CA2935594C - 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation - Google Patents
5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation Download PDFInfo
- Publication number
- CA2935594C CA2935594C CA2935594A CA2935594A CA2935594C CA 2935594 C CA2935594 C CA 2935594C CA 2935594 A CA2935594 A CA 2935594A CA 2935594 A CA2935594 A CA 2935594A CA 2935594 C CA2935594 C CA 2935594C
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- Prior art keywords
- compound
- formula
- molar ratio
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- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
- C07D333/08—Hydrogen atoms or radicals containing only hydrogen and carbon atoms
- C07D333/10—Thiophene
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Wood Science & Technology (AREA)
- Environmental Sciences (AREA)
- Plant Pathology (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- General Health & Medical Sciences (AREA)
- Agronomy & Crop Science (AREA)
- Zoology (AREA)
- Pest Control & Pesticides (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Detergent Compositions (AREA)
- Cosmetics (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201361922572P | 2013-12-31 | 2013-12-31 | |
| US201361922582P | 2013-12-31 | 2013-12-31 | |
| US61/922,572 | 2013-12-31 | ||
| US61/922,582 | 2013-12-31 | ||
| PCT/US2014/072566 WO2015103142A1 (en) | 2013-12-31 | 2014-12-29 | 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1- (arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CA2935594A1 CA2935594A1 (en) | 2015-07-09 |
| CA2935594C true CA2935594C (en) | 2022-05-03 |
Family
ID=53480979
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA2935594A Active CA2935594C (en) | 2013-12-31 | 2014-12-29 | 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation |
| CA2935601A Active CA2935601C (en) | 2013-12-31 | 2014-12-29 | 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA2935601A Active CA2935601C (en) | 2013-12-31 | 2014-12-29 | 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation |
Country Status (24)
| Country | Link |
|---|---|
| US (8) | US20150183749A1 (enExample) |
| EP (4) | EP3862346A1 (enExample) |
| JP (3) | JP6804297B2 (enExample) |
| CN (4) | CN106061972B (enExample) |
| AP (1) | AP2016009342A0 (enExample) |
| AU (2) | AU2014373959B2 (enExample) |
| BR (2) | BR102014033037B1 (enExample) |
| CA (2) | CA2935594C (enExample) |
| CL (1) | CL2016001677A1 (enExample) |
| CR (2) | CR20210172A (enExample) |
| DO (1) | DOP2016000163A (enExample) |
| EA (2) | EA201691353A1 (enExample) |
| EC (1) | ECSP16064249A (enExample) |
| IL (3) | IL246512B (enExample) |
| MX (2) | MX392211B (enExample) |
| NI (1) | NI201600094A (enExample) |
| NZ (2) | NZ722438A (enExample) |
| PE (1) | PE20161174A1 (enExample) |
| PH (1) | PH12016501284A1 (enExample) |
| SG (2) | SG11201605372QA (enExample) |
| TW (2) | TWI722979B (enExample) |
| UA (2) | UA129860C2 (enExample) |
| UY (2) | UY35942A (enExample) |
| WO (2) | WO2015103142A1 (enExample) |
Families Citing this family (27)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US9321734B2 (en) | 2012-12-28 | 2016-04-26 | Dow Agrosciences Llc | N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1(2H)-carboxamide derivatives |
| KR20150103096A (ko) | 2012-12-28 | 2015-09-09 | 다우 아그로사이언시즈 엘엘씨 | N-(치환된)-5-플루오로-4-이미노-3-메틸-2-옥소-3,4-디히드로피리미딘-1(2h)-카르복실레이트 유도체 |
| US9642368B2 (en) | 2012-12-31 | 2017-05-09 | Adama Makhteshim Ltd. | 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1H)-one derivatives as fungicides |
