ECSP16064249A - 5-flúor-4-imino-3-(alquil/alquilo sustituido)-1-(arilsulfonil)-3,4-dihidropirimidin-2(1h)-ona y los procesos para su preparación - Google Patents

5-flúor-4-imino-3-(alquil/alquilo sustituido)-1-(arilsulfonil)-3,4-dihidropirimidin-2(1h)-ona y los procesos para su preparación

Info

Publication number
ECSP16064249A
ECSP16064249A ECIEPI201664249A ECPI201664249A ECSP16064249A EC SP16064249 A ECSP16064249 A EC SP16064249A EC IEPI201664249 A ECIEPI201664249 A EC IEPI201664249A EC PI201664249 A ECPI201664249 A EC PI201664249A EC SP16064249 A ECSP16064249 A EC SP16064249A
Authority
EC
Ecuador
Prior art keywords
alkyl
dihydropyrimidin
imino
processes
preparation
Prior art date
Application number
ECIEPI201664249A
Other languages
English (en)
Inventor
Nakyen Choy
Ross, Jr
Original Assignee
Adama Makhteshim Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Adama Makhteshim Ltd filed Critical Adama Makhteshim Ltd
Publication of ECSP16064249A publication Critical patent/ECSP16064249A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/08—Hydrogen atoms or radicals containing only hydrogen and carbon atoms
    • C07D333/10—Thiophene
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Environmental Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Health & Medical Sciences (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Detergent Compositions (AREA)
  • Cosmetics (AREA)

Abstract

Se proporcionan, en el presente documento, 5-flúor-4-imino-3- (alquil/alquilo sustituido)-1- (arilsulfonilo)-3,4-dihidropirimidin-2(1H)-ona y los procedimientos para su preparación, que pueden incluir el uso de un carbonato alcalino y un agente alquilante.
ECIEPI201664249A 2013-12-31 2016-07-29 5-flúor-4-imino-3-(alquil/alquilo sustituido)-1-(arilsulfonil)-3,4-dihidropirimidin-2(1h)-ona y los procesos para su preparación ECSP16064249A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201361922572P 2013-12-31 2013-12-31
US201361922582P 2013-12-31 2013-12-31

Publications (1)

Publication Number Publication Date
ECSP16064249A true ECSP16064249A (es) 2019-07-31

Family

ID=53480979

Family Applications (1)

Application Number Title Priority Date Filing Date
ECIEPI201664249A ECSP16064249A (es) 2013-12-31 2016-07-29 5-flúor-4-imino-3-(alquil/alquilo sustituido)-1-(arilsulfonil)-3,4-dihidropirimidin-2(1h)-ona y los procesos para su preparación

Country Status (24)

Country Link
US (8) US20150183749A1 (es)
EP (4) EP3097096A4 (es)
JP (3) JP6804297B2 (es)
CN (4) CN106061972B (es)
AP (1) AP2016009342A0 (es)
AU (2) AU2014373959B2 (es)
BR (2) BR102014033037B1 (es)
CA (2) CA2935601C (es)
CL (1) CL2016001677A1 (es)
CR (2) CR20160343A (es)
DO (1) DOP2016000163A (es)
EA (2) EA036389B1 (es)
EC (1) ECSP16064249A (es)
IL (3) IL246511B (es)
MX (2) MX2016008758A (es)
NI (1) NI201600094A (es)
NZ (2) NZ722438A (es)
PE (1) PE20161174A1 (es)
PH (1) PH12016501284A1 (es)
SG (2) SG11201605377VA (es)
TW (2) TWI667229B (es)
UA (1) UA122200C2 (es)
UY (2) UY35942A (es)
WO (2) WO2015103144A1 (es)

