KR100704717B1 - 사이클릭 뎁시펩타이드 및 피페라진을 함유하는내부기생충 구제용 상승적 배합물 - Google Patents

사이클릭 뎁시펩타이드 및 피페라진을 함유하는내부기생충 구제용 상승적 배합물 Download PDF

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Publication number
KR100704717B1
KR100704717B1 KR1020017013555A KR20017013555A KR100704717B1 KR 100704717 B1 KR100704717 B1 KR 100704717B1 KR 1020017013555 A KR1020017013555 A KR 1020017013555A KR 20017013555 A KR20017013555 A KR 20017013555A KR 100704717 B1 KR100704717 B1 KR 100704717B1
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KR
South Korea
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spp
alkyl
optionally substituted
independently
cyclic depsipeptide
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Expired - Fee Related
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KR1020017013555A
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English (en)
Korean (ko)
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KR20010109527A (ko
Inventor
하더아힘
폰잠존-힘멜스트예르나게오르그
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바이엘 악티엔게젤샤프트
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/15—Depsipeptides; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Immunology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Steroid Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
KR1020017013555A 1999-05-12 2000-05-04 사이클릭 뎁시펩타이드 및 피페라진을 함유하는내부기생충 구제용 상승적 배합물 Expired - Fee Related KR100704717B1 (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19921887.0 1999-05-12
DE19921887A DE19921887A1 (de) 1999-05-12 1999-05-12 Endoparasitizide Mittel

Publications (2)

Publication Number Publication Date
KR20010109527A KR20010109527A (ko) 2001-12-10
KR100704717B1 true KR100704717B1 (ko) 2007-04-09

Family

ID=7907825

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020017013555A Expired - Fee Related KR100704717B1 (ko) 1999-05-12 2000-05-04 사이클릭 뎁시펩타이드 및 피페라진을 함유하는내부기생충 구제용 상승적 배합물

Country Status (26)

Country Link
EP (1) EP1189615B1 (enExample)
JP (1) JP2002544224A (enExample)
KR (1) KR100704717B1 (enExample)
CN (1) CN1224391C (enExample)
AT (1) ATE258795T1 (enExample)
AU (1) AU768910B2 (enExample)
BR (1) BR0010499A (enExample)
CA (1) CA2373827C (enExample)
CZ (1) CZ300782B6 (enExample)
DE (2) DE19921887A1 (enExample)
DK (1) DK1189615T3 (enExample)
ES (1) ES2211558T3 (enExample)
HK (1) HK1047228B (enExample)
HR (1) HRP20010918B1 (enExample)
HU (1) HUP0201201A3 (enExample)
MX (1) MXPA01011455A (enExample)
NO (1) NO328870B1 (enExample)
PL (1) PL200951B1 (enExample)
PT (1) PT1189615E (enExample)
RS (1) RS50169B (enExample)
RU (1) RU2250779C2 (enExample)
SK (1) SK285494B6 (enExample)
TR (2) TR200103240T2 (enExample)
UA (1) UA72520C2 (enExample)
WO (1) WO2000069425A2 (enExample)
ZA (1) ZA200108238B (enExample)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10008128A1 (de) * 2000-02-22 2001-08-23 Bayer Ag Endoparasitizide Mittel
DE10358525A1 (de) * 2003-12-13 2005-07-07 Bayer Healthcare Ag Endoparasitizide Mittel zur topischen Applikation
KR101671325B1 (ko) * 2015-01-09 2016-11-02 한국생명공학연구원 신규한 고리형 뎁시펩타이드계 화합물, 이의 제조방법 및 이를 유효성분으로 함유하는 항균용 약학적 조성물
US10081656B2 (en) 2015-05-20 2018-09-25 Merial, Inc. Anthelmintic depsipeptide compounds
CA3009867C (en) 2015-12-28 2022-05-31 Merial, Inc. Anthelmintic cyclic depsipeptide compounds
WO2018093920A1 (en) 2016-11-16 2018-05-24 Merial, Inc. Anthelmintic depsipeptide compounds
US20230339874A1 (en) * 2020-09-11 2023-10-26 The Governing Council Of The University Of Toronto Piperazinyl compounds and methods for treating nematode infections

