NO20000301L - Termodynamisk stabil modifikasjon av 1-(4-karbazolyloksy)-3- [2-(2-metoksyfenoksy)etylamino]-2-propanol, fremgangsmåte for fremstilling derav og farmasøytiske blandinger som inneholder den - Google Patents

Termodynamisk stabil modifikasjon av 1-(4-karbazolyloksy)-3- [2-(2-metoksyfenoksy)etylamino]-2-propanol, fremgangsmåte for fremstilling derav og farmasøytiske blandinger som inneholder den

Info

Publication number
NO20000301L
NO20000301L NO20000301A NO20000301A NO20000301L NO 20000301 L NO20000301 L NO 20000301L NO 20000301 A NO20000301 A NO 20000301A NO 20000301 A NO20000301 A NO 20000301A NO 20000301 L NO20000301 L NO 20000301L
Authority
NO
Norway
Prior art keywords
carbazolyloxy
methoxyphenoxy
ethylamino
propanol
preparation
Prior art date
Application number
NO20000301A
Other languages
English (en)
Other versions
NO20000301D0 (no
NO313588B1 (no
Inventor
Erhard Reinholz
Peter Beyer
Original Assignee
Roche Diagnostics Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roche Diagnostics Gmbh filed Critical Roche Diagnostics Gmbh
Publication of NO20000301D0 publication Critical patent/NO20000301D0/no
Publication of NO20000301L publication Critical patent/NO20000301L/no
Publication of NO313588B1 publication Critical patent/NO313588B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/56—Ring systems containing three or more rings
    • C07D209/80—[b, c]- or [b, d]-condensed
    • C07D209/82—Carbazoles; Hydrogenated carbazoles
    • C07D209/88—Carbazoles; Hydrogenated carbazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
NO20000301A 1997-07-22 2000-01-21 Termodynamisk stabil modifikasjon av 1-(4-karbazolyloksy)-3- [2-(2-metoksyfenoksy)etylamino]-2-propanol, fremgangsmåte forfremstilling derav og farmasöytiske blandinger som inneholder den NO313588B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP97112491A EP0893440A1 (en) 1997-07-22 1997-07-22 Thermodynamically stable modification of 1-(4-carbazolyloxy)-3-[2-(2-methoxyphenoxy)ethylamino]-2-propanole, process for its preparation and pharmaceutical compositions containing it
PCT/EP1998/004475 WO1999005105A1 (en) 1997-07-22 1998-07-18 Thermodynamically stable modification of 1-(4-carbazolyloxy)-3-[2-(2-methoxyphenoxy)ethylamino]-2-propanole, process for its preparation and pharmaceutical compositions containing it

Publications (3)

Publication Number Publication Date
NO20000301D0 NO20000301D0 (no) 2000-01-21
NO20000301L true NO20000301L (no) 2000-01-21
NO313588B1 NO313588B1 (no) 2002-10-28

Family

ID=8227094

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20000301A NO313588B1 (no) 1997-07-22 2000-01-21 Termodynamisk stabil modifikasjon av 1-(4-karbazolyloksy)-3- [2-(2-metoksyfenoksy)etylamino]-2-propanol, fremgangsmåte forfremstilling derav og farmasöytiske blandinger som inneholder den

Country Status (32)