| AU2014373853A1 (en) | 2013-12-31 | 2016-08-11 | Adama Makhteshim Ltd. | Synergistic fungicidal mixtures and compositions for fungal control |
| MX392211B (es) | 2013-12-31 | 2025-03-21 | Adama Makhteshim Ltd | 5-flúor-4-imino-3-(alquil/alquilo sustituido)-1-(arilsulfonil)-3,4-dihidropirimidin-2(1h)-ona y los procesos para su preparación. |
| UY36964A (es) | 2015-10-27 | 2017-05-31 | Bayer Cropscience Ag | Combinaciones de principios activos que comprenden un derivado de (tio) carboxamida y un compuesto funguicida |
| JP6922271B2 (ja) * | 2016-03-11 | 2021-08-18 | 住友化学株式会社 | 植物病害防除組成物及び植物病害防除方法 |
| CN118515619A (zh) | 2017-07-17 | 2024-08-20 | 阿达玛克西姆股份有限公司 | 5-氟-4-亚氨基-3-甲基-1-甲苯磺酰基-3,4-二氢嘧啶-2-酮的多晶型物 |
| EA202191250A1 (ru) | 2018-11-05 | 2021-08-20 | Адама Мактешим Лтд. | Смеси и композиции, включающие 5-фтор-4-имино-3-метил-1-тозил-3,4-дигидропиримидин-2-он, и способы их применения |
| TWI765301B (zh) | 2019-07-22 | 2022-05-21 | 以色列商亞當馬赫特希姆有限公司 | 殺真菌組合、混合物及組成物及其用途 |
| AR120035A1 (es) * | 2019-09-23 | 2022-01-26 | Adama Makhteshim Ltd | Proceso para preparar 5-(fluoro-4-imino-3-metil)-1-tosil-3,4-dihidropirimidin-(1h)-ona y derivados del compuesto |
| WO2021181274A1 (en) * | 2020-03-09 | 2021-09-16 | Adama Makhteshim Ltd. | Process for preparing 5-fluoro-4-imino-3-methyl-1-(toluene-4-sulfonyl)-3,4-dihydro-1h-pyrimidin-2-one |
| BR112022022281A2 (pt) * | 2020-05-04 | 2023-01-03 | Adama Makhteshim Ltd | Misturas e composições compreendendo 5-fluoro-4-imino-3-metil- 1-tosil-3,4-dihidropirimidin-2-ona e métodos de uso das mesmas |
| EP4649827A2 (en) | 2020-07-08 | 2025-11-19 | Adama Makhteshim Ltd. | Fungicidal mixtures |
| CU20230035A7 (es) | 2021-01-27 | 2024-04-08 | Adama Makhteshim Ltd | 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2(1h)-ona para control de enfermedades de las plantas |
| BR112023023105A2 (pt) | 2021-05-04 | 2024-01-30 | Adama Makhteshim Ltd | Formas cristalinas de 5-fluoro-4-imino-3-metil-1-tosil-3,4-di-hidropirimidin-2-ona, e misturas, composições e métodos de uso das mesmas |
| WO2023042126A1 (en) | 2021-09-15 | 2023-03-23 | Adama Makhteshim Ltd. | Process for preparing 5-fluoro-4-imino-3-methyl-1-(toluene-4-sulfonyl)-3,4-dihydro-1h-pyrimidin-2-one |
| AR128692A1 (es) | 2022-03-03 | 2024-06-05 | Adama Makhteshim Ltd | Combinaciones, mezclas y composiciones fungicidas y usos de las mismas |
| EP4531570A1 (en) | 2022-05-26 | 2025-04-09 | Adama Makhteshim Ltd. | Fungicidal combinations, mixtures and compositions and uses thereof |
| UY40385A (es) | 2022-08-03 | 2024-02-15 | Adama Makhteshim Ltd | 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2(1h)-ona para hongos resistentes a fungicidas |
| AR132077A1 (es) | 2023-03-09 | 2025-05-21 | Adama Makhteshim Ltd | Combinaciones, mezclas y composiciones fungicidas y usos de las mismas |
| WO2024189563A1 (en) | 2023-03-14 | 2024-09-19 | Adama Makhteshim Ltd. | Liquid compositions containing 5-(fluoro-4-imino-3-methyl)-1-tosyl-3,4 dihydropyrimidine-(1h)-one and derivatives thereof and a uv absorber |
| AR132182A1 (es) * | 2023-03-23 | 2025-06-04 | Adama Makhteshim Ltd | Proceso para preparar 5-fluoro-4-imino-3-metil-1-(tolueno-4-sulfonil)-3,4-dihidro-1h-pirimidin-2-ona |
| AR133680A1 (es) | 2023-08-31 | 2025-10-22 | Adama Makhteshim Ltd | Combinaciones, mezclas y composiciones fungicidas y usos de las mismas |
