JP5705748B2 - Ｃｂ２受容体を変調する複素環化合物 - Google Patents

Ｃｂ２受容体を変調する複素環化合物 Download PDF

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JP5705748B2
JP5705748B2 JP2011551161A JP2011551161A JP5705748B2 JP 5705748 B2 JP5705748 B2 JP 5705748B2 JP 2011551161 A JP2011551161 A JP 2011551161A JP 2011551161 A JP2011551161 A JP 2011551161A JP 5705748 B2 JP5705748 B2 JP 5705748B2
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alkyl
carboxylic acid
tert
mmol
butyl
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JP2012518038A5 (https=
JP2012518038A (ja
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アレサンドラ バルトロッツィ
アレサンドラ バルトロッツィ
アンジェラ ベリー
アンジェラ ベリー
ピエール フランチェスコ チリロ
ピエール フランチェスコ チリロ
ユージーン リチャード ヒッキー
ユージーン リチャード ヒッキー
ドリス リーター
ドリス リーター
リーフェン ウー
リーフェン ウー
ルネ エム ジンデル
ルネ エム ジンデル
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ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング
ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング
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    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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  • Health & Medical Sciences (AREA)
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  • Chemical & Material Sciences (AREA)
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  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
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  • Veterinary Medicine (AREA)
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  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Immunology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Pulmonology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Diabetes (AREA)
  • Urology & Nephrology (AREA)
  • Hospice & Palliative Care (AREA)
  • Dermatology (AREA)
  • Otolaryngology (AREA)
  • Vascular Medicine (AREA)
  • Transplantation (AREA)
  • Psychiatry (AREA)
  • Hematology (AREA)
  • Rheumatology (AREA)
  • Endocrinology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
JP2011551161A 2009-02-18 2010-02-16 Ｃｂ２受容体を変調する複素環化合物 Active JP5705748B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US15333309P 2009-02-18 2009-02-18
US61/153,333 2009-02-18
PCT/US2010/024270 WO2010096371A2 (en) 2009-02-18 2010-02-16 Heterocyclic compounds which modulate the cb2 receptor

Publications (3)

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JP2012518038A JP2012518038A (ja) 2012-08-09
JP2012518038A5 JP2012518038A5 (https=) 2014-09-18
JP5705748B2 true JP5705748B2 (ja) 2015-04-22

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US (1) US8889670B2 (https=)
EP (1) EP2398771B1 (https=)
JP (1) JP5705748B2 (https=)
WO (1) WO2010096371A2 (https=)

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WO2008048914A1 (en) 2006-10-17 2008-04-24 Boehringer Ingelheim International Gmbh Polycyclic compounds which modulate the cb2 receptor
WO2008064054A2 (en) 2006-11-21 2008-05-29 Boehringer Ingelheim International Gmbh Compounds which modulate the cb2 receptor
JP5492092B2 (ja) * 2007-11-07 2014-05-14 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Ｃｂ２受容体を調節する化合物
EP2265585B1 (en) 2008-02-21 2014-09-17 Boehringer Ingelheim International GmbH Amine and ether compounds which modulate the cb2 receptor
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US8629157B2 (en) 2009-01-05 2014-01-14 Boehringer Ingelheim International Gmbh Pyrrolidine compounds which modulate the CB2 receptor
WO2010096371A2 (en) 2009-02-18 2010-08-26 Boehringer Ingelheim International Gmbh Heterocyclic compounds which modulate the cb2 receptor
US8299103B2 (en) 2009-06-15 2012-10-30 Boehringer Ingelheim International Gmbh Compounds which selectively modulate the CB2 receptor
JP5756800B2 (ja) 2009-06-16 2015-07-29 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Ｃｂ２受容体を調節するアゼチジン２−カルボキサミド誘導体
JP2013505295A (ja) 2009-09-22 2013-02-14 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Ｃｂ２受容体を選択的に調節する化合物
US9315454B2 (en) 2010-01-15 2016-04-19 Boehringer Ingelheim International Gmbh Compounds which modulate the CB2 receptor
EP2542539B1 (en) 2010-03-05 2014-02-26 Boehringer Ingelheim International GmbH Tetrazole compounds which selectively modulate the cb2 receptor
JP5746764B2 (ja) 2010-07-22 2015-07-08 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Ｃｂ２受容体を調節する化合物
WO2012090179A2 (en) 2010-12-30 2012-07-05 Lupin Limited Isoquinoline derivatives as cannabinoid receptor modulators
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JP6223563B2 (ja) 2013-10-14 2017-11-01 エーザイ・アール・アンド・ディー・マネジメント株式会社 選択的に置換されたキノリン化合物
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