JP6585057B2 - ５−フルオロ−４−イミノ−３−（アルキル／置換アルキル）−１−（アリールスルホニル）−３，４−ジヒドロピリミジン−２（１ｈ）−オンおよびそれらの調製方法 - Google Patents
５−フルオロ−４−イミノ−３−（アルキル／置換アルキル）−１−（アリールスルホニル）−３，４−ジヒドロピリミジン−２（１ｈ）−オンおよびそれらの調製方法 Download PDFInfo
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- JP6585057B2 JP6585057B2 JP2016543735A JP2016543735A JP6585057B2 JP 6585057 B2 JP6585057 B2 JP 6585057B2 JP 2016543735 A JP2016543735 A JP 2016543735A JP 2016543735 A JP2016543735 A JP 2016543735A JP 6585057 B2 JP6585057 B2 JP 6585057B2
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
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- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
- C07D333/08—Hydrogen atoms or radicals containing only hydrogen and carbon atoms
- C07D333/10—Thiophene
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Agronomy & Crop Science (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- General Health & Medical Sciences (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Detergent Compositions (AREA)
- Cosmetics (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201361922582P | 2013-12-31 | 2013-12-31 | |
| US201361922572P | 2013-12-31 | 2013-12-31 | |
| US61/922,572 | 2013-12-31 | ||
| US61/922,582 | 2013-12-31 | ||
| PCT/US2014/072569 WO2015103144A1 (en) | 2013-12-31 | 2014-12-29 | 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2019160781A Division JP2019218396A (ja) | 2013-12-31 | 2019-09-04 | ５−フルオロ−４−イミノ−３−（アルキル／置換アルキル）−１−（アリールスルホニル）−３，４−ジヒドロピリミジン−２（１ｈ）−オンおよびそれらの調製方法 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2017501197A JP2017501197A (ja) | 2017-01-12 |
| JP2017501197A5 JP2017501197A5 (enExample) | 2018-02-15 |
| JP6585057B2 true JP6585057B2 (ja) | 2019-10-02 |
Family
ID=53480979
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2016543735A Active JP6585057B2 (ja) | 2013-12-31 | 2014-12-29 | ５−フルオロ−４−イミノ−３−（アルキル／置換アルキル）−１−（アリールスルホニル）−３，４−ジヒドロピリミジン−２（１ｈ）−オンおよびそれらの調製方法 |
| JP2016543746A Active JP6804297B2 (ja) | 2013-12-31 | 2014-12-29 | ５−フルオロ−４−イミノ−３−（アルキル／置換アルキル）−１−（アリールスルホニル）−３，４−ジヒドロピリミジン−２（１ｈ）−オンおよびそれらの調製方法 |
| JP2019160781A Withdrawn JP2019218396A (ja) | 2013-12-31 | 2019-09-04 | ５−フルオロ−４−イミノ−３−（アルキル／置換アルキル）−１−（アリールスルホニル）−３，４−ジヒドロピリミジン−２（１ｈ）−オンおよびそれらの調製方法 |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2016543746A Active JP6804297B2 (ja) | 2013-12-31 | 2014-12-29 | ５−フルオロ−４−イミノ−３−（アルキル／置換アルキル）−１−（アリールスルホニル）−３，４−ジヒドロピリミジン−２（１ｈ）−オンおよびそれらの調製方法 |
| JP2019160781A Withdrawn JP2019218396A (ja) | 2013-12-31 | 2019-09-04 | ５−フルオロ−４−イミノ−３−（アルキル／置換アルキル）−１−（アリールスルホニル）−３，４−ジヒドロピリミジン−２（１ｈ）−オンおよびそれらの調製方法 |
Country Status (24)
| Country | Link |
|---|---|
| US (8) | US20150183749A1 (enExample) |
| EP (4) | EP3862347A1 (enExample) |
| JP (3) | JP6585057B2 (enExample) |
| CN (4) | CN111217759A (enExample) |
| AP (1) | AP2016009342A0 (enExample) |
| AU (2) | AU2014373959B2 (enExample) |
| BR (2) | BR102014033010B1 (enExample) |
| CA (2) | CA2935601C (enExample) |