Country Link
EP (2) EP0893440A1 (no)
JP (1) JP2001510824A (no)
KR (1) KR100336229B1 (no)
CN (1) CN1125047C (no)
AR (1) AR015133A1 (no)
AT (1) ATE236123T1 (no)
AU (1) AU740453B2 (no)
BR (1) BR9810776A (no)
CA (1) CA2296637C (no)
CZ (1) CZ296947B6 (no)
DE (1) DE69812964T2 (no)
DK (1) DK1000027T3 (no)
ES (1) ES2195366T3 (no)
HK (1) HK1029339A1 (no)
HR (1) HRP980406A2 (no)
HU (1) HUP0003198A3 (no)
IL (1) IL133677A (no)
MA (1) MA26523A1 (no)
MY (1) MY117734A (no)
NO (1) NO313588B1 (no)
NZ (1) NZ502136A (no)
PE (1) PE96999A1 (no)
PL (1) PL191602B1 (no)
PT (1) PT1000027E (no)
RU (1) RU2202542C2 (no)
SI (1) SI1000027T1 (no)
TR (1) TR200000148T2 (no)
TW (1) TW505631B (no)
UY (1) UY25108A1 (no)
WO (1) WO1999005105A1 (no)
YU (1) YU2200A (no)
ZA (1) ZA986475B (no)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2402336C (en) * 2000-04-03 2008-03-11 F. Hoffmann-La Roche Ag Concentrated solutions of carvedilol
EP1655285A1 (en) * 2000-06-28 2006-05-10 Teva Pharmaceutical Industries Ltd. Method for preparation of a crystalline form of carvedilol (form II)
CN1245974C (zh) * 2000-06-28 2006-03-22 特瓦制药工业有限公司 卡维地洛
AU2002326391A1 (en) * 2001-07-13 2003-01-29 Smithkline Beecham Corporation Carvedilol polymorph
WO2003024426A1 (en) 2001-09-21 2003-03-27 Egalet A/S Controlled release solid dispersions
CN1308307C (zh) * 2001-09-28 2007-04-04 弗·哈夫曼-拉罗切有限公司 假多晶型的卡维地洛
MXPA04006909A (es) 2002-01-15 2005-04-19 Teva Pharma Solidos cristalinos de carvedilol y procesos para su preparacion.
US20050148779A1 (en) * 2002-04-30 2005-07-07 Wei Chen Carvedilol monocitrate monohydrate
CA2492084A1 (en) 2002-06-27 2004-01-08 Sb Pharmco Puerto Rico Inc. Carvedilol hydobromide
CN1678305A (zh) 2002-06-27 2005-10-05 Sb药物波多黎各公司 卡维地洛磷酸盐和/或其溶剂合物和/或相应组合物和/或治疗方法
WO2004041252A1 (en) * 2002-11-08 2004-05-21 Egalet A/S Controlled release carvedilol compositions
WO2004084868A1 (en) 2003-03-26 2004-10-07 Egalet A/S Morphine controlled release system
EP1615888A1 (en) * 2003-04-21 2006-01-18 Matrix Laboratories Ltd Process for the preparation of carvedilol form-ii
SI21616A (sl) * 2003-09-02 2005-04-30 Krka, Tovarna Zdravil, D.D., Novo Mesto Nove kristalne oblike karvedilola
WO2005051383A1 (en) * 2003-11-25 2005-06-09 Sb Pharmco Puerto Rico Inc. Carvedilol salts, corresponding compositions, methods of delivery and/or treatment
DK1838670T3 (da) * 2004-12-09 2010-03-01 Zach System Spa Fremgangsmåde til fremstilling af carvedilol og dets enantiomere
US20070043099A1 (en) * 2005-06-09 2007-02-22 Igor Lifshitz Crystalline forms of carvedilol and processes for their preparation
WO2008002683A2 (en) 2006-06-28 2008-01-03 Teva Pharmaceutical Industries Ltd. Polymorphous forms of carvedilol phosphate
US20080249317A1 (en) * 2007-04-04 2008-10-09 Apotex Inc. Novel amorphous form of carvedilol phosphate and processes for the preparation thereof
CA2687192C (en) 2007-06-04 2015-11-24 Egalet A/S Controlled release pharmaceutical compositions for prolonged effect
CA2751667C (en) 2009-02-06 2016-12-13 Egalet Ltd. Immediate release composition resistant to abuse by intake of alcohol
NZ597283A (en) 2009-06-24 2013-07-26 Egalet Ltd Controlled release formulations

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2815926A1 (de) * 1978-04-13 1979-10-18 Boehringer Mannheim Gmbh Neue carbazolyl-(4)-oxy-propanolamin-derivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
DE3319027A1 (de) * 1983-05-26 1984-11-29 Boehringer Mannheim Gmbh, 6800 Mannheim Verfahren zur herstellung von optisch aktiven carbazol-derivaten, neue r- und s-carbazol-derivate, sowie arzneimittel, die diese verbindungen enthalten

Also Published As

Publication number Publication date
IL133677A0 (en) 2001-04-30
WO1999005105A1 (en) 1999-02-04
EP1000027B1 (en) 2003-04-02
UY25108A1 (es) 2000-12-29
DE69812964T2 (de) 2004-03-04
CZ296947B6 (cs) 2006-08-16
ZA986475B (en) 2000-01-21
PL338432A1 (en) 2000-11-06
CZ2000221A3 (cs) 2000-05-17
JP2001510824A (ja) 2001-08-07
DK1000027T3 (da) 2003-07-21
EP0893440A1 (en) 1999-01-27
SI1000027T1 (en) 2003-10-31
NO20000301D0 (no) 2000-01-21
CN1264366A (zh) 2000-08-23
CN1125047C (zh) 2003-10-22
MY117734A (en) 2004-07-31
IL133677A (en) 2004-06-01
HUP0003198A3 (en) 2002-10-28
ES2195366T3 (es) 2003-12-01
PL191602B1 (pl) 2006-06-30
PE96999A1 (es) 1999-10-12
PT1000027E (pt) 2003-07-31
NO313588B1 (no) 2002-10-28
NZ502136A (en) 2002-05-31
ATE236123T1 (de) 2003-04-15
DE69812964D1 (de) 2003-05-08
AU740453B2 (en) 2001-11-01
CA2296637C (en) 2005-11-15
MA26523A1 (fr) 2004-12-20
CA2296637A1 (en) 1999-02-04
AU8631998A (en) 1999-02-16
YU2200A (sh) 2002-03-18
KR20010022097A (ko) 2001-03-15
KR100336229B1 (ko) 2002-05-09
TW505631B (en) 2002-10-11
BR9810776A (pt) 2000-09-19
EP1000027A1 (en) 2000-05-17
HUP0003198A2 (en) 2001-03-28
TR200000148T2 (tr) 2000-07-21
AR015133A1 (es) 2001-04-18
HK1029339A1 (en) 2001-03-30
RU2202542C2 (ru) 2003-04-20
HRP980406A2 (en) 1999-04-30

