TWI818985B - 作為類視色素相關孤兒受體γ（ＲＯＲγ）調節劑之苯并咪唑衍生物及其醫藥用途 - Google Patents

作為類視色素相關孤兒受體γ（ＲＯＲγ）調節劑之苯并咪唑衍生物及其醫藥用途 Download PDF

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TWI818985B
TWI818985B TW108115438A TW108115438A TWI818985B TW I818985 B TWI818985 B TW I818985B TW 108115438 A TW108115438 A TW 108115438A TW 108115438 A TW108115438 A TW 108115438A TW I818985 B TWI818985 B TW I818985B
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cycloalkyl
heterocyclyl
aryl
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TW108115438A
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TW202014185A (zh
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銀發 燕
民生 張
東 劉
鳳岐 張
蘇星 劉
儒民 張
峰 賀
維康 陶
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中國大陸商江蘇恒瑞醫藥股份有限公司
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TW108115438A 2018-05-03 2019-05-03 作為類視色素相關孤兒受體γ（ＲＯＲγ）調節劑之苯并咪唑衍生物及其醫藥用途 TWI818985B (zh)

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US201862666312P 2018-05-03 2018-05-03
US62/666,312 2018-05-03

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MY208400A (en) * 2018-05-03 2025-05-07 Shanghai hengrui pharmaceutical co ltd Benzimidazole derivatives as modulators of retinoid-related orphan receptor gamma (ror) and pharmaceutical uses thereof
US20220411380A1 (en) * 2019-10-31 2022-12-29 Jiangsu Hengrui Medicine Co., Ltd. ACID ADDITION SALT OF RORy REGULATOR
CN112745268B (zh) * 2019-10-31 2022-09-16 江苏恒瑞医药股份有限公司 苯并咪唑衍生物的晶型及制备方法
TW202136238A (zh) * 2020-01-06 2021-10-01 大陸商廣東東陽光藥業有限公司 RORγt抑制劑及其製備方法和用途
TW202136237A (zh) * 2020-01-06 2021-10-01 大陸商廣東東陽光藥業有限公司 RORγt抑制劑及其製備方法和用途
CN111269126B (zh) * 2020-03-12 2023-04-07 北京理工大学重庆创新中心 一种熔铸载体1,2-二氟-4,5-二硝基苯的制备方法
CA3179686A1 (en) * 2020-04-07 2021-10-14 UCB Biopharma SRL Difluorocyclohexyl derivatives as il-17 modulators
TW202146381A (zh) * 2020-05-15 2021-12-16 大陸商上海輝启生物醫藥科技有限公司 可用作RORγ調節劑的聯芳基類化合物
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