CL2016001677A1 - 5-flúor-4-imino-3-(alquil/alquilo sustituido)-1-(arilsulfonil)-3,4-dihidropirimidin-2(1h)-ona y los procesos para su preparación. - Google Patents
5-flúor-4-imino-3-(alquil/alquilo sustituido)-1-(arilsulfonil)-3,4-dihidropirimidin-2(1h)-ona y los procesos para su preparación.Info
- Publication number
- CL2016001677A1 CL2016001677A1 CL2016001677A CL2016001677A CL2016001677A1 CL 2016001677 A1 CL2016001677 A1 CL 2016001677A1 CL 2016001677 A CL2016001677 A CL 2016001677A CL 2016001677 A CL2016001677 A CL 2016001677A CL 2016001677 A1 CL2016001677 A1 CL 2016001677A1
- Authority
- CL
- Chile
- Prior art keywords
- alkyl
- imino
- dihydropyrimidin
- arylsulfonyl
- fluoro
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 2
- 125000000217 alkyl group Chemical group 0.000 title 1
- 125000004391 aryl sulfonyl group Chemical group 0.000 title 1
- 125000000547 substituted alkyl group Chemical group 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
- C07D333/08—Hydrogen atoms or radicals containing only hydrogen and carbon atoms
- C07D333/10—Thiophene
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Wood Science & Technology (AREA)
- Environmental Sciences (AREA)
- Plant Pathology (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- General Health & Medical Sciences (AREA)
- Agronomy & Crop Science (AREA)
- Zoology (AREA)
- Pest Control & Pesticides (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Detergent Compositions (AREA)
- Cosmetics (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201361922582P | 2013-12-31 | 2013-12-31 | |
| US201361922572P | 2013-12-31 | 2013-12-31 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CL2016001677A1 true CL2016001677A1 (es) | 2016-12-09 |
Family
ID=53480979
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CL2016001677A CL2016001677A1 (es) | 2013-12-31 | 2016-06-29 | 5-flúor-4-imino-3-(alquil/alquilo sustituido)-1-(arilsulfonil)-3,4-dihidropirimidin-2(1h)-ona y los procesos para su preparación. |
Country Status (24)
| Country | Link |
|---|---|
| US (8) | US20150183749A1 (enExample) |
| EP (4) | EP3097096A4 (enExample) |
| JP (3) | JP6585057B2 (enExample) |
| CN (4) | CN106061972B (enExample) |
| AP (1) | AP2016009342A0 (enExample) |
| AU (2) | AU2014373961B2 (enExample) |
| BR (2) | BR102014033010B1 (enExample) |
| CA (2) | CA2935594C (enExample) |
| CL (1) | CL2016001677A1 (enExample) |
| CR (2) | CR20210172A (enExample) |
| DO (1) | DOP2016000163A (enExample) |
| EA (2) | EA201691353A1 (enExample) |
| EC (1) | ECSP16064249A (enExample) |
| IL (3) | IL246512B (enExample) |
| MX (2) | MX375727B (enExample) |
| NI (1) | NI201600094A (enExample) |
| NZ (2) | NZ722439A (enExample) |
| PE (1) | PE20161174A1 (enExample) |
| PH (1) | PH12016501284A1 (enExample) |
| SG (2) | SG11201605377VA (enExample) |
| TW (2) | TWI667229B (enExample) |
| UA (2) | UA122200C2 (enExample) |
| UY (2) | UY35942A (enExample) |
| WO (2) | WO2015103144A1 (enExample) |
Families Citing this family (27)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN110003118A (zh) | 2012-12-28 | 2019-07-12 | 阿达玛马克西姆股份有限公司 | 制备羧酸酯衍生物的方法 |
| AU2013370490B2 (en) | 2012-12-28 | 2018-05-10 | Adama Makhteshim Ltd. | N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1 (2H)-carboxamide derivatives |
| KR102309245B1 (ko) | 2012-12-31 | 2021-10-06 | 아다마 마켓심 리미티드 | 살진균제로서의 3-알킬-5-플루오로-4-치환된-이미노-3,4-디히드로피리미딘-2(1h)-온 유도체 |
| JP6585057B2 (ja) | 2013-12-31 | 2019-10-02 | アダマ・マクテシム・リミテッド | ５−フルオロ−４−イミノ−３−（アルキル／置換アルキル）−１−（アリールスルホニル）−３，４−ジヒドロピリミジン−２（１ｈ）−オンおよびそれらの調製方法 |
| EA030056B1 (ru) | 2013-12-31 | 2018-06-29 | Адама Мактешим Лтд. | Синергетические фунгицидные смеси и синергетические фунгицидные композиции для борьбы с грибами |
| UY36964A (es) | 2015-10-27 | 2017-05-31 | Bayer Cropscience Ag | Combinaciones de principios activos que comprenden un derivado de (tio) carboxamida y un compuesto funguicida |
| JP6922271B2 (ja) * | 2016-03-11 | 2021-08-18 | 住友化学株式会社 | 植物病害防除組成物及び植物病害防除方法 |
| EP3655396A1 (en) * | 2017-07-17 | 2020-05-27 | Adama Makhteshim Ltd. | Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one |
| IL282939B2 (en) * | 2018-11-05 | 2024-10-01 | Adama Makhteshim Ltd | Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4- dihydropyrimidin-2-one, and methods of use thereof |
| EP4003017A1 (en) | 2019-07-22 | 2022-06-01 | Adama Makhteshim Ltd. | Fungicidal combinations, mixtures and compositions and uses thereof |
