JPH1036346A5 - - Google Patents

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Publication number
JPH1036346A5
JPH1036346A5 JP1997101563A JP10156397A JPH1036346A5 JP H1036346 A5 JPH1036346 A5 JP H1036346A5 JP 1997101563 A JP1997101563 A JP 1997101563A JP 10156397 A JP10156397 A JP 10156397A JP H1036346 A5 JPH1036346 A5 JP H1036346A5
Authority
JP
Japan
Prior art keywords
compound
pharmaceutically acceptable
acceptable salt
azepan
indol
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP1997101563A
Other languages
English (en)
Japanese (ja)
Other versions
JP4093611B2 (ja
JPH1036346A (ja
Filing date
Publication date
Priority claimed from US08/833,271 external-priority patent/US5998402A/en
Application filed filed Critical
Publication of JPH1036346A publication Critical patent/JPH1036346A/ja
Publication of JPH1036346A5 publication Critical patent/JPH1036346A5/ja
Application granted granted Critical
Publication of JP4093611B2 publication Critical patent/JP4093611B2/ja
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

JP10156397A 1996-04-19 1997-04-18 エストロゲン剤 Expired - Lifetime JP4093611B2 (ja)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US63397496A 1996-04-19 1996-04-19
US08/633974 1996-04-19
US08/833,271 US5998402A (en) 1996-04-19 1997-04-04 2-phenyl-1-[4-(2-aminoethoxy)-benzyl]-indoles as estrogenic agents
US08/833271 1997-04-04

Publications (3)

Publication Number Publication Date
JPH1036346A JPH1036346A (ja) 1998-02-10
JPH1036346A5 true JPH1036346A5 (https=) 2008-02-14
JP4093611B2 JP4093611B2 (ja) 2008-06-04

Family

ID=27092026

Family Applications (1)

Application Number Title Priority Date Filing Date
JP10156397A Expired - Lifetime JP4093611B2 (ja) 1996-04-19 1997-04-18 エストロゲン剤

Country Status (26)

Country Link
EP (1) EP0802183B1 (https=)
JP (1) JP4093611B2 (https=)
KR (1) KR100480193B1 (https=)
CN (1) CN1106383C (https=)
AR (1) AR011503A1 (https=)
AT (1) ATE206701T1 (https=)
AU (1) AU710149B2 (https=)
BR (1) BRPI9715334B8 (https=)
CO (1) CO4900051A1 (https=)
CY (2) CY2325B1 (https=)
CZ (1) CZ291701B6 (https=)
DE (2) DE69707189T2 (https=)
DK (1) DK0802183T3 (https=)
EA (1) EA001448B1 (https=)
ES (1) ES2162198T3 (https=)
FR (1) FR09C0048I2 (https=)
HU (1) HU227077B1 (https=)
IL (1) IL120701A (https=)
LU (1) LU91608I2 (https=)
MX (1) MX9702865A (https=)
NL (1) NL300416I2 (https=)
NO (2) NO309564B1 (https=)
NZ (1) NZ314601A (https=)
PT (1) PT802183E (https=)
SK (1) SK281737B6 (https=)
UA (1) UA48148C2 (https=)

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WO2002003989A2 (en) * 2000-07-06 2002-01-17 Wyeth Use of substituted indole compounds for treating sphincter incontinence
US6358991B2 (en) * 2000-07-06 2002-03-19 American Home Products Corporation Methods of treating neuropeptide Y-related conditions
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ATE321754T1 (de) 2001-05-22 2006-04-15 Lilly Co Eli 2-substituierte 1,2,3,4-tetrahydrochinoline und derivate davon, zusammensetzungen und verfahren
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ATE433322T1 (de) 2002-07-22 2009-06-15 Lilly Co Eli Selektive östrogenrezeptor modulatoren, die eine phenylsulfonyl-gruppe enthalten
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US7250440B2 (en) * 2003-08-12 2007-07-31 Wyeth (Hydroxyphenyl)-1H-indole-3-carbaldehyde oxime derivatives as estrogenic agents
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CN1946689A (zh) 2004-04-08 2007-04-11 惠氏公司 作为选择性雌激素受体调节剂的巴西多昔芬抗坏血酸盐
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CN101977897A (zh) * 2008-02-11 2011-02-16 惠氏有限责任公司 制备乙酸巴多昔芬的多晶型a的方法
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KR20200144591A (ko) 2010-06-16 2020-12-29 앙도르쉐르슈 인코포레이티드 에스트로겐-관련 질병의 치료 또는 예방 방법
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FI3834824T3 (fi) 2014-03-28 2025-12-05 Univ Duke Estrogeenireseptoripositiivisen rintasyövän hoito selektiivisellä estrogeenireseptorin modulaattorilla
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KR20190110400A (ko) 2018-03-20 2019-09-30 엠에프씨 주식회사 새로운 중간체를 이용한 바제독시펜의 제조방법
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US11246874B1 (en) 2021-04-20 2022-02-15 Oxygen Biotech LLC Treatment of COVID-19

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