TNSN00106A1 - Composition pharmaceutique nouvelle comprenant un inhibiteur de nos, et procede pour sa preparation - Google Patents

Composition pharmaceutique nouvelle comprenant un inhibiteur de nos, et procede pour sa preparation

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Publication number
TNSN00106A1
TNSN00106A1 TNTNSN00106A TNSN00106A TNSN00106A1 TN SN00106 A1 TNSN00106 A1 TN SN00106A1 TN TNSN00106 A TNTNSN00106 A TN TNSN00106A TN SN00106 A TNSN00106 A TN SN00106A TN SN00106 A1 TNSN00106 A1 TN SN00106A1
Authority
TN
Tunisia
Prior art keywords
preparation
inhibitor
pharmaceutical composition
novel pharmaceutical
treatment
Prior art date
Application number
TNTNSN00106A
Other languages
English (en)
Inventor
Adams Lowe John Iii
David Saltarelli Mario
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of TNSN00106A1 publication Critical patent/TNSN00106A1/fr

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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
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    • A61K31/138—Aryloxyalkylamines, e.g. propranolol, tamoxifen, phenoxybenzamine
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    • A61K31/15—Oximes (>C=N—O—); Hydrazines (>N—N<); Hydrazones (>N—N=) ; Imines (C—N=C)
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    • A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
    • A61K31/343—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Psychiatry (AREA)
  • Hematology (AREA)
  • Emergency Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Hospice & Palliative Care (AREA)
  • Anesthesiology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Diabetes (AREA)
  • Pulmonology (AREA)
  • Obesity (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pyridine Compounds (AREA)

Abstract

L'INVENTION CONCERNE DES COMPOSITIONS PHAMACEUTIQUES COMPRENANT UN COMPOSE INHIBITEUR DE NOS, SEUL OU EN ASSOCIATION AVEC UN ANTAGONISTE DES RECEPTEURS DE NK -1 OU UN SSRI. ELLE CONCERNE EGALEMENT UN PROCEDE POUR LEUR PREPARATION. APPLICATION : UTILISATION DE CES COMPOSITIONS POUR LE TRAITEMENT DE DIVERS TROUBLES DONT LE TRAITEMENT PEUT ETRE EFFECTUE OU FACILITE PAR LA MODIFICATION DES RYTHMES CIRCADIENS.
TNTNSN00106A 1999-05-21 2000-05-17 Composition pharmaceutique nouvelle comprenant un inhibiteur de nos, et procede pour sa preparation TNSN00106A1 (fr)

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EP (1) EP1178784A1 (fr)
JP (1) JP2003523941A (fr)
KR (1) KR20020010916A (fr)
CN (1) CN1617743A (fr)
AP (1) AP2001002326A0 (fr)
AR (1) AR022640A1 (fr)
AU (1) AU2935300A (fr)
BG (1) BG106208A (fr)
BR (1) BR0010820A (fr)
CA (1) CA2374668A1 (fr)
CO (1) CO5160295A1 (fr)
DZ (1) DZ3041A1 (fr)
EA (1) EA200101110A1 (fr)
EE (1) EE200100611A (fr)
GT (1) GT200000071A (fr)
HN (1) HN2000000045A (fr)
HR (1) HRP20010862A2 (fr)
HU (1) HUP0301287A3 (fr)
IL (1) IL145955A0 (fr)
IS (1) IS6126A (fr)
MA (1) MA26732A1 (fr)
MX (1) MXPA01011978A (fr)
NO (1) NO20015651L (fr)
OA (1) OA11943A (fr)
PA (1) PA8494601A1 (fr)
PE (1) PE20010157A1 (fr)
PL (1) PL358538A1 (fr)
SK (1) SK16602001A3 (fr)
TN (1) TNSN00106A1 (fr)
TR (1) TR200103351T2 (fr)
UY (1) UY26148A1 (fr)
WO (1) WO2000071107A2 (fr)
ZA (1) ZA200109555B (fr)