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA842571B (en) * 1983-04-07 1985-11-27 Merck & Co Inc Novel synergistic antiparasitic combinations
JPS6471865A (en) * 1987-09-11 1989-03-16 Nichibai Boeki Kk 1-alkylcarbamoyl-4-methylpiperazine derivative
NO176766C (no) * 1989-02-07 1995-05-24 Meiji Seika Kaisha Fremgangsmåte for fremstilling av en forbindelse med anthelmintaktivitet
EP0718293B1 (en) * 1993-09-06 2002-03-13 Fujisawa Pharmaceutical Co., Ltd. Cyclodepsipeptide compound
DE4400464A1 (de) * 1994-01-11 1995-07-13 Bayer Ag Endoparasitizide Mittel
DE19520275A1 (de) * 1995-06-02 1996-12-05 Bayer Ag Endoparasitizide Mittel
WO1997009331A1 (en) * 1995-09-07 1997-03-13 Pharmacia & Upjohn Company Cycloanthelmintic inhibitors
WO1998037088A1 (en) * 1997-02-19 1998-08-27 Meiji Seika Kaisha Ltd. Derivatives of cyclodepsipeptide, pf1022 substance
JP2002502398A (ja) * 1997-06-04 2002-01-22 バイエル・アクチエンゲゼルシヤフト デソキシシクロデプシペプチド及び内部寄生性生物の防除のためのその使用
EP1028126A4 (en) * 1998-08-04 2004-11-10 Nisshin Seifun Group Inc DEPSIPEPTIDE DERIVATIVES WITH PIPERAZINE RINGS

Also Published As

Publication number Publication date
EP1189615A2 (de) 2002-03-27
SK285494B6 (sk) 2007-02-01
KR20010109527A (ko) 2001-12-10
WO2000069425A3 (de) 2001-03-15
NO20015398D0 (no) 2001-11-05
TR200103240T2 (tr) 2002-04-22
TR200401875T2 (tr) 2005-01-24
SK16262001A3 (sk) 2002-03-05
WO2000069425A2 (de) 2000-11-23
AU5523700A (en) 2000-12-05
CA2373827A1 (en) 2000-11-23
HUP0201201A3 (en) 2003-03-28
AU768910B2 (en) 2004-01-08
ES2211558T3 (es) 2004-07-16
CZ20014060A3 (cs) 2002-06-12
CN1224391C (zh) 2005-10-26
JP2002544224A (ja) 2002-12-24
HRP20010918A2 (en) 2003-04-30
NO20015398L (no) 2001-11-05
CN1352559A (zh) 2002-06-05
YU80501A (sh) 2004-09-03
RS50169B (sr) 2009-05-06
PL200951B1 (pl) 2009-02-27
DK1189615T3 (da) 2004-06-07
NO328870B1 (no) 2010-06-07
DE19921887A1 (de) 2000-11-16
ATE258795T1 (de) 2004-02-15
HRP20010918B1 (en) 2011-01-31
HK1047228A1 (en) 2003-02-14
PL351376A1 (en) 2003-04-07
BR0010499A (pt) 2002-02-13
CZ300782B6 (cs) 2009-08-12
HUP0201201A2 (en) 2002-08-28
MXPA01011455A (es) 2002-07-30
CA2373827C (en) 2008-09-16
RU2250779C2 (ru) 2005-04-27
UA72520C2 (uk) 2005-03-15
PT1189615E (pt) 2004-05-31
EP1189615B1 (de) 2004-02-04
DE50005213D1 (de) 2004-03-11
HK1047228B (zh) 2006-07-21
ZA200108238B (en) 2002-12-24

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