JP5705748B2 - Ｃｂ２受容体を変調する複素環化合物 - Google Patents

Ｃｂ２受容体を変調する複素環化合物 Download PDF

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JP5705748B2
JP5705748B2 JP2011551161A JP2011551161A JP5705748B2 JP 5705748 B2 JP5705748 B2 JP 5705748B2 JP 2011551161 A JP2011551161 A JP 2011551161A JP 2011551161 A JP2011551161 A JP 2011551161A JP 5705748 B2 JP5705748 B2 JP 5705748B2
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alkyl
carboxylic acid
tert
mmol
butyl
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JP2012518038A5 (enExample
JP2012518038A (ja
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アレサンドラ バルトロッツィ
アレサンドラ バルトロッツィ
アンジェラ ベリー
アンジェラ ベリー
ピエール フランチェスコ チリロ
ピエール フランチェスコ チリロ
ユージーン リチャード ヒッキー
ユージーン リチャード ヒッキー
ドリス リーター
ドリス リーター
リーフェン ウー
リーフェン ウー
ルネ エム ジンデル
ルネ エム ジンデル
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ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング
ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング
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    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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  • Health & Medical Sciences (AREA)
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  • Animal Behavior & Ethology (AREA)
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  • General Chemical & Material Sciences (AREA)
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  • Immunology (AREA)
  • Biomedical Technology (AREA)
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  • Neurology (AREA)
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  • Heart & Thoracic Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Diabetes (AREA)
  • Urology & Nephrology (AREA)
  • Hospice & Palliative Care (AREA)
  • Dermatology (AREA)
  • Otolaryngology (AREA)
  • Vascular Medicine (AREA)
  • Transplantation (AREA)
  • Psychiatry (AREA)
  • Hematology (AREA)
  • Rheumatology (AREA)
  • Endocrinology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
JP2011551161A 2009-02-18 2010-02-16 Ｃｂ２受容体を変調する複素環化合物 Active JP5705748B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US15333309P 2009-02-18 2009-02-18
US61/153,333 2009-02-18
PCT/US2010/024270 WO2010096371A2 (en) 2009-02-18 2010-02-16 Heterocyclic compounds which modulate the cb2 receptor

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JP2012518038A JP2012518038A (ja) 2012-08-09
JP2012518038A5 JP2012518038A5 (enExample) 2014-09-18
JP5705748B2 true JP5705748B2 (ja) 2015-04-22

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US (1) US8889670B2 (enExample)
EP (1) EP2398771B1 (enExample)
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WO (1) WO2010096371A2 (enExample)

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EP2326629B1 (en) * 2008-07-10 2013-10-02 Boehringer Ingelheim International GmbH Sulfone compounds which modulate the cb2 receptor
NZ591111A (en) 2008-09-25 2013-08-30 Boehringer Ingelheim Int Sulfonyl compounds which selectively modulate the cb2 receptor
US8629157B2 (en) 2009-01-05 2014-01-14 Boehringer Ingelheim International Gmbh Pyrrolidine compounds which modulate the CB2 receptor
WO2010096371A2 (en) 2009-02-18 2010-08-26 Boehringer Ingelheim International Gmbh Heterocyclic compounds which modulate the cb2 receptor
US8299103B2 (en) 2009-06-15 2012-10-30 Boehringer Ingelheim International Gmbh Compounds which selectively modulate the CB2 receptor
US8383615B2 (en) 2009-06-16 2013-02-26 Boehringer Ingelheim International Gmbh Azetidine 2-carboxamide derivatives which modulate the CB2 receptor
EP2480544A1 (en) 2009-09-22 2012-08-01 Boehringer Ingelheim International GmbH Compounds which selectively modulate the cb2 receptor
EP2523936A1 (en) 2010-01-15 2012-11-21 Boehringer Ingelheim International GmbH Compounds which modulate the cb2 receptor
WO2011109324A1 (en) 2010-03-05 2011-09-09 Boehringer Ingelheim International Gmbh Tetrazole compounds which selectively modulate the cb2 receptor
JP5746764B2 (ja) 2010-07-22 2015-07-08 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Ｃｂ２受容体を調節する化合物
WO2012090177A2 (en) 2010-12-30 2012-07-05 Lupin Limited Cannabinoid receptor modulators
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JPWO2013147161A1 (ja) 2012-03-29 2015-12-14 東レ株式会社 ニペコチン酸誘導体及びその医薬用途
EP2803668A1 (en) 2013-05-17 2014-11-19 Boehringer Ingelheim International Gmbh Novel (cyano-dimethyl-methyl)-isoxazoles and -[1,3,4]thiadiazoles
MX363708B (es) 2013-10-14 2019-03-29 Eisai R&D Man Co Ltd Compuestos de quinolina selectivamente sustituidos.
SG10201704327RA (en) 2013-10-14 2017-06-29 Eisai R&D Man Co Ltd Selectively substituted quinoline compounds
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TWI691486B (zh) 2016-01-29 2020-04-21 日商東麗股份有限公司 環狀胺衍生物及其醫藥用途
CN108218846A (zh) * 2016-12-22 2018-06-29 四川海思科制药有限公司 噻吩衍生物的新固态形式及其制备方法和用途
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