JPH0119395B2 - - Google Patents

Info

Publication number
JPH0119395B2
JPH0119395B2 JP58071315A JP7131583A JPH0119395B2 JP H0119395 B2 JPH0119395 B2 JP H0119395B2 JP 58071315 A JP58071315 A JP 58071315A JP 7131583 A JP7131583 A JP 7131583A JP H0119395 B2 JPH0119395 B2 JP H0119395B2
Authority
JP
Japan
Prior art keywords
crystalline
salt
salts
formula
water
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
JP58071315A
Other languages
English (en)
Japanese (ja)
Other versions
JPS58201792A (ja
Inventor
Aanesuto Baasu Uein
Jon Jashisu Baitootasu
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
PFIZER
Original Assignee
PFIZER
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by PFIZER filed Critical PFIZER
Publication of JPS58201792A publication Critical patent/JPS58201792A/ja
Publication of JPH0119395B2 publication Critical patent/JPH0119395B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/28—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with modified 2-carboxyl group
    • C07D499/32—Esters
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Cephalosporin Compounds (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
JP58071315A 1982-04-23 1983-04-22 結晶性の、サルタミシリンのベンゼンスルホン酸塩 Granted JPS58201792A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US06/371,156 US4432987A (en) 1982-04-23 1982-04-23 Crystalline benzenesulfonate salts of sultamicillin
US371156 1982-04-23

Publications (2)

Publication Number Publication Date
JPS58201792A JPS58201792A (ja) 1983-11-24
JPH0119395B2 true JPH0119395B2 (ref) 1989-04-11

Family

ID=23462725

Family Applications (1)

Application Number Title Priority Date Filing Date
JP58071315A Granted JPS58201792A (ja) 1982-04-23 1983-04-22 結晶性の、サルタミシリンのベンゼンスルホン酸塩

Country Status (27)

Country Link
US (1) US4432987A (ref)
EP (1) EP0092968B1 (ref)
JP (1) JPS58201792A (ref)
KR (1) KR860001279B1 (ref)
AU (1) AU536854B2 (ref)
CA (1) CA1187484A (ref)
CS (1) CS235320B2 (ref)
DD (1) DD209632A5 (ref)
DE (1) DE3362502D1 (ref)
DK (1) DK162168C (ref)
EG (1) EG16412A (ref)
ES (1) ES521728A0 (ref)
FI (1) FI76092C (ref)
GR (1) GR78582B (ref)
HK (1) HK20588A (ref)
HU (1) HU187068B (ref)
IE (1) IE54628B1 (ref)
IL (1) IL68453A (ref)
NO (1) NO156202C (ref)
NZ (1) NZ203988A (ref)
PH (1) PH18035A (ref)
PL (1) PL134978B1 (ref)
PT (1) PT76587B (ref)
SG (1) SG104087G (ref)
SU (1) SU1138030A3 (ref)
YU (1) YU43170B (ref)
ZA (1) ZA832845B (ref)

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EP0247156B1 (en) * 1985-11-18 1993-06-23 Access Pharmaceuticals Inc. Polychelating agents for image and spectral enhancement (and spectral shift)
US5336762A (en) * 1985-11-18 1994-08-09 Access Pharmaceuticals, Inc. Polychelating agents for image and spectral enhancement (and spectral shift)
KR910009271B1 (ko) * 1989-06-20 1991-11-08 김영설 1,1-디옥소페닐실라노일 옥시메틸 D-6-[α-(메틸렌아미노)페닐-아세트아미도]-페니실라네이트와 그의 파라-톨루엔술폰산염
AU700545B2 (en) * 1994-05-02 1999-01-07 Shionogi & Co., Ltd. Crystal of pyrrolidylthiocarbapenem derivative, lyophilized preparation containing said crystal, and process for producing the same
JP3382159B2 (ja) * 1998-08-05 2003-03-04 株式会社東芝 情報記録媒体とその再生方法及び記録方法
ZA200501418B (en) 2002-08-29 2006-10-25 Taisho Pharmaceutical Co Ltd Benzenesulfonate salts of 4-fluoro-2-cyanopyrrolidine derivatives
BRPI0408716B1 (pt) * 2003-03-27 2017-08-29 Basilea Pharmaceutica Ag. Cefalosporin in crystalline form, process for its preparation and its uses, and preparation of cephalosporin
EP1677759A1 (en) * 2003-10-31 2006-07-12 Alza Corporation Compositions and dosage forms for enhanced absorption of gabapentin and pregabalin
FR2877696B1 (fr) 2004-11-09 2009-09-18 Renault Sas Dispositif et procede d'estimation en temps reel de l'angle de debut de combustion d'un moteur a combustion interne
SA08290520B1 (ar) 2007-08-22 2012-02-22 استرازينيكا ايه بي مشتقات سيكلو بروبيل أميد وتركيبات صيدلية تحتوي عليها لعلاج حالة مرضية سببها مستقبلات هيستامين h3
TWI469971B (zh) 2007-10-26 2015-01-21 Univ California 二芳基乙內醯脲類化合物
US20110288142A1 (en) * 2009-01-30 2011-11-24 Chen Pingyun Y CRYSTALLINE N--5-chloro-4-(4-chloro-1-methyl-1H-pyrazol-5-yl)-2-thiophenecarboxamide hydrochloride
TW201039825A (en) 2009-02-20 2010-11-16 Astrazeneca Ab Cyclopropyl amide derivatives 983
JP2012532886A (ja) * 2009-07-10 2012-12-20 エボルバ アクチェンゲゼルシャフト ジイン組成物
RU2012139082A (ru) * 2010-02-18 2014-03-27 Астразенека Аб Способы получения производных циклопропиламида и связанных с ними промежуточных соединений
JP5746718B2 (ja) * 2010-02-18 2015-07-08 アストラゼネカ・アクチエボラーグＡｓｔｒａｚｅｎｅｃａ Ａｋｔｉｅｂｏｌａｇ シクロプロピルアミド誘導体からなる固体形態
US9518004B2 (en) * 2012-12-03 2016-12-13 Kaneka Corporation Reduced coenzyme Q10 derivative and method for production thereof
KR20230159631A (ko) * 2013-09-05 2023-11-21 미쓰비시 타나베 파마 코퍼레이션 신규한 결정성 아릴알킬아민 화합물 및 그의 제조 방법
CN111825717A (zh) 2014-10-21 2020-10-27 阿瑞雅德制药公司 5-氯-n4-[2-(二甲基磷酰基)苯基]-n2-{2-甲氧基-4-[4-(4-甲基哌嗪-1-基)哌啶-1-基]苯基}嘧啶-2,4-二胺的晶形
CN104958318A (zh) * 2015-08-04 2015-10-07 青岛蓝盛洋医药生物科技有限责任公司 一种治疗感染性疾病的药物舒巴坦钠组合物
EP3778567A1 (en) * 2016-01-22 2021-02-17 Sandoz Ag Crystalline eravacycline bis-hydrochloride
MX389964B (es) * 2016-07-07 2025-03-19 Cyclerion Therapeutics Inc Formas sólidas de un estimulador de guanilato ciclasa soluble (sgc).
EP3703686A4 (en) * 2017-10-30 2021-11-17 Theracaine LLC HYDROPHOBIC ARENE SULFONATE SALTS
US11186556B1 (en) * 2018-10-16 2021-11-30 Celgene Corporation Salts of a thiazolidinone compound, solid forms, compositions and methods of use thereof
UA119735C2 (uk) 2018-12-20 2019-07-25 Анатолій Семенович Редер Фармацевтична сполука, спосіб її отримання та застосування як лікарського засобу
USD998740S1 (en) 2019-02-13 2023-09-12 Hs Produkt D.O.O. Firearm
USD1071069S1 (en) 2019-02-13 2025-04-15 Hs Produkt D.O.O. Stippled textured body for a firearm or the like
USD994822S1 (en) 2019-02-13 2023-08-08 Hs Produkt D.O.O. Pistol
USD994821S1 (en) 2019-02-13 2023-08-08 Hs Produkt D.O.O. Pistol
USD1077123S1 (en) 2019-02-13 2025-05-27 Hs Produkt D.O.O. Firearm sight
USD1057880S1 (en) 2019-08-09 2025-01-14 Hs Produkt D.O.O. Pistol
CN117120034A (zh) * 2021-02-15 2023-11-24 普洛佩拉治疗公司 阿比特龙前药
USD1049292S1 (en) * 2021-04-06 2024-10-29 Springfield, Inc. Pistol
WO2022237808A1 (zh) * 2021-05-12 2022-11-17 浙江龙传生物医药科技有限公司 吡咯并嘧啶类化合物的晶型及其制备方法
EP4337659A1 (en) * 2021-05-14 2024-03-20 Global Blood Therapeutics, Inc. Solid forms of a modulator of hemoglobin
JP2024523518A (ja) * 2021-06-24 2024-06-28 サンド・アクチエンゲゼルシヤフト ソトラシブの結晶形態
USD1069964S1 (en) 2021-11-03 2025-04-08 Hs Produkt D.O.O. Pistol slide
US12410155B2 (en) * 2021-12-28 2025-09-09 Zhejiang Yangli Pharmaceutical Technology Co., Ltd. Salt form and crystal form of tetrahydrocyclohepta indazole compound
US20250388537A1 (en) * 2022-05-20 2025-12-25 Caamtech, Inc. Tryptamine derivatives
USD1072997S1 (en) 2022-08-29 2025-04-29 Springfield, Inc. Firearm
USD1057882S1 (en) 2022-08-29 2025-01-14 Springfield, Inc. Combined serrations for a firearm slide
USD1061781S1 (en) 2022-11-30 2025-02-11 Hs Produkt D.O.O. Pistol
ZAA202301175S (en) 2023-04-28 2024-06-26 Hs Produkt D O O Firearm
TW202517650A (zh) * 2023-07-17 2025-05-01 美商庫拉腫瘤技術股份有限公司 包含ｍｅｎｉｎ抑制劑之醫藥組合物
KR20260039698A (ko) * 2023-07-17 2026-03-20 쿠라 온콜로지, 인크. 결정 형태의 메닌 억제제

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US4234579A (en) * 1977-06-07 1980-11-18 Pfizer Inc. Penicillanic acid 1,1-dioxides as β-lactamase inhibitors
IE49881B1 (en) * 1979-02-13 1986-01-08 Leo Pharm Prod Ltd B-lactam intermediates
KR830001903B1 (ko) * 1979-02-13 1983-09-19 레오 파마슈티칼 프로덕츠 리미티드 페니실란산유도체의 제조방법
US4244951A (en) * 1979-05-16 1981-01-13 Pfizer Inc. Bis-esters of methanediol with penicillins and penicillanic acid 1,1-dioxide
IE51516B1 (en) * 1980-10-06 1987-01-07 Leo Pharm Prod Ltd 1,1-dioxapenicillanoyloxymethyl 6-(d-alpha-amino-alpha-phenylacetamido)penicillanate napsylate
GB2084572B (en) * 1980-10-06 1984-07-11 Leo Pharm Prod Ltd 1,1-dioxopenicillanoyloxymethyl 6-(d-aphenylacetamido)penicillanate napsylate
IL64009A (en) * 1980-10-31 1984-09-30 Rech Applications Therap Crystalline 1,1-dioxopenicillanoyloxymethyl 6-(d-alpha-amino-alpha-phenylacetamido)penicillanate tosylate hydrates,their production and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
DD209632A5 (de) 1984-05-16
EP0092968B1 (en) 1986-03-12
EP0092968A1 (en) 1983-11-02
IE54628B1 (en) 1989-12-20
IE830926L (en) 1983-10-23
KR860001279B1 (ko) 1986-09-05
FI76092B (fi) 1988-05-31
PL241553A1 (en) 1983-11-21
SU1138030A3 (ru) 1985-01-30
ES8406075A1 (es) 1984-07-01
EG16412A (en) 1989-03-30
FI831392A0 (fi) 1983-04-22
KR840004437A (ko) 1984-10-15
ES521728A0 (es) 1984-07-01
IL68453A0 (en) 1983-07-31
YU90483A (en) 1986-04-30
PT76587B (en) 1986-02-27
DE3362502D1 (en) 1986-04-17
HK20588A (en) 1988-03-25
PL134978B1 (en) 1985-09-30
DK101783D0 (da) 1983-02-28
CA1187484A (en) 1985-05-21
YU43170B (en) 1989-04-30
AU536854B2 (en) 1984-05-24
FI76092C (fi) 1988-09-09
NO831430L (no) 1983-10-24
NZ203988A (en) 1986-01-24
PT76587A (en) 1983-05-01
CS235320B2 (en) 1985-05-15
FI831392L (fi) 1983-10-24
HU187068B (en) 1985-11-28
DK162168C (da) 1992-03-02
IL68453A (en) 1986-08-31
ZA832845B (en) 1984-11-28
SG104087G (en) 1988-07-15
AU1387183A (en) 1983-11-17
NO156202B (no) 1987-05-04
US4432987A (en) 1984-02-21
NO156202C (no) 1987-08-19
JPS58201792A (ja) 1983-11-24
PH18035A (en) 1985-03-06
GR78582B (ref) 1984-09-27
DK101783A (da) 1983-10-24
DK162168B (da) 1991-09-23

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