| BR112022005464A2 (pt) | 2019-09-23 | 2022-08-16 | Adama Makhteshim Ltd | Processo para a preparação de 5-(flúor-4-imino-3-metil)-1-tosil-3,4-diidropirimidina-(1h)-ona |
| CN115776980A (zh) * | 2020-03-09 | 2023-03-10 | 阿达玛马克西姆有限公司 | 用于制备5-氟-4-亚氨基-3-甲基-1-(甲苯-4-磺酰基)-3,4-二氢-1h-嘧啶-2-酮的方法 |
| AU2021267206A1 (en) | 2020-05-04 | 2022-12-08 | Adama Makhteshim Ltd. | Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof |
| AU2021306905A1 (en) | 2020-07-08 | 2023-02-23 | Adama Makhteshim Ltd. | Fungicidal mixtures |
| PE20250069A1 (es) | 2021-01-27 | 2025-01-13 | Adama Makhteshim Ltd | 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2(1h)-ona para control de enfermedades de plantas |
| CA3216622A1 (en) | 2021-05-04 | 2022-11-10 | Stefano Luca Giaffreda | Crystalline forms of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4- dihydropyrimidin-2-one, and mixtures, compositions and methods of use thereof |
| CN118139845A (zh) | 2021-09-15 | 2024-06-04 | 安道麦马克西姆有限公司 | 用于制备5-氟-4-亚氨基-3-甲基-1-(甲苯-4-磺酰基)-3,4-二氢-1h-嘧啶-2-酮的方法 |
| EP4486126A1 (en) | 2022-03-03 | 2025-01-08 | Adama Makhteshim Ltd. | Fungicidal combinations, mixtures and compositions and uses thereof |
| US20250338845A1 (en) | 2022-05-26 | 2025-11-06 | Adama Makhteshim Ltd. | Fungicidal combinations, mixtures and compositions and uses thereof |
| AU2023318916A1 (en) | 2022-08-03 | 2025-02-20 | Adama Makhteshim Ltd. | 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2(1h)-one for fungicide-resistant fungus |
| WO2024184859A1 (en) | 2023-03-09 | 2024-09-12 | Conese Salvatore | Fungicidal combinations, mixtures and compositions and uses thereof |
| AU2024236967A1 (en) | 2023-03-14 | 2025-09-25 | Adama Makhteshim Ltd. | Liquid compositions containing 5-(fluoro-4-imino-3-methyl)-1-tosyl-3,4 dihydropyrimidine-(1h)-one and derivatives thereof and a uv absorber |
| AR132182A1 (es) | 2023-03-23 | 2025-06-04 | Adama Makhteshim Ltd | Proceso para preparar 5-fluoro-4-imino-3-metil-1-(tolueno-4-sulfonil)-3,4-dihidro-1h-pirimidin-2-ona |
| AR133680A1 (es) | 2023-08-31 | 2025-10-22 | Adama Makhteshim Ltd | Combinaciones, mezclas y composiciones fungicidas y usos de las mismas |
| IL308593A (en) | 2023-11-15 | 2025-06-01 | Adama Makhteshim Ltd | Reducing environmental impact of fungicidal enhancement |
| WO2025114931A1 (en) | 2023-11-28 | 2025-06-05 | Adama Makhteshim Ltd. | Fungicidal combinations, mixtures and compositions and uses thereof |
| WO2025203024A1 (en) | 2024-03-26 | 2025-10-02 | Adama Makhteshim Ltd. | Process for preparing 5-fluoro-4-imino-3-methyl-1-(toluene-4-sulfonyl)-3,4-dihydro-1h-pyrimidin-2-one |
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| AU2013370490B2 (en) | 2012-12-28 | 2018-05-10 | Adama Makhteshim Ltd. | N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1 (2H)-carboxamide derivatives |
| KR102309245B1 (ko) * | 2012-12-31 | 2021-10-06 | 아다마 마켓심 리미티드 | 살진균제로서의 3-알킬-5-플루오로-4-치환된-이미노-3,4-디히드로피리미딘-2(1h)-온 유도체 |
| EA030056B1 (ru) | 2013-12-31 | 2018-06-29 | Адама Мактешим Лтд. | Синергетические фунгицидные смеси и синергетические фунгицидные композиции для борьбы с грибами |
| JP6585057B2 (ja) | 2013-12-31 | 2019-10-02 | アダマ・マクテシム・リミテッド | ５−フルオロ−４−イミノ−３−（アルキル／置換アルキル）−１−（アリールスルホニル）−３，４−ジヒドロピリミジン−２（１ｈ）−オンおよびそれらの調製方法 |
| MA41272A (fr) | 2014-12-23 | 2017-10-31 | Adama Makhteshim Ltd | 5-fluoro-4-imino-3-(alkyle/alkyle substitué)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one en tant que traitement des semences |
-
2014
- 2014-12-29 JP JP2016543735A patent/JP6585057B2/ja active Active
- 2014-12-29 EP EP14877285.8A patent/EP3097096A4/en not_active Ceased
- 2014-12-29 EA EA201691353A patent/EA201691353A1/ru unknown
- 2014-12-29 SG SG11201605377VA patent/SG11201605377VA/en unknown
- 2014-12-29 UA UAA201608339A patent/UA122200C2/uk unknown
- 2014-12-29 CR CR20210172A patent/CR20210172A/es unknown
- 2014-12-29 CN CN201480076583.4A patent/CN106061972B/zh active Active
- 2014-12-29 CN CN201480076563.7A patent/CN106068268A/zh active Pending
- 2014-12-29 CN CN201911357017.1A patent/CN111362881A/zh active Pending
- 2014-12-29 JP JP2016543746A patent/JP6804297B2/ja active Active
- 2014-12-29 CA CA2935594A patent/CA2935594C/en active Active
- 2014-12-29 MX MX2016008758A patent/MX375727B/es active IP Right Grant
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