CN116514722A - 作为维甲酸相关孤儿受体γ（RORγ）的调节剂的苯并咪唑衍生物及其药物用途 - Google Patents

作为维甲酸相关孤儿受体γ（RORγ）的调节剂的苯并咪唑衍生物及其药物用途 Download PDF

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Publication number
CN116514722A
CN116514722A CN202310017171.4A CN202310017171A CN116514722A CN 116514722 A CN116514722 A CN 116514722A CN 202310017171 A CN202310017171 A CN 202310017171A CN 116514722 A CN116514722 A CN 116514722A
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alkyl
cycloalkyl
heteroaryl
aryl
heterocyclyl
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Chinese (zh)
Inventor
燕银发
张民生
刘�东
张凤岐
刘苏星
张儒民
贺峰
陶维康
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Jiangsu Hengrui Medicine Co Ltd
Shanghai Hengrui Pharmaceutical Co Ltd
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Jiangsu Hengrui Medicine Co Ltd
Shanghai Hengrui Pharmaceutical Co Ltd
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CN202310017171.4A 2018-05-03 2019-05-03 作为维甲酸相关孤儿受体γ（RORγ）的调节剂的苯并咪唑衍生物及其药物用途 Pending CN116514722A (zh)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201862666312P 2018-05-03 2018-05-03
US62/666,312 2018-05-03
CN201980027956.1A CN112135611B (zh) 2018-05-03 2019-05-03 作为维甲酸相关孤儿受体γ（RORγ）的调节剂的苯并咪唑衍生物及其药物用途
PCT/US2019/030526 WO2019213470A1 (en) 2018-05-03 2019-05-03 Benzimidazole derivatives as modulators of retinoid-related orphan receptor gamma (rorϒ) and pharmaceutical uses thereof

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CN201980027956.1A Active CN112135611B (zh) 2018-05-03 2019-05-03 作为维甲酸相关孤儿受体γ（RORγ）的调节剂的苯并咪唑衍生物及其药物用途

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US (2) US11512055B2 (https=)
EP (1) EP3781161B1 (https=)
JP (1) JP7351851B2 (https=)
KR (1) KR102709804B1 (https=)
CN (2) CN116514722A (https=)
AU (1) AU2019262169B2 (https=)
BR (1) BR112020021967A2 (https=)
CA (1) CA3097519A1 (https=)
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MY208400A (en) * 2018-05-03 2025-05-07 Shanghai hengrui pharmaceutical co ltd Benzimidazole derivatives as modulators of retinoid-related orphan receptor gamma (ror) and pharmaceutical uses thereof
US20220411380A1 (en) * 2019-10-31 2022-12-29 Jiangsu Hengrui Medicine Co., Ltd. ACID ADDITION SALT OF RORy REGULATOR
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