DZ3041A1 - Composition pharmaceutique nouvelle comprenant un inhibiteur de nos, et procédé pour sa préparation. - Google Patents

Composition pharmaceutique nouvelle comprenant un inhibiteur de nos, et procédé pour sa préparation.

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Publication number
DZ3041A1
DZ3041A1 DZ000084A DZ000084A DZ3041A1 DZ 3041 A1 DZ3041 A1 DZ 3041A1 DZ 000084 A DZ000084 A DZ 000084A DZ 000084 A DZ000084 A DZ 000084A DZ 3041 A1 DZ3041 A1 DZ 3041A1
Authority
DZ
Algeria
Prior art keywords
preparation
pharmaceutical composition
novel pharmaceutical
nos inhibitor
inhibitor
Prior art date
Application number
DZ000084A
Other languages
English (en)
Inventor
Marlo David Saltarelli
John Adams Lowe Iii
Original Assignee
Pfizer Prod Inc
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Publication date
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Publication of DZ3041A1 publication Critical patent/DZ3041A1/fr

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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/138Aryloxyalkylamines, e.g. propranolol, tamoxifen, phenoxybenzamine
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    • A61K31/13Amines
    • A61K31/15Oximes (>C=N—O—); Hydrazines (>N—N<); Hydrazones (>N—N=) ; Imines (C—N=C)
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    • A61K31/34Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
    • A61K31/343Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
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    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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    • A61K31/439Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
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  • Pyridine Compounds (AREA)
DZ000084A 1999-05-21 2000-05-17 Composition pharmaceutique nouvelle comprenant un inhibiteur de nos, et procédé pour sa préparation. DZ3041A1 (fr)

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JP (1) JP2003523941A (fr)
KR (1) KR20020010916A (fr)
CN (1) CN1617743A (fr)
AP (1) AP2001002326A0 (fr)
AR (1) AR022640A1 (fr)
AU (1) AU2935300A (fr)
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EE (1) EE200100611A (fr)
GT (1) GT200000071A (fr)
HN (1) HN2000000045A (fr)
HR (1) HRP20010862A2 (fr)
HU (1) HUP0301287A3 (fr)
IL (1) IL145955A0 (fr)
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MA (1) MA26732A1 (fr)
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PA (1) PA8494601A1 (fr)
PE (1) PE20010157A1 (fr)
PL (1) PL358538A1 (fr)
SK (1) SK16602001A3 (fr)
TN (1) TNSN00106A1 (fr)
TR (1) TR200103351T2 (fr)
UY (1) UY26148A1 (fr)
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DE10001785A1 (de) * 2000-01-18 2001-07-19 Boehringer Ingelheim Pharma NK¶1¶-Rezeptor-Antagonisten zur Behandlung des Restless Legs Syndroms
GB0019006D0 (en) * 2000-08-04 2000-09-20 Astrazeneca Ab Novel compounds
US20030045449A1 (en) * 2001-08-15 2003-03-06 Pfizer, Inc. Pharmaceutical combinations for the treatment of neurodegenerative diseases
DOP2002000467A (es) * 2001-10-10 2003-04-15 Pfizer Prod Inc 2-amino-6 (fenilo sustituido en las posiciones 2,4,5)-piridinas
US6803470B2 (en) * 2001-10-10 2004-10-12 Pfizer Inc 2-amino-6-(2,4,5-substituted-phenyl)-pyridines
UA82517C2 (uk) * 2003-06-24 2008-04-25 Ньюросерч А/С Нові похідні 8-аза-біцикло[3.2.1]октану та їх застосування як інгібіторів ресорбції моноамінових медіаторів
EP1634598A1 (fr) * 2004-09-07 2006-03-15 Laboratorios Del Dr. Esteve, S.A. Utilisation de dérivés de piperazine et ses analogues pour prevenir et traiter des désordres liés à l'ingestion de nourriture
JO2972B1 (en) 2007-06-08 2016-03-15 جانسين فارماسوتيكا ان. في Piperidine / piperazine derivatives
CA2687912C (fr) 2007-06-08 2015-11-03 Janssen Pharmaceutica N.V. Derives de piperidine/piperazine
JP5464709B2 (ja) 2007-06-08 2014-04-09 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ ピペリジン/ピペラジン誘導体
AU2008258487B2 (en) 2007-06-08 2012-11-15 Janssen Pharmaceutica N.V. Piperidine/piperazine derivatives
AU2009253892B2 (en) 2008-06-05 2015-07-30 Janssen Pharmaceutica Nv Drug combinations comprising a DGAT inhibitor and a PPAR-agonist
WO2010101246A1 (fr) * 2009-03-05 2010-09-10 塩野義製薬株式会社 Dérivés de la pipéridine et de la pyrrolidine dotés d'un antagonisme pour les récepteurs npy y5
EP2919788A4 (fr) 2012-11-14 2016-05-25 Univ Johns Hopkins Méthodes et compositions pour le traitement de la schizophrénie
AU2020291468A1 (en) * 2019-06-14 2022-01-06 Srx Cardio, Llc Compounds for the modulation of proprotein convertase subtilisin/kexin type 9 (PCSK9)

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JP2003523941A (ja) 2003-08-12
CO5160295A1 (es) 2002-05-30
WO2000071107A2 (fr) 2000-11-30
NO20015651D0 (no) 2001-11-20
EA200101110A1 (ru) 2002-08-29
GT200000071A (es) 2001-11-08
ZA200109555B (en) 2004-04-07
HUP0301287A3 (en) 2005-03-29
TNSN00106A1 (fr) 2005-11-10
PE20010157A1 (es) 2001-02-16
TR200103351T2 (tr) 2002-06-21
MA26732A1 (fr) 2004-12-20
IS6126A (is) 2001-10-26
PL358538A1 (en) 2004-08-09
AU2935300A (en) 2000-12-12
SK16602001A3 (sk) 2003-03-04
HUP0301287A2 (hu) 2003-08-28
PA8494601A1 (es) 2002-08-29
EP1178784A1 (fr) 2002-02-13
CN1617743A (zh) 2005-05-18
UY26148A1 (es) 2000-12-29
OA11943A (en) 2006-04-12
KR20020010916A (ko) 2002-02-06
IL145955A0 (en) 2002-07-25
HRP20010862A2 (en) 2003-06-30
BR0010820A (pt) 2002-03-05
AR022640A1 (es) 2002-09-04
NO20015651L (no) 2002-01-18
WO2000071107A8 (fr) 2002-01-24
CA2374668A1 (fr) 2000-11-30
MXPA01011978A (es) 2002-05-06
EE200100611A (et) 2003-02-17
BG106208A (en) 2002-09-30
AP2001002326A0 (en) 2001-12-31
HN2000000045A (es) 2001-03-02

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