| IL308593A (en) | 2023-11-15 | 2025-06-01 | Adama Makhteshim Ltd | Reducing environmental impact of fungicidal enhancement |
| WO2025114931A1 (en) | 2023-11-28 | 2025-06-05 | Adama Makhteshim Ltd. | Fungicidal combinations, mixtures and compositions and uses thereof |
| WO2025203024A1 (en) | 2024-03-26 | 2025-10-02 | Adama Makhteshim Ltd. | Process for preparing 5-fluoro-4-imino-3-methyl-1-(toluene-4-sulfonyl)-3,4-dihydro-1h-pyrimidin-2-one |
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| UA106889C2 (uk) | 2009-08-07 | 2014-10-27 | ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі | Похідні n1-ацил-5-фторпіримідинону |
| CN102548979B (zh) | 2009-08-07 | 2015-05-13 | 陶氏益农公司 | 5-氟代-2-氧代嘧啶-1(2h)-甲酸酯衍生物 |
| UA112284C2 (uk) * | 2009-08-07 | 2016-08-25 | ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі | Похідні 5-фторпіримідинону |
| RS53395B (sr) * | 2009-08-07 | 2014-10-31 | Dow Agrosciences Llc | Derivati n1-sulfonil-5-fluorpirimidinona |
| IN2012DN03094A (enExample) | 2009-10-07 | 2015-09-18 | Dow Agrosciences Llc | |
| UA108101C2 (xx) * | 2010-04-26 | 2015-03-25 | Похідні n3-заміщених n1-сульфоніл-5-фторпіримідинонів | |
| RS56609B1 (sr) * | 2011-08-17 | 2018-02-28 | Adama Makhteshim Ltd | 1-supstituisani derivati 5-fluor-3,6-dihidro-6-imino-2(1h)-pirimidinona kao fungicidna sredstva za upotrebu u proizvodnji bilja |
| EP2917952B1 (en) | 2012-11-07 | 2016-04-13 | Toyota Jidosha Kabushiki Kaisha | Method for producing a catalyst for fuel cells |
| KR20150103096A (ko) | 2012-12-28 | 2015-09-09 | 다우 아그로사이언시즈 엘엘씨 | N-(치환된)-5-플루오로-4-이미노-3-메틸-2-옥소-3,4-디히드로피리미딘-1(2h)-카르복실레이트 유도체 |
| RU2656101C2 (ru) * | 2012-12-28 | 2018-05-31 | Адама Мактешим Лтд. | Производные 1-(замещенный бензоил)-5-фтор-4-имино-3-метил-3,4-дигидропиримидин-2(1h)-она |
| US9321734B2 (en) | 2012-12-28 | 2016-04-26 | Dow Agrosciences Llc | N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1(2H)-carboxamide derivatives |
| US9642368B2 (en) * | 2012-12-31 | 2017-05-09 | Adama Makhteshim Ltd. | 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1H)-one derivatives as fungicides |
| AU2014373853A1 (en) | 2013-12-31 | 2016-08-11 | Adama Makhteshim Ltd. | Synergistic fungicidal mixtures and compositions for fungal control |
| MX392211B (es) | 2013-12-31 | 2025-03-21 | Adama Makhteshim Ltd | 5-flúor-4-imino-3-(alquil/alquilo sustituido)-1-(arilsulfonil)-3,4-dihidropirimidin-2(1h)-ona y los procesos para su preparación. |
| MA41272A (fr) | 2014-12-23 | 2017-10-31 | Adama Makhteshim Ltd | 5-fluoro-4-imino-3-(alkyle/alkyle substitué)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one en tant que traitement des semences |
-
2014
- 2014-12-29 MX MX2016008759A patent/MX392211B/es unknown
- 2014-12-29 WO PCT/US2014/072566 patent/WO2015103142A1/en not_active Ceased
- 2014-12-29 US US14/584,347 patent/US20150183749A1/en not_active Abandoned
- 2014-12-29 EP EP21151090.4A patent/EP3862346A1/en active Pending
- 2014-12-29 CR CR20210172A patent/CR20210172A/es unknown
- 2014-12-29 EP EP14877285.8A patent/EP3097096A4/en not_active Ceased
- 2014-12-29 JP JP2016543746A patent/JP6804297B2/ja active Active
- 2014-12-29 EA EA201691353A patent/EA201691353A1/ru unknown
- 2014-12-29 SG SG11201605372QA patent/SG11201605372QA/en unknown
- 2014-12-29 UA UAA201909738A patent/UA129860C2/uk unknown
- 2014-12-29 US US14/584,368 patent/US20150183750A1/en not_active Abandoned
- 2014-12-29 AU AU2014373959A patent/AU2014373959B2/en active Active
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