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Publication number Priority date Publication date Assignee Title
DE10001785A1 (de) * 2000-01-18 2001-07-19 Boehringer Ingelheim Pharma NK¶1¶-Rezeptor-Antagonisten zur Behandlung des Restless Legs Syndroms
GB0019006D0 (en) * 2000-08-04 2000-09-20 Astrazeneca Ab Novel compounds
US20030045449A1 (en) * 2001-08-15 2003-03-06 Pfizer, Inc. Pharmaceutical combinations for the treatment of neurodegenerative diseases
DOP2002000467A (es) * 2001-10-10 2003-04-15 Pfizer Prod Inc 2-amino-6 (fenilo sustituido en las posiciones 2,4,5)-piridinas
US6803470B2 (en) * 2001-10-10 2004-10-12 Pfizer Inc 2-amino-6-(2,4,5-substituted-phenyl)-pyridines
UA82517C2 (uk) * 2003-06-24 2008-04-25 Ньюросерч А/С Нові похідні 8-аза-біцикло[3.2.1]октану та їх застосування як інгібіторів ресорбції моноамінових медіаторів
EP1634598A1 (fr) * 2004-09-07 2006-03-15 Laboratorios Del Dr. Esteve, S.A. Utilisation de dérivés de piperazine et ses analogues pour prevenir et traiter des désordres liés à l'ingestion de nourriture
JO2972B1 (en) 2007-06-08 2016-03-15 جانسين فارماسوتيكا ان. في Piperidine / piperazine derivatives
CA2687912C (fr) 2007-06-08 2015-11-03 Janssen Pharmaceutica N.V. Derives de piperidine/piperazine
JP5464709B2 (ja) 2007-06-08 2014-04-09 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ ピペリジン／ピペラジン誘導体
AU2008258487B2 (en) 2007-06-08 2012-11-15 Janssen Pharmaceutica N.V. Piperidine/piperazine derivatives
AU2009253892B2 (en) 2008-06-05 2015-07-30 Janssen Pharmaceutica Nv Drug combinations comprising a DGAT inhibitor and a PPAR-agonist
WO2010101246A1 (fr) * 2009-03-05 2010-09-10 塩野義製薬株式会社 Dérivés de la pipéridine et de la pyrrolidine dotés d'un antagonisme pour les récepteurs npy y5
EP2919788A4 (fr) 2012-11-14 2016-05-25 Univ Johns Hopkins Méthodes et compositions pour le traitement de la schizophrénie
AU2020291468A1 (en) * 2019-06-14 2022-01-06 Srx Cardio, Llc Compounds for the modulation of proprotein convertase subtilisin/kexin type 9 (PCSK9)

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JP2003523941A (ja) 2003-08-12
CO5160295A1 (es) 2002-05-30
WO2000071107A2 (fr) 2000-11-30
NO20015651D0 (no) 2001-11-20
EA200101110A1 (ru) 2002-08-29
DZ3041A1 (fr) 2004-03-27
GT200000071A (es) 2001-11-08
ZA200109555B (en) 2004-04-07
HUP0301287A3 (en) 2005-03-29
PE20010157A1 (es) 2001-02-16
TR200103351T2 (tr) 2002-06-21
MA26732A1 (fr) 2004-12-20
IS6126A (is) 2001-10-26
PL358538A1 (en) 2004-08-09
AU2935300A (en) 2000-12-12
SK16602001A3 (sk) 2003-03-04
HUP0301287A2 (hu) 2003-08-28
PA8494601A1 (es) 2002-08-29
EP1178784A1 (fr) 2002-02-13
CN1617743A (zh) 2005-05-18
UY26148A1 (es) 2000-12-29
OA11943A (en) 2006-04-12
KR20020010916A (ko) 2002-02-06
IL145955A0 (en) 2002-07-25
HRP20010862A2 (en) 2003-06-30
BR0010820A (pt) 2002-03-05
AR022640A1 (es) 2002-09-04
NO20015651L (no) 2002-01-18
WO2000071107A8 (fr) 2002-01-24
CA2374668A1 (fr) 2000-11-30
MXPA01011978A (es) 2002-05-06
EE200100611A (et) 2003-02-17
BG106208A (en) 2002-09-30
AP2001002326A0 (en) 2001-12-31
HN2000000045A (es) 2001-03-02

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