JPH0637394B2 - 腫瘍治療剤 - Google Patents

腫瘍治療剤

Info

Publication number
JPH0637394B2
JPH0637394B2 JP60273161A JP27316185A JPH0637394B2 JP H0637394 B2 JPH0637394 B2 JP H0637394B2 JP 60273161 A JP60273161 A JP 60273161A JP 27316185 A JP27316185 A JP 27316185A JP H0637394 B2 JPH0637394 B2 JP H0637394B2
Authority
JP
Japan
Prior art keywords
formula
desoxy
compound
difluororibose
amino
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
JP60273161A
Other languages
English (en)
Japanese (ja)
Other versions
JPS61148193A (ja
Inventor
ジエラルド・ブアー・グリンデイー
ラリー・ウエイン・ハーテル
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Eli Lilly and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27101898&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=JPH0637394(B2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Eli Lilly and Co filed Critical Eli Lilly and Co
Publication of JPS61148193A publication Critical patent/JPS61148193A/ja
Publication of JPH0637394B2 publication Critical patent/JPH0637394B2/ja
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16—Purine radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06—Pyrimidine radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Polymers With Sulfur, Phosphorus Or Metals In The Main Chain (AREA)
  • Steroid Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
JP60273161A 1984-12-04 1985-12-03 腫瘍治療剤 Expired - Lifetime JPH0637394B2 (ja)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US67778384A 1984-12-04 1984-12-04
US78641985A 1985-10-10 1985-10-10
US677783 1985-10-10
US786419 1985-10-10

Publications (2)

Publication Number Publication Date
JPS61148193A JPS61148193A (ja) 1986-07-05
JPH0637394B2 true JPH0637394B2 (ja) 1994-05-18

Family

ID=27101898

Family Applications (1)

Application Number Title Priority Date Filing Date
JP60273161A Expired - Lifetime JPH0637394B2 (ja) 1984-12-04 1985-12-03 腫瘍治療剤

Country Status (21)

Country Link
US (1) US5464826A (enExample)
EP (1) EP0184365B1 (enExample)
JP (1) JPH0637394B2 (enExample)
KR (2) KR890003439B1 (enExample)
CN (1) CN1020194C (enExample)
AT (1) ATE92499T1 (enExample)
AU (1) AU581269B2 (enExample)
CA (1) CA1264738A (enExample)
CY (1) CY1806A (enExample)
DE (1) DE3587500T2 (enExample)
DK (1) DK162965C (enExample)
EG (1) EG17765A (enExample)
ES (1) ES8801546A1 (enExample)
GR (1) GR852858B (enExample)
HK (1) HK113693A (enExample)
HU (1) HU194273B (enExample)
IE (1) IE60328B1 (enExample)
IL (1) IL77133A (enExample)
NZ (1) NZ214364A (enExample)
PH (1) PH23172A (enExample)
PT (1) PT81559B (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2008010571A1 (fr) 2006-07-21 2008-01-24 Taiho Pharmaceutical Co., Ltd. Composé nucléosidique de 2'cyanopyrimidine

Families Citing this family (156)

* Cited by examiner, † Cited by third party
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US5464826A (en) 1995-11-07
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