| CL (1) | CL2016001677A1 (enExample) |
| CR (2) | CR20160343A (enExample) |
| DO (1) | DOP2016000163A (enExample) |
| EA (2) | EA201691353A1 (enExample) |
| EC (1) | ECSP16064249A (enExample) |
| IL (3) | IL246512B (enExample) |
| MX (2) | MX375727B (enExample) |
| NI (1) | NI201600094A (enExample) |
| NZ (2) | NZ722439A (enExample) |
| PE (1) | PE20161174A1 (enExample) |
| PH (1) | PH12016501284A1 (enExample) |
| SG (2) | SG11201605372QA (enExample) |
| TW (2) | TWI722979B (enExample) |
| UA (2) | UA129860C2 (enExample) |
| UY (2) | UY35943A (enExample) |
| WO (2) | WO2015103144A1 (enExample) |
Families Citing this family (28)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN104902757B (zh) | 2012-12-28 | 2019-01-08 | 阿达玛马克西姆股份有限公司 | N-(取代的)-5-氟-4-亚氨基-3-甲基-2-氧代-3,4-二氢嘧啶-1(2h)-羧酸酯衍生物 |
| JP6258969B2 (ja) | 2012-12-28 | 2018-01-10 | アダマ・マクテシム・リミテッド | Ｎ−（置換）−５−フルオロ−４−イミノ−３−メチル−２−オキソ−３，４−ジヒドロピリミジン−１（２ｈ）−カルボキサミド誘導体 |
| CN112094262A (zh) | 2012-12-31 | 2020-12-18 | 阿达玛马克西姆股份有限公司 | 作为杀真菌剂的化合物 |
| CR20160344A (es) | 2013-12-31 | 2016-12-19 | Adama Makhteshim Ltd | Mezclas fungicidas sinérgicas para el control fúngico en cereales |
| UA129860C2 (uk) | 2013-12-31 | 2025-08-27 | Адама Махтешім Лтд. | 5-фтор-4-іміно-3-(алкіл/заміщений алкіл)-1-(арилсульфоніл)-3,4-дигідропіримідин-2(1h)-он і способи його одержання |
| UY36964A (es) | 2015-10-27 | 2017-05-31 | Bayer Cropscience Ag | Combinaciones de principios activos que comprenden un derivado de (tio) carboxamida y un compuesto funguicida |
| JP6922271B2 (ja) * | 2016-03-11 | 2021-08-18 | 住友化学株式会社 | 植物病害防除組成物及び植物病害防除方法 |
| IL271950B2 (en) * | 2017-07-17 | 2024-06-01 | Adama Makhteshim Ltd | Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one |
| CA3118729A1 (en) * | 2018-11-05 | 2020-05-14 | Adama Makhteshim Ltd. | Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof |
| MX2022000944A (es) | 2019-07-22 | 2022-04-06 | Adama Makhteshim Ltd | Combinaciones, mezclas y composiciones fungicidas y usos de las mismas. |
| US12466796B2 (en) | 2019-09-23 | 2025-11-11 | Adama Makhteshim Ltd. | Process for preparing 5-(fluoro-4-imino-3-methyl)-1-tosyl-3,4 dihydropyrimidine-(1H)-one and derivatives of the compound |
| EP4118073A1 (en) * | 2020-03-09 | 2023-01-18 | Adama Makhteshim Ltd. | Process for preparing 5-fluoro-4-imino-3-methyl-1-(toluene-4-sulfonyl)-3,4-dihydro-1h-pyrimidin-2-one |
| PY2135531A (es) * | 2020-05-04 | 2022-02-01 | Adama Makhteshim Ltd | Mezclas y composiciones que comprenden 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2-ona, y métodos de uso de las mismas |
| US20230270113A1 (en) | 2020-07-08 | 2023-08-31 | Adama Makhteshim Ltd. | Fungicidal mixtures |
| CA3206570A1 (en) | 2021-01-27 | 2022-08-04 | Alexandra ROSENMUND | 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2(1 h)-one for controlling plant diseases |