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PL2953463T3 (pl) 2012-12-31 2022-01-03 Adama Makhteshim Ltd. Pochodne 3-alkilo-5-fluoro-4-podstawione-imino-3,4-dihydropirymidyn-2(1h)-onu jako środki grzybobójcze
PE20161174A1 (es) 2013-12-31 2016-10-26 Adama Makhteshim Ltd 5-fluor-4-imino-3-(alquil/alquilo sustituido)-1-(arilsulfonil)-3,4-dihidropirimidin-2(1h)-ona y los procesos para su preparacion
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EP4003017A1 (en) 2019-07-22 2022-06-01 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof
EP4034529A1 (en) * 2019-09-23 2022-08-03 Adama Makhteshim Ltd. Process for preparing 5-(fluoro-4-imino-3-methyl)-1-tosyl-3,4 dihydropyrimidine -(1h)-one
CN115776980A (zh) * 2020-03-09 2023-03-10 阿达玛马克西姆有限公司 用于制备5-氟-4-亚氨基-3-甲基-1-(甲苯-4-磺酰基)-3,4-二氢-1h-嘧啶-2-酮的方法
UY39197A (es) 2020-05-04 2021-11-30 Adama Makhteshim Ltd Mezclas y composiciones que comprenden 5-fluoro-4-imino-3- metil-1-tosil-3,4-dihidropirimidin-2-ona, y métodos de uso de las mismas
IL299711A (en) 2020-07-08 2023-03-01 Adama Makhteshim Ltd Fungicide mixtures
CU20230035A7 (es) 2021-01-27 2024-04-08 Adama Makhteshim Ltd 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2(1h)-ona para control de enfermedades de las plantas
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WO2023228148A1 (en) 2022-05-26 2023-11-30 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof
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PE20161174A1 (es) 2013-12-31 2016-10-26 Adama Makhteshim Ltd 5-fluor-4-imino-3-(alquil/alquilo sustituido)-1-(arilsulfonil)-3,4-dihidropirimidin-2(1h)-ona y los procesos para su preparacion
AU2014373850A1 (en) 2013-12-31 2016-08-11 Adama Makhteshim Ltd. Synergistic fungicidal mixtures and compositions for fungal control
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US9850215B2 (en) 2017-12-26
AU2014373959B2 (en) 2017-10-26
NZ722438A (en) 2018-01-26
TWI667229B (zh) 2019-08-01
PH12016501284A1 (en) 2016-08-15
EP3862347A1 (en) 2021-08-11
CL2016001677A1 (es) 2016-12-09
MX2016008758A (es) 2017-05-09
EP3094632A4 (en) 2017-10-18
UA122200C2 (uk) 2020-10-12
US20190308941A1 (en) 2019-10-10
CR20210172A (es) 2021-05-11
NI201600094A (es) 2016-08-09
IL246512A0 (en) 2016-08-31
AU2014373961B2 (en) 2017-10-26
CA2935601C (en) 2023-03-14
NZ722439A (en) 2018-01-26
EA036389B1 (ru) 2020-11-03
WO2015103144A1 (en) 2015-07-09
US20200148649A1 (en) 2020-05-14
IL246511B (en) 2019-10-31
CA2935594A1 (en) 2015-07-09
EA201691353A1 (ru) 2016-12-30
US9840476B2 (en) 2017-12-12
CN106061972B (zh) 2020-01-17
US10919864B2 (en) 2021-02-16
TWI722979B (zh) 2021-04-01
EP3097096A1 (en) 2016-11-30
IL269694B (en) 2021-09-30
MX2016008759A (es) 2017-05-09
UY35942A (es) 2015-07-31
US20150183750A1 (en) 2015-07-02
CA2935601A1 (en) 2015-07-09
PE20161174A1 (es) 2016-10-26
US20160280662A1 (en) 2016-09-29
CA2935594C (en) 2022-05-03
CR20160343A (es) 2016-12-14
CN106061972A (zh) 2016-10-26
SG11201605377VA (en) 2016-08-30
US20180072686A1 (en) 2018-03-15
IL269694A (en) 2019-11-28
JP6585057B2 (ja) 2019-10-02
EA201691351A1 (ru) 2016-12-30
CN106068268A (zh) 2016-11-02
CN111362881A (zh) 2020-07-03
JP2017502963A (ja) 2017-01-26
BR102014033037A2 (pt) 2015-11-17
UY35943A (es) 2015-07-31
JP2019218396A (ja) 2019-12-26
WO2015103142A1 (en) 2015-07-09
CN111217759A (zh) 2020-06-02
EP3862346A1 (en) 2021-08-11
IL246511A0 (en) 2016-08-31
BR102014033037B1 (pt) 2021-07-13
IL246512B (en) 2019-09-26
AU2014373959A1 (en) 2016-08-11
BR102014033010B1 (pt) 2021-07-13
JP2017501197A (ja) 2017-01-12
US20150183749A1 (en) 2015-07-02
DOP2016000163A (es) 2016-09-30
TW201609669A (zh) 2016-03-16
SG11201605372QA (en) 2016-08-30
US20160280663A1 (en) 2016-09-29
EP3094632A1 (en) 2016-11-23
US20200024238A1 (en) 2020-01-23
BR102014033010A2 (pt) 2015-10-20
JP6804297B2 (ja) 2020-12-23
AU2014373961A1 (en) 2016-08-11
AP2016009342A0 (en) 2016-07-31
EP3097096A4 (en) 2017-10-11
TW201609670A (zh) 2016-03-16

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