MA26523A1 - Modification thermodynamiquement stable de 1-(4-carbazolyloxy)-3-(2-(2-methoxyphenoxy) ethylamino)-2-propanole, procede pour sa preparation et compositions pharmaceutiques le comprenant - Google Patents
Modification thermodynamiquement stable de 1-(4-carbazolyloxy)-3-(2-(2-methoxyphenoxy) ethylamino)-2-propanole, procede pour sa preparation et compositions pharmaceutiques le comprenantInfo
- Publication number
- MA26523A1 MA26523A1 MA25178A MA25178A MA26523A1 MA 26523 A1 MA26523 A1 MA 26523A1 MA 25178 A MA25178 A MA 25178A MA 25178 A MA25178 A MA 25178A MA 26523 A1 MA26523 A1 MA 26523A1
- Authority
- MA
- Morocco
- Prior art keywords
- carbazolyloxy
- propanole
- methoxyphenoxy
- ethylamino
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/56—Ring systems containing three or more rings
- C07D209/80—[b, c]- or [b, d]-condensed
- C07D209/82—Carbazoles; Hydrogenated carbazoles
- C07D209/88—Carbazoles; Hydrogenated carbazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the ring system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP97112491A EP0893440A1 (fr) | 1997-07-22 | 1997-07-22 | Une modification thermodynamique stabilisée de 1-(4-carbazolyloxy)-3[2-(2-methoxyphenoxy)ethylamino]- 2-propanole, un procédé pour sa préparation et une composition pharmaceutique qui la contient |
Publications (1)
Publication Number | Publication Date |
---|---|
MA26523A1 true MA26523A1 (fr) | 2004-12-20 |
Family
ID=8227094
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MA25178A MA26523A1 (fr) | 1997-07-22 | 1998-07-20 | Modification thermodynamiquement stable de 1-(4-carbazolyloxy)-3-(2-(2-methoxyphenoxy) ethylamino)-2-propanole, procede pour sa preparation et compositions pharmaceutiques le comprenant |
Country Status (32)
Country | Link |
---|---|
EP (2) | EP0893440A1 (fr) |
JP (1) | JP2001510824A (fr) |
KR (1) | KR100336229B1 (fr) |
CN (1) | CN1125047C (fr) |
AR (1) | AR015133A1 (fr) |
AT (1) | ATE236123T1 (fr) |
AU (1) | AU740453B2 (fr) |
BR (1) | BR9810776A (fr) |
CA (1) | CA2296637C (fr) |
CZ (1) | CZ296947B6 (fr) |
DE (1) | DE69812964T2 (fr) |
DK (1) | DK1000027T3 (fr) |
ES (1) | ES2195366T3 (fr) |
HK (1) | HK1029339A1 (fr) |
HR (1) | HRP980406A2 (fr) |
HU (1) | HUP0003198A3 (fr) |
IL (1) | IL133677A (fr) |
MA (1) | MA26523A1 (fr) |
MY (1) | MY117734A (fr) |
NO (1) | NO313588B1 (fr) |
NZ (1) | NZ502136A (fr) |
PE (1) | PE96999A1 (fr) |
PL (1) | PL191602B1 (fr) |
PT (1) | PT1000027E (fr) |
RU (1) | RU2202542C2 (fr) |
SI (1) | SI1000027T1 (fr) |
TR (1) | TR200000148T2 (fr) |
TW (1) | TW505631B (fr) |
UY (1) | UY25108A1 (fr) |
WO (1) | WO1999005105A1 (fr) |
YU (1) | YU2200A (fr) |
ZA (1) | ZA986475B (fr) |
Families Citing this family (22)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2003528914A (ja) * | 2000-04-03 | 2003-09-30 | エフ.ホフマン−ラ ロシュ アーゲー | カルベジロールの濃縮溶液 |
EP1655285A1 (fr) * | 2000-06-28 | 2006-05-10 | Teva Pharmaceutical Industries Ltd. | Procédé de préparation d'une forme crystalline de carvedilol (forme II) |
KR20030017569A (ko) * | 2000-06-28 | 2003-03-03 | 테바 파마슈티컬 인더스트리즈 리미티드 | 카르베딜올 |
EP1406614B1 (fr) * | 2001-07-13 | 2006-06-07 | Smithkline Beecham Corporation | Polymorphe de carvedilol |
EP1929998A3 (fr) | 2001-09-21 | 2008-11-26 | Egalet A/S | Dispersions solides à libération contrôlée de carvedilol |
BR0212927A (pt) * | 2001-09-28 | 2004-10-13 | Hoffmann La Roche | Formas pseudopolimórficas de carvedilol |
KR20040077872A (ko) | 2002-01-15 | 2004-09-07 | 테바 파마슈티컬 인더스트리즈 리미티드 | 카베디롤의 결정질 고체 및 그 제조 방법 |
WO2003092622A2 (fr) * | 2002-04-30 | 2003-11-13 | Sb Pharmco Puerto Rico Inc. | Monocitrate monohydrate de carvedilol |
EP1534270A4 (fr) | 2002-06-27 | 2006-05-17 | Sb Pharmco Inc | Sels de phospate de carvedilol et/ou solvates de celui-ci, compositions et/ou methodes de traitement associees |
EP1539140A4 (fr) * | 2002-06-27 | 2005-12-07 | Sb Pharmco Inc | Hydobromure de carvedilol |
WO2004041252A1 (fr) * | 2002-11-08 | 2004-05-21 | Egalet A/S | Compositions de carvedilol a liberation commandee |
ES2570454T3 (es) | 2003-03-26 | 2016-05-18 | Egalet Ltd | Sistema de liberación controlada de morfina |
