JP6022442B2 - 男性用避妊組成物および使用方法 - Google Patents

男性用避妊組成物および使用方法 Download PDF

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Publication number
JP6022442B2
JP6022442B2 JP2013510361A JP2013510361A JP6022442B2 JP 6022442 B2 JP6022442 B2 JP 6022442B2 JP 2013510361 A JP2013510361 A JP 2013510361A JP 2013510361 A JP2013510361 A JP 2013510361A JP 6022442 B2 JP6022442 B2 JP 6022442B2
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Prior art keywords
compound
pharmaceutical composition
salt
brdt
sperm
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Expired - Fee Related
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JP2013510361A
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English (en)
Japanese (ja)
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JP2013528600A5 (enExample
JP2013528600A (ja
Inventor
ブラドナー，ジェームズ，エリオット
マツック，マーティン
チー，チュン
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Baylor College of Medicine
Dana Farber Cancer Institute Inc
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Baylor College of Medicine
Dana Farber Cancer Institute Inc
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • A61K31/5513—1,4-Benzodiazepines, e.g. diazepam or clozapine
    • A61K31/5517—1,4-Benzodiazepines, e.g. diazepam or clozapine condensed with five-membered rings having nitrogen as a ring hetero atom, e.g. imidazobenzodiazepines, triazolam
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/16—Masculine contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D495/14—Ortho-condensed systems

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicinal Preparation (AREA)
JP2013510361A 2010-05-14 2011-05-16 男性用避妊組成物および使用方法 Expired - Fee Related JP6022442B2 (ja)

Applications Claiming Priority (11)

Application Number Priority Date Filing Date Title
US33499110P 2010-05-14 2010-05-14
US61/334,991 2010-05-14
US37074510P 2010-08-04 2010-08-04
US61/370,745 2010-08-04
US37586310P 2010-08-22 2010-08-22
US61/375,863 2010-08-22
US201161467299P 2011-03-24 2011-03-24
US201161467376P 2011-03-24 2011-03-24
US61/467,299 2011-03-24
US61/467,376 2011-03-24
PCT/US2011/036667 WO2011143657A1 (en) 2010-05-14 2011-05-16 Male contraceptive compositions and methods of use

Publications (3)

Publication Number Publication Date
JP2013528600A JP2013528600A (ja) 2013-07-11
JP2013528600A5 JP2013528600A5 (enExample) 2014-07-03
JP6022442B2 true JP6022442B2 (ja) 2016-11-09

Family

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JP2013510361A Expired - Fee Related JP6022442B2 (ja) 2010-05-14 2011-05-16 男性用避妊組成物および使用方法

Country Status (6)

Country Link
US (2) US9301962B2 (enExample)
EP (1) EP2571875A4 (enExample)
JP (1) JP6022442B2 (enExample)
CN (1) CN103180318B (enExample)
CA (1) CA2799381A1 (enExample)
WO (1) WO2011143657A1 (enExample)

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US9789120B2 (en) 2017-10-17
US20130210813A1 (en) 2013-08-15
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US9301962B2 (en) 2016-04-05
CA2799381A1 (en) 2011-11-17
JP2013528600A (ja) 2013-07-11

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