JP6893173B2 - Ｃｎｓ障害を処置するための組成物および方法 - Google Patents
Ｃｎｓ障害を処置するための組成物および方法 Download PDFInfo
- Publication number
- JP6893173B2 JP6893173B2 JP2017528154A JP2017528154A JP6893173B2 JP 6893173 B2 JP6893173 B2 JP 6893173B2 JP 2017528154 A JP2017528154 A JP 2017528154A JP 2017528154 A JP2017528154 A JP 2017528154A JP 6893173 B2 JP6893173 B2 JP 6893173B2
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- substituted
- unsubstituted
- compound
- alkyl
- hydrogen
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- 0 CC(CC1)([C@@](CC2)C(CC3)C1[C@@](CC1)[C@@]3C[C@@]1(O)I)[C@]2C(C1(CCC*=C)*CC1)=O Chemical compound CC(CC1)([C@@](CC2)C(CC3)C1[C@@](CC1)[C@@]3C[C@@]1(O)I)[C@]2C(C1(CCC*=C)*CC1)=O 0.000 description 24
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
- C07J41/0055—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the 17-beta position being substituted by an uninterrupted chain of at least three carbon atoms which may or may not be branched, e.g. cholane or cholestane derivatives, optionally cyclised, e.g. 17-beta-phenyl or 17-beta-furyl derivatives
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J17/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, having an oxygen-containing hetero ring not condensed with the cyclopenta(a)hydrophenanthrene skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J3/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
- C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J33/00—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
- C07J33/002—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
- C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J9/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
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Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2021130698A (ja) * | 2014-11-27 | 2021-09-09 | セージ セラピューティクス， インコーポレイテッド | Ｃｎｓ障害を処置するための組成物および方法 |
| JP7186259B2 (ja) | 2014-11-27 | 2022-12-08 | セージ セラピューティクス， インコーポレイテッド | Ｃｎｓ障害を処置するための組成物および方法 |
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| HRP20200840T1 (hr) | 2020-11-13 |
| US10774108B2 (en) | 2020-09-15 |
| ME03749B (me) | 2021-04-20 |
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| DK3224269T3 (da) | 2020-05-25 |
| JP2017535586A (ja) | 2017-11-30 |
| US20170342102A1 (en) | 2017-11-30 |
| WO2016082789A1 (en) | 2016-06-02 |
| PL3224269T3 (pl) | 2020-08-24 |
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| US20250042934A1 (en) | 2025-02-06 |
| HUE049014T2 (hu) | 2020-09-28 |
| EP3719029A1 (en) | 2020-10-07 |
| US20210017218A1 (en) | 2021-01-21 |
| RS60343B1 (sr) | 2020-07-31 |
| PT3224269T (pt) | 2020-06-01 |
| EP3224269A1 (en) | 2017-10-04 |
| CY1123200T1 (el) | 2021-10-29 |
| EP3224269A4 (en) | 2018-07-25 |
| SMT202000276T1 (it) | 2020-07-08 |
| LT3224269T (lt) | 2020-07-10 |
| SI3224269T1 (sl) | 2020-10-30 |
| JP2021130698A (ja) | 2021-09-09 |
| US11945836B2 (en) | 2024-04-02 |
| ES2793237T3 (es) | 2020-11-13 |
| JP2023022187A (ja) | 2023-02-14 |
| US20230279043A1 (en) | 2023-09-07 |
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