WO2004094378A1 (fr) * | 2003-04-21 | 2004-11-04 | Matrix Laboratories Ltd | Procede de fabrication de carvedilol, forme-ii |
SI21616A (sl) * | 2003-09-02 | 2005-04-30 | Krka, Tovarna Zdravil, D.D., Novo Mesto | Nove kristalne oblike karvedilola |
US7750036B2 (en) | 2003-11-25 | 2010-07-06 | Sb Pharmco Puerto Rico Inc. | Carvedilol salts, corresponding compositions, methods of delivery and/or treatment |
CA2589699A1 (fr) * | 2004-12-09 | 2006-06-15 | Zach System S.P.A. | Procede de preparation de carvedilol et de ses enantiomeres |
KR20070088507A (ko) * | 2005-06-09 | 2007-08-29 | 테바 파마슈티컬 인더스트리즈 리미티드 | 카베딜올의 결정질 형태 및 이것의 제조 방법 |
EP1991527A2 (fr) | 2006-06-28 | 2008-11-19 | Teva Pharmaceutical Industries Ltd | Formes polymorphes de carvédilol phosphate |
US20080249317A1 (en) * | 2007-04-04 | 2008-10-09 | Apotex Inc. | Novel amorphous form of carvedilol phosphate and processes for the preparation thereof |
WO2008148798A2 (fr) | 2007-06-04 | 2008-12-11 | Egalet A/S | Compositions pharmaceutiques à libération contrôlée pour un effet prolongé |
EP2393484A1 (fr) | 2009-02-06 | 2011-12-14 | Egalet Ltd. | Composition à libération immédiate résistant à une maltraitance par prise d'alcool |
AU2010265213B2 (en) | 2009-06-24 | 2012-08-23 | Egalet Ltd. | Controlled release formulations |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2815926A1 (de) * | 1978-04-13 | 1979-10-18 | Boehringer Mannheim Gmbh | Neue carbazolyl-(4)-oxy-propanolamin-derivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel |
DE3319027A1 (de) * | 1983-05-26 | 1984-11-29 | Boehringer Mannheim Gmbh, 6800 Mannheim | Verfahren zur herstellung von optisch aktiven carbazol-derivaten, neue r- und s-carbazol-derivate, sowie arzneimittel, die diese verbindungen enthalten |
-
1997
- 1997-07-22 EP EP97112491A patent/EP0893440A1/fr not_active Withdrawn
-
1998
- 1998-07-15 PE PE1998000626A patent/PE96999A1/es not_active Application Discontinuation
- 1998-07-15 MY MYPI98003245A patent/MY117734A/en unknown
- 1998-07-18 BR BR9810776-3A patent/BR9810776A/pt not_active Application Discontinuation
- 1998-07-18 IL IL13367798A patent/IL133677A/en not_active IP Right Cessation
- 1998-07-18 CN CN98807436A patent/CN1125047C/zh not_active Expired - Fee Related
- 1998-07-18 HU HU0003198A patent/HUP0003198A3/hu unknown
- 1998-07-18 KR KR1020007000667A patent/KR100336229B1/ko not_active IP Right Cessation
- 1998-07-18 TR TR2000/00148T patent/TR200000148T2/xx unknown
- 1998-07-18 AU AU86319/98A patent/AU740453B2/en not_active Ceased
- 1998-07-18 SI SI9830442T patent/SI1000027T1/xx unknown
- 1998-07-18 PT PT98937576T patent/PT1000027E/pt unknown
- 1998-07-18 ES ES98937576T patent/ES2195366T3/es not_active Expired - Lifetime
- 1998-07-18 CZ CZ20000221A patent/CZ296947B6/cs not_active IP Right Cessation
- 1998-07-18 WO PCT/EP1998/004475 patent/WO1999005105A1/fr active IP Right Grant
- 1998-07-18 YU YU2200A patent/YU2200A/sh unknown
- 1998-07-18 RU RU2000103033/04A patent/RU2202542C2/ru not_active IP Right Cessation
- 1998-07-18 AT AT98937576T patent/ATE236123T1/de not_active IP Right Cessation
- 1998-07-18 PL PL338432A patent/PL191602B1/pl unknown
- 1998-07-18 DK DK98937576T patent/DK1000027T3/da active
- 1998-07-18 NZ NZ502136A patent/NZ502136A/en unknown
- 1998-07-18 DE DE69812964T patent/DE69812964T2/de not_active Expired - Fee Related
- 1998-07-18 JP JP2000504104A patent/JP2001510824A/ja active Pending
- 1998-07-18 CA CA002296637A patent/CA2296637C/fr not_active Expired - Fee Related
- 1998-07-18 TW TW087111738A patent/TW505631B/zh not_active IP Right Cessation
- 1998-07-18 EP EP98937576A patent/EP1000027B1/fr not_active Expired - Lifetime
- 1998-07-20 MA MA25178A patent/MA26523A1/fr unknown
- 1998-07-21 ZA ZA9806475A patent/ZA986475B/xx unknown
- 1998-07-21 AR ARP980103547A patent/AR015133A1/es unknown
- 1998-07-22 HR HR97112491.2A patent/HRP980406A2/hr not_active Application Discontinuation
- 1998-07-22 UY UY25108A patent/UY25108A1/es not_active IP Right Cessation
-
2000
- 2000-01-21 NO NO20000301A patent/NO313588B1/no unknown
-
2001
- 2001-01-02 HK HK01100012A patent/HK1029339A1/xx not_active IP Right Cessation
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