JP5690823B2 - Ｊａｋ受容体およびタンパク質チロシンキナーゼ阻害薬としての複素環化合物 - Google Patents

Ｊａｋ受容体およびタンパク質チロシンキナーゼ阻害薬としての複素環化合物 Download PDF

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JP5690823B2
JP5690823B2 JP2012518753A JP2012518753A JP5690823B2 JP 5690823 B2 JP5690823 B2 JP 5690823B2 JP 2012518753 A JP2012518753 A JP 2012518753A JP 2012518753 A JP2012518753 A JP 2012518753A JP 5690823 B2 JP5690823 B2 JP 5690823B2
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pyrrolo
pyrimidin
diazaspiro
oct
octane
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JP2012532152A (ja
JP2012532152A5 (enExample
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シモン・フェルドベク・ニルセン
ダニエル・ロドリゲス・グレーヴェ
カルステン・リッテルスゴー
グンナー・グルエ−セレンセン
エリック・リッター・オットセン
ティナ・ダーレルプ・ポウルセン
セレン・クリスティアン・ショウ
アンソニー・マーレイ
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Leo Pharma AS
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    • C07—ORGANIC CHEMISTRY
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    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • C07D—HETEROCYCLIC COMPOUNDS
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  • Animal Behavior & Ethology (AREA)
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  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Dermatology (AREA)
  • Diabetes (AREA)
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  • Hematology (AREA)
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  • Rheumatology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Obesity (AREA)
  • Endocrinology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Ophthalmology & Optometry (AREA)
  • Hospice & Palliative Care (AREA)
  • Oncology (AREA)
  • Transplantation (AREA)
  • Emergency Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
JP2012518753A 2009-07-08 2010-07-08 Ｊａｋ受容体およびタンパク質チロシンキナーゼ阻害薬としての複素環化合物 Expired - Fee Related JP5690823B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US22394309P 2009-07-08 2009-07-08
US61/223,943 2009-07-08
PCT/DK2010/000105 WO2011003418A1 (en) 2009-07-08 2010-07-08 Heterocyclic compounds as jak receptor and protein tyrosine kinase inhibitors

Publications (3)

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JP2012532152A JP2012532152A (ja) 2012-12-13
JP2012532152A5 JP2012532152A5 (enExample) 2013-08-22
JP5690823B2 true JP5690823B2 (ja) 2015-03-25

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US (1) US9346809B2 (enExample)
EP (1) EP2451813B1 (enExample)
JP (1) JP5690823B2 (enExample)
CN (1) CN102574857B (enExample)
AR (1) AR077465A1 (enExample)
BR (1) BR112012000422A2 (enExample)
CA (1) CA2767079A1 (enExample)
TW (1) TW201105674A (enExample)
WO (1) WO2011003418A1 (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2014501772A (ja) * 2011-01-07 2014-01-23 レオ ファーマ アクティーゼルスカブ タンパク質チロシンキナーゼ阻害薬としての新規スルファミドピペラジン誘導体およびその医薬用途

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