| MX2023012897A (es) | 2021-05-04 | 2023-12-06 | Adama Makhteshim Ltd | Formas cristalinas de 5-fluoro-4-imino-3-metil-1-tosil-3,4- dihidropirimidin-2-ona, y mezclas, composiciones y metodos de uso de las mismas. |
| EP4402131A1 (en) | 2021-09-15 | 2024-07-24 | Adama Makhteshim Ltd. | Process for preparing 5-fluoro-4-imino-3-methyl-1-(toluene-4-sulfonyl)-3,4-dihydro-1h-pyrimidin-2-one |
| UY40172A (es) | 2022-03-03 | 2023-10-13 | Adama Makhteshim Ltd | Combinaciones, mezclas y composiciones fungicidas y usos de las mismas |
| EP4531570A1 (en) | 2022-05-26 | 2025-04-09 | Adama Makhteshim Ltd. | Fungicidal combinations, mixtures and compositions and uses thereof |
| EP4565066A1 (en) | 2022-08-03 | 2025-06-11 | Adama Makhteshim Ltd. | 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2(1h)-one for fungicide-resistant fungus |
| CN120882310A (zh) | 2023-03-09 | 2025-10-31 | 安道麦马克西姆有限公司 | 杀真菌组合、混合物及组合物以及其用途 |
| EP4680029A1 (en) | 2023-03-14 | 2026-01-21 | Adama Makhteshim Ltd. | Liquid compositions containing 5-(fluoro-4-imino-3-methyl)-1-tosyl-3,4 dihydropyrimidine-(1h)-one and derivatives thereof and a uv absorber |
| EP4683910A1 (en) | 2023-03-23 | 2026-01-28 | Adama Makhteshim Ltd. | Process for preparing 5-fluoro-4-imino-3-methyl-1-(toluene-4-sulfonyl)-3,4-dihydro-1h-pyrimidin-2-one |
| AU2024334814A1 (en) | 2023-08-31 | 2026-03-12 | Adama Makhteshim Ltd. | Fungicidal combinations, mixtures and compositions and uses thereo |
| IL308593A (en) | 2023-11-15 | 2025-06-01 | Adama Makhteshim Ltd | Reducing environmental impact of fungicidal enhancement |
| WO2025114931A1 (en) | 2023-11-28 | 2025-06-05 | Adama Makhteshim Ltd. | Fungicidal combinations, mixtures and compositions and uses thereof |
| WO2025203024A1 (en) | 2024-03-26 | 2025-10-02 | Adama Makhteshim Ltd. | Process for preparing 5-fluoro-4-imino-3-methyl-1-(toluene-4-sulfonyl)-3,4-dihydro-1h-pyrimidin-2-one |
| WO2026038217A1 (en) | 2024-08-15 | 2026-02-19 | Adama Makhteshim Ltd. | Mixtures and compositions comprising flumetylsulforim and methods of use thereof |
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| CN104902757B (zh) * | 2012-12-28 | 2019-01-08 | 阿达玛马克西姆股份有限公司 | N-(取代的)-5-氟-4-亚氨基-3-甲基-2-氧代-3,4-二氢嘧啶-1(2h)-羧酸酯衍生物 |
| WO2014105821A1 (en) | 2012-12-28 | 2014-07-03 | Dow Agrosciences Llc | 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1h)-one derivatives |
| CN112094262A (zh) * | 2012-12-31 | 2020-12-18 | 阿达玛马克西姆股份有限公司 | 作为杀真菌剂的化合物 |
| CR20160344A (es) | 2013-12-31 | 2016-12-19 | Adama Makhteshim Ltd | Mezclas fungicidas sinérgicas para el control fúngico en cereales |
| UA129860C2 (uk) | 2013-12-31 | 2025-08-27 | Адама Махтешім Лтд. | 5-фтор-4-іміно-3-(алкіл/заміщений алкіл)-1-(арилсульфоніл)-3,4-дигідропіримідин-2(1h)-он і способи його одержання |
| MA41272A (fr) | 2014-12-23 | 2017-10-31 | Adama Makhteshim Ltd | 5-fluoro-4-imino-3-(alkyle/alkyle substitué)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one en tant que traitement des semences |
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