그의 다이펩티딜 펩티다제-iv저해제로서의 용도 - Google Patents

프롤린 유도체 및 그의 다이펩티딜 펩티다제-iv저해제로서의 용도 Download PDF

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KR100869616B1
KR100869616B1 KR1020067023663A KR20067023663A KR100869616B1 KR 100869616 B1 KR100869616 B1 KR 100869616B1 KR 1020067023663 A KR1020067023663 A KR 1020067023663A KR 20067023663 A KR20067023663 A KR 20067023663A KR 100869616 B1 KR100869616 B1 KR 100869616B1
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pyrrolidin
methanone
compound
alkyl
compounds
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KR20070009699A (ko
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베르나드 휼린
데이비드 왈터 피오트로스키
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화이자 프로덕츠 인코포레이티드
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KR1020067023663A 2004-05-12 2005-04-29 프롤린 유도체 및 그의 다이펩티딜 펩티다제-iv저해제로서의 용도 Expired - Fee Related KR100869616B1 (ko)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US57030004P 2004-05-12 2004-05-12
US60/570,300 2004-05-12
US66430505P 2005-03-21 2005-03-21
US60/664,305 2005-03-21

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KR20070009699A KR20070009699A (ko) 2007-01-18
KR100869616B1 true KR100869616B1 (ko) 2008-11-21

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US (4) US7291618B2 (https=)
EP (2) EP2116541B1 (https=)
JP (1) JP4227660B2 (https=)
KR (1) KR100869616B1 (https=)
AP (1) AP2320A (https=)
AR (1) AR049894A1 (https=)
AT (1) ATE437870T1 (https=)
AU (1) AU2005247684B2 (https=)
BR (1) BRPI0510284A (https=)
CA (1) CA2566108C (https=)
CR (1) CR8744A (https=)
CY (1) CY1109322T1 (https=)
DE (1) DE602005015699D1 (https=)
DK (1) DK1753748T3 (https=)
EA (1) EA011086B9 (https=)
EC (1) ECSP066985A (https=)
ES (1) ES2327857T3 (https=)
GE (1) GEP20084421B (https=)
HR (1) HRP20090471T1 (https=)
IL (1) IL178339A (https=)
MA (1) MA28578B1 (https=)
MX (1) MXPA06013114A (https=)
MY (1) MY139805A (https=)
NL (1) NL1029015C2 (https=)
NO (1) NO20064400L (https=)
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PA (1) PA8632701A1 (https=)
PE (1) PE20060316A1 (https=)
PL (1) PL1753748T3 (https=)
PT (1) PT1753748E (https=)
RS (1) RS51106B (https=)
SI (1) SI1753748T1 (https=)
SV (1) SV2006002110A (https=)
TW (1) TWI347322B (https=)
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KR100926247B1 (ko) * 2001-02-24 2009-11-12 베링거 잉겔하임 파르마 게엠베하 운트 코 카게 크산틴 유도체를 포함하는 약제학적 조성물 및 이의제조방법
US7407955B2 (en) 2002-08-21 2008-08-05 Boehringer Ingelheim Pharma Gmbh & Co., Kg 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions
US7501426B2 (en) 2004-02-18 2009-03-10 Boehringer Ingelheim International Gmbh 8-[3-amino-piperidin-1-yl]-xanthines, their preparation and their use as pharmaceutical compositions
KR100869616B1 (ko) 2004-05-12 2008-11-21 화이자 프로덕츠 인코포레이티드 프롤린 유도체 및 그의 다이펩티딜 펩티다제-iv저해제로서의 용도
DE102004054054A1 (de) 2004-11-05 2006-05-11 Boehringer Ingelheim Pharma Gmbh & Co. Kg Verfahren zur Herstellung chiraler 8-(3-Amino-piperidin-1-yl)-xanthine
US7635698B2 (en) 2004-12-29 2009-12-22 Millennium Pharmaceuticals, Inc. Compounds useful as chemokine receptor antagonists
US7880002B2 (en) 2004-12-29 2011-02-01 Millennium Pharmaceuticals, Inc. Substituted piperazinyl-pyrrolidine compounds useful as chemokine receptor antagonists
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