JP5662325B2 - アザインドール誘導体 - Google Patents
アザインドール誘導体 Download PDFInfo
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- JP5662325B2 JP5662325B2 JP2011532512A JP2011532512A JP5662325B2 JP 5662325 B2 JP5662325 B2 JP 5662325B2 JP 2011532512 A JP2011532512 A JP 2011532512A JP 2011532512 A JP2011532512 A JP 2011532512A JP 5662325 B2 JP5662325 B2 JP 5662325B2
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- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
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- C07D—HETEROCYCLIC COMPOUNDS
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Landscapes
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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| DE102008052943.5 | 2008-10-23 | ||
| PCT/EP2009/006911 WO2010046013A1 (de) | 2008-10-23 | 2009-09-24 | Azaindolderivate |
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| GB201217285D0 (en) * | 2012-09-27 | 2012-11-14 | Univ Central Lancashire | Indole derivatives |
| US9227976B2 (en) | 2012-10-25 | 2016-01-05 | Usher Iii Initiative, Inc. | Pyrazolopyridazines and methods for treating retinal-degenerative diseases and hearing loss associated with usher syndrome |
| EP2968282B1 (en) * | 2013-03-12 | 2018-05-09 | Celgene Quanticel Research, Inc. | Histone dementhylase inhibitors |
| US9499551B2 (en) | 2014-01-24 | 2016-11-22 | Confluence Life Sciences, Inc. | Substituted pyrrolo[2,3-b]pyridines for treating cancer or inflammatory diseases |
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| CA2994917A1 (en) | 2015-08-10 | 2017-02-16 | Pfizer Inc. | 3-indol substituted derivatives, pharmaceutical compositions and methods for use |
| US10590079B2 (en) * | 2016-03-01 | 2020-03-17 | Novartis Ag | Cyano-substituted indoles as LSD1 inhibitors |
| US10513509B2 (en) * | 2016-05-26 | 2019-12-24 | Recurium Ip Holdings, Llc | EGFR inhibitor compounds |
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| WO2018210660A1 (en) | 2017-05-15 | 2018-11-22 | Basf Se | Heteroaryl compounds as agrochemical fungicides |
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| KR102513463B1 (ko) * | 2020-11-26 | 2023-03-29 | 주식회사 에스앤케이테라퓨틱스 | 엔도솜 톨-유사 수용체를 제어하는 신규 소분자 화합물 및 이를 이용한 자가면역질환 치료제 |
| CN116332940B (zh) * | 2023-02-14 | 2024-09-13 | 广西民族大学 | 一种7-脱氮嘌呤衍生物及其制备方法和应用 |
| WO2024245193A1 (zh) * | 2023-05-26 | 2024-12-05 | 上海艾力斯医药科技股份有限公司 | 杂芳环类化合物、其药物组合物及其应用 |
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| GB9900334D0 (en) | 1999-01-07 | 1999-02-24 | Angiogene Pharm Ltd | Tricylic vascular damaging agents |
| GB9900752D0 (en) | 1999-01-15 | 1999-03-03 | Angiogene Pharm Ltd | Benzimidazole vascular damaging agents |
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| CN1713910A (zh) | 2002-10-09 | 2005-12-28 | 西奥斯股份有限公司 | 作为p38激酶抑制剂的氮杂吲哚衍生物 |
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| GB0708141D0 (en) * | 2007-04-26 | 2007-06-06 | Syngenta Participations Ag | Improvements in or relating to organic compounds |
-
2008
- 2008-10-23 DE DE102008052943A patent/DE102008052943A1/de not_active Withdrawn
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2009
- 2009-09-24 US US13/125,816 patent/US20110207732A1/en not_active Abandoned
- 2009-09-24 CA CA2741428A patent/CA2741428C/en not_active Expired - Fee Related
- 2009-09-24 ES ES09778705.5T patent/ES2559427T3/es active Active
- 2009-09-24 EP EP09778705.5A patent/EP2342202B1/de not_active Not-in-force
- 2009-09-24 WO PCT/EP2009/006911 patent/WO2010046013A1/de not_active Ceased
- 2009-09-24 JP JP2011532512A patent/JP5662325B2/ja not_active Expired - Fee Related
- 2009-09-24 AU AU2009306795A patent/AU2009306795B2/en not_active Ceased
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2011
- 2011-04-12 IL IL212285A patent/IL212285A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CA2741428C (en) | 2017-05-09 |
| IL212285A0 (en) | 2011-06-30 |
| EP2342202A1 (de) | 2011-07-13 |
| AU2009306795B2 (en) | 2015-07-16 |
| AU2009306795A1 (en) | 2010-04-29 |
| JP2012506389A (ja) | 2012-03-15 |
| CA2741428A1 (en) | 2010-04-29 |
| ES2559427T3 (es) | 2016-02-12 |
| DE102008052943A1 (de) | 2010-04-29 |
| WO2010046013A1 (de) | 2010-04-29 |
| EP2342202B1 (de) | 2015-11-11 |
| US20110207732A1 (en) | 2011-08-25 |
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