Similar Documents

Publication Publication Date Title
NO20000301D0 (no) Termodynamisk stabil modifikasjon av 1-(4-karbazolyloksy)-3- [2-(2-metoksyfenoksy)etylamino]-2-propanol, fremgangsmåte for fremstilling derav og farmasoeytiske blandinger som inneholder den
DK1202965T3 (da) Indolderivater, fremgangsmåde til fremstilling deraf, farmaceutiske præparater indeholdende disse og deres medicinske anvendelse
HUP0203257A3 (en) Polymorphic forms of atorvastatin calcium, process for their preparations and pharmaceutical compositions containing them
EE200000707A (et) Oksasolidinooni derivaadid, nende valmistamismeetod ja neid sisaldavad farmatseutilised kompositsioonid
HUP9701694A3 (en) Indolinone derivatives for the treatment of disease, use thereof, pharmaceutical compositions containing these compounds
EE04779B1 (et) 1,3-dihüdro-2H-indool-2-ooni derivaadid, nende valmistamismeetod ja neid sisaldavad farmatseutilised kompositsioonid
CO5160257A1 (es) La n-piperidino-5-(4-bromofenil)-1-(2,4-diclorofenil)-4-etilpirazol-3-carboxamida, sus sales, su preparacion y las composiciones farmaceuticas que la contienen
IS1850B (is) Kristölluð a-fjölgervingsmynd af indól afleiðu, notkun hennar, aðferð til framleiðslu og lyfjaefnablanda
NO20015309L (no) 1- (P-tienylbenzyl)-imidazoler som anginotensin-(1-7) reseptoragonister, fremgangsmåte for fremstilling og anvendelse avde samme og farmasöytiske preparater som inneholder nevnteforbindelser
NO20005430L (no) 1-[(1-substituerte-4-piperidinyl)metyl]-4-piperidinderivater, fremgangsmåter for fremstilling av disse, medisinske preparater inneholdende disse, og mellomprodukter for disse forbindelser
NO20024891L (no) Farmasöytiske sammensetninger
HUP0203873A3 (en) Substituted indole mannich bases, process for their preparation and pharmaceutical compositions containing them
NO984290L (no) Farmas°ytisk nyttige forbindelser
HK1027563A1 (en) Novel 2-(iminomethyl) amino-phenyl derivatives, preparation, application as medicines and pharmaceutical compositions containing same.
HUP0401499A3 (en) Indole derivatives as cox ii inhibitors, process for their preparation and pharmaceutical compositions containing them
PL370412A1 (en) Pseudopolymorphic forms of carvedilol
HUP0201338A2 (en) Novel indole derivatives, pharmaceutical compositions containing them and their use
ZA200303113B (en) Derivatives of tryptamine and analogous compounds, and pharmaceutical formulations containing them.
AU2002346457A1 (en) Pharmaceutical formulations comprising indolinone derivatives
EE04778B1 (et) Hargnenud ahelaga asendatud 3-amino-1-fenüül-1H-[1,2,4]triasooli aminoderivaadid, nende valmistamismeetod ja neid sisaldavad farmatseutilised kompositsioonid
DK1037613T3 (da) Fremgangsmåde til fremstilling af farmaceutiske formuleringer, der indeholder en ekstrakt
EE04437B1 (et) (1-fenatsüül-3-fenüül-3-piperidinüületüül)piperidiini derivaadid, nende valmistamismeetod ja neid sisaldavad farmatseutilised kompositsioonid
EE200100499A (et) Uued morfoliini derivaadid, nende valmistamismeetod ja neid sisaldavad farmatseutilised kompositsioonid
HUP0004432A3 (en) Thermodynamically stable form of (r)-3-[[(4-fluorophenyl)sulphonyl]amino]-1,2,3,4-tetrahydro-9h-carbazole-9-propanoic acid (ramatroban) and pharmaceutical composition containing it
NO20005158L (no) FremgangsmÕte for fremstilling av R-(+)-6-karboksamido-3-N- metylamino-1,2,3,4-tetrahydrokarbazol