JP7351851B2 - レチノイド関連オルファン受容体ガンマ（ＲＯＲγ）のモジュレーターとしてのベンジイミダゾール誘導体およびそれらの医薬品用途 - Google Patents

レチノイド関連オルファン受容体ガンマ（ＲＯＲγ）のモジュレーターとしてのベンジイミダゾール誘導体およびそれらの医薬品用途 Download PDF

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JP7351851B2
JP7351851B2 JP2020560186A JP2020560186A JP7351851B2 JP 7351851 B2 JP7351851 B2 JP 7351851B2 JP 2020560186 A JP2020560186 A JP 2020560186A JP 2020560186 A JP2020560186 A JP 2020560186A JP 7351851 B2 JP7351851 B2 JP 7351851B2
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alkyl
cycloalkyl
heterocyclyl
aryl
heteroaryl
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JP2021522262A (ja
JP2021522262A5 (https=
JPWO2019213470A5 (https=
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インファ ヤン
ミンシェン チャン
ドン リウ
フェンキ チャン
スーシン リウ
ルーミン チャン
フェン ヘ
ウェイカン タオ
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Jiangsu Hengrui Medicine Co Ltd
Shanghai Hengrui Pharmaceutical Co Ltd
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Jiangsu Hengrui Medicine Co Ltd
Shanghai Hengrui Pharmaceutical Co Ltd
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JP2020560186A 2018-05-03 2019-05-03 レチノイド関連オルファン受容体ガンマ（ＲＯＲγ）のモジュレーターとしてのベンジイミダゾール誘導体およびそれらの医薬品用途 Active JP7351851B2 (ja)

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US201862666312P 2018-05-03 2018-05-03
US62/666,312 2018-05-03
PCT/US2019/030526 WO2019213470A1 (en) 2018-05-03 2019-05-03 Benzimidazole derivatives as modulators of retinoid-related orphan receptor gamma (rorϒ) and pharmaceutical uses thereof

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JP2021522262A JP2021522262A (ja) 2021-08-30
JP2021522262A5 JP2021522262A5 (https=) 2022-05-12
JPWO2019213470A5 JPWO2019213470A5 (https=) 2022-05-12
JP7351851B2 true JP7351851B2 (ja) 2023-09-27

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US (2) US11512055B2 (https=)
EP (1) EP3781161B1 (https=)
JP (1) JP7351851B2 (https=)
KR (1) KR102709804B1 (https=)
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AU (1) AU2019262169B2 (https=)
BR (1) BR112020021967A2 (https=)
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MY208400A (en) * 2018-05-03 2025-05-07 Shanghai hengrui pharmaceutical co ltd Benzimidazole derivatives as modulators of retinoid-related orphan receptor gamma (ror) and pharmaceutical uses thereof
US20220411380A1 (en) * 2019-10-31 2022-12-29 Jiangsu Hengrui Medicine Co., Ltd. ACID ADDITION SALT OF RORy REGULATOR
CN112745268B (zh) * 2019-10-31 2022-09-16 江苏恒瑞医药股份有限公司 苯并咪唑衍生物的晶型